DK153795C - Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte - Google Patents

Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte

Info

Publication number
DK153795C
DK153795C DK087783A DK87783A DK153795C DK 153795 C DK153795 C DK 153795C DK 087783 A DK087783 A DK 087783A DK 87783 A DK87783 A DK 87783A DK 153795 C DK153795 C DK 153795C
Authority
DK
Denmark
Prior art keywords
tylosin
deoxo
analogue
preparation
acceptable salts
Prior art date
Application number
DK087783A
Other languages
Danish (da)
English (en)
Other versions
DK153795B (da
DK87783D0 (da
DK87783A (da
Inventor
Satoshi Omura
Akira Nakagawa
Original Assignee
Satoshi Omura
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Satoshi Omura filed Critical Satoshi Omura
Publication of DK87783D0 publication Critical patent/DK87783D0/da
Publication of DK87783A publication Critical patent/DK87783A/da
Publication of DK153795B publication Critical patent/DK153795B/da
Application granted granted Critical
Publication of DK153795C publication Critical patent/DK153795C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK087783A 1982-02-25 1983-02-24 Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte DK153795C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2948082 1982-02-25
JP57029480A JPS58146595A (ja) 1982-02-25 1982-02-25 マクロライド系抗生物質

Publications (4)

Publication Number Publication Date
DK87783D0 DK87783D0 (da) 1983-02-24
DK87783A DK87783A (da) 1983-08-26
DK153795B DK153795B (da) 1988-09-05
DK153795C true DK153795C (da) 1989-01-23

Family

ID=12277244

Family Applications (1)

Application Number Title Priority Date Filing Date
DK087783A DK153795C (da) 1982-02-25 1983-02-24 Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte

Country Status (24)

Country Link
US (1) US4440759A (fr)
EP (1) EP0087921B1 (fr)
JP (1) JPS58146595A (fr)
KR (1) KR850000962B1 (fr)
AT (1) ATE16008T1 (fr)
AU (1) AU555979B2 (fr)
CA (1) CA1202022A (fr)
CS (1) CS235309B2 (fr)
DD (1) DD210283A5 (fr)
DE (1) DE3360951D1 (fr)
DK (1) DK153795C (fr)
ES (2) ES8403926A1 (fr)
FI (1) FI72322C (fr)
GB (1) GB2115813B (fr)
GR (1) GR78112B (fr)
HU (1) HU194269B (fr)
IL (1) IL67973A0 (fr)
NZ (1) NZ203365A (fr)
PH (1) PH18435A (fr)
PL (1) PL138759B1 (fr)
PT (1) PT76272B (fr)
RO (1) RO85833B (fr)
SU (1) SU1360588A3 (fr)
ZA (1) ZA831206B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820695A (en) * 1982-09-13 1989-04-11 Eli Lilly And Company C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
IL69666A (en) * 1982-09-13 1987-10-20 Lilly Co Eli 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
ZA841277B (en) * 1983-02-28 1985-09-25 Lilly Co Eli C-20-and c-23-modified macrolide derivatives
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
US4801721A (en) * 1984-08-16 1989-01-31 Ryan James W Stereospecific synthesis of carboxyalkyl peptides
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW309505B (fr) * 1993-03-31 1997-07-01 Toto Ltd
WO1996009312A1 (fr) * 1994-09-22 1996-03-28 Pfizer Inc. Macrolides antibiotiques
EP0778283A3 (fr) * 1995-12-05 1998-01-28 Pfizer Inc. Macrolides antibiotiques
CN110590885A (zh) * 2019-09-30 2019-12-20 郑州大学 20-取代-5-o-碳霉胺糖基-泰乐内酯衍生物
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178341A (en) * 1960-06-27 1965-04-13 Lilly Co Eli Antibiotics tylosin and desmycosin and derivatives thereof
GB1587685A (en) * 1977-03-09 1981-04-08 Microbial Chem Res Found Macrolactone derivatives and their production
JPS53132584A (en) * 1977-04-26 1978-11-18 Toyo Jozo Co Ltd 18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents

Also Published As

Publication number Publication date
AU555979B2 (en) 1986-10-16
ES520037A0 (es) 1984-04-01
US4440759A (en) 1984-04-03
DK153795B (da) 1988-09-05
RO85833B (ro) 1984-11-30
KR850000962B1 (ko) 1985-07-02
FI72322B (fi) 1987-01-30
FI830585L (fi) 1983-08-26
GB2115813A (en) 1983-09-14
DE3360951D1 (en) 1985-11-14
CA1202022A (fr) 1986-03-18
DK87783D0 (da) 1983-02-24
FI72322C (fi) 1987-05-11
AU1180183A (en) 1983-09-01
ZA831206B (en) 1983-11-30
PH18435A (en) 1985-07-08
GR78112B (fr) 1984-09-26
PL138759B1 (en) 1986-10-31
HU194269B (en) 1988-01-28
GB8305005D0 (en) 1983-03-30
ES8505207A1 (es) 1985-05-16
CS235309B2 (en) 1985-05-15
RO85833A (fr) 1984-11-25
ES526529A0 (es) 1985-05-16
EP0087921A1 (fr) 1983-09-07
DK87783A (da) 1983-08-26
SU1360588A3 (ru) 1987-12-15
ES8403926A1 (es) 1984-04-01
KR840003646A (ko) 1984-09-15
PT76272B (en) 1986-02-04
PT76272A (en) 1983-03-01
DD210283A5 (de) 1984-06-06
ATE16008T1 (de) 1985-10-15
GB2115813B (en) 1985-09-11
JPH0142277B2 (fr) 1989-09-11
JPS58146595A (ja) 1983-09-01
NZ203365A (en) 1985-07-12
FI830585A0 (fi) 1983-02-22
PL240735A1 (en) 1983-09-26
EP0087921B1 (fr) 1985-10-09
IL67973A0 (en) 1983-06-15

Similar Documents

Publication Publication Date Title
DK153795C (da) Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte
DK161770C (da) Analogifremgangsmaade til fremstilling af cyklobutylaminderivater eller farmaceutisk acceptable salte deraf
DK245883A (da) Fremgangsmaade til fremstilling af en eller flere af de rene enkeltfaktorer 1, 2, 3, 4 og 5 af teichomycin a2 eller farmaceutisk acceptable salte deraf
DK153555C (da) Analogifremgangsmaade til fremstilling af 20-amino-derivater af tylosin, desmycosin, macrosin eller lactenocin eller syreadditionssalte deraf
DK156252C (da) Analogifremgangsmaade til fremstilling af di-, tri- eller tetrapeptidderivater eller salte deraf
DK145381C (da) Fremgangsmaade til fremstilling af et antibiotisk stof,kaldet n-acetyldehydrothienamycin,eller farmaceutisk acceptable salte deraf
DK413883A (da) Fremgangsmaade til fremstilling af c-20-modificerede macrolidderivater eller farmaceutisk acceptable salte deraf
DK158658C (da) Analogifremgangsmaade til fremstilling af 9-aminoalkylfluorener eller farmaceutisk acceptable salte deraf
IT8224053A0 (it) Procedimento per la preparazione di derivati di eburnamonina.
DK138498B (da) Analogifremgangsmåde til fremstilling af antibiotikum A204I-derivater eller fysiologisk acceptable kationiske salte deraf.
DK165983C (da) Fremgangsmaade til fremstilling af phosphorholdige antibiotiske forbindelser betegnet cl 1565-a, cl 1565-b og cl 1565-t eller farmaceutisk acceptable salte deraf
IT8522327A0 (it) Derivati macromolecolarizzati di cdp-colina, procedimento per laloro preparazione e composizioni farmaceutiche che li contengono.
DK144855C (da) Fremgangsmaade til fremstilling af det antibiotiske stof sisomicin eller terapeutisk acceptable salte deraf
NO872331D0 (no) Farmasoeytiske preparater for behandling av bakterielle infeksjoner.
DK163300C (da) Analogifremgangsmaade til fremstilling af fluorerede alkandiaminderivater eller pharmaceutisk acceptable salte deraf
DK149064C (da) Analogifremgangsmaade til fremstilling af enkefalin-analoge tetrapeptidhydrazidderivater eller farmaceutisk acceptable salte deraf
DK494282A (da) Cycliske iminderivater eller salte deraf, deres fremstilling og anvendelse som antiarytmiske midler
DK440880A (da) Benzimidazolderivater eller salte deraf og fremgangsmaade til deres fr&mstilling
DK154075C (da) Analogifremgangsmaade til fremstilling af 4-carbamoyl-5-hydroxy-imidazolderivater eller farmaceutisk acceptable salte deraf
DK497983D0 (da) Fremgangsmade til fremstilling af 5-phenyl-hydantoin-derivater eller farmaceutisk acceptable salte deraf
DK40882A (da) Fremgangsmaade til fremstilling af antibiotikummet tue 1718 eller derivater eller salte deraf
IT8120781A0 (it) Derivati di benzilalcool e procedimenti per preparare glistessi.
DK98788A (da) Benzylaminoaryl-dihydropyridinlactoner, fremgangmsaade til deres fremstilling samt deres anvendelse som laegemidler
DK152123C (da) Analogifremgangsmaade til fremstilling af 3,4,5-trihydroxypiperidinderivater eller farmaceutisk acceptable salte eller stereoisomere deraf
DK377883D0 (da) Fremgangsmade til fremstilling af a-58365, dets enkelte faktorer eller farmaceutisk acceptable salte deraf og mikroorganismer dertil

Legal Events

Date Code Title Description
PBP Patent lapsed