DK413883A - Fremgangsmaade til fremstilling af c-20-modificerede macrolidderivater eller farmaceutisk acceptable salte deraf - Google Patents
Fremgangsmaade til fremstilling af c-20-modificerede macrolidderivater eller farmaceutisk acceptable salte deraf Download PDFInfo
- Publication number
- DK413883A DK413883A DK413883A DK413883A DK413883A DK 413883 A DK413883 A DK 413883A DK 413883 A DK413883 A DK 413883A DK 413883 A DK413883 A DK 413883A DK 413883 A DK413883 A DK 413883A
- Authority
- DK
- Denmark
- Prior art keywords
- preparing
- procedure
- acceptable salts
- pharmaceutical acceptable
- macrolide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fodder In General (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/417,248 US4443436A (en) | 1982-09-13 | 1982-09-13 | C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK413883D0 DK413883D0 (da) | 1983-09-12 |
| DK413883A true DK413883A (da) | 1984-03-14 |
Family
ID=23653187
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK413883A DK413883A (da) | 1982-09-13 | 1983-09-12 | Fremgangsmaade til fremstilling af c-20-modificerede macrolidderivater eller farmaceutisk acceptable salte deraf |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4443436A (da) |
| EP (2) | EP0203621B1 (da) |
| JP (1) | JPS5973599A (da) |
| KR (1) | KR850001952B1 (da) |
| AT (1) | AT381708B (da) |
| AU (1) | AU565892B2 (da) |
| CA (1) | CA1229336A (da) |
| DE (2) | DE3381289D1 (da) |
| DK (1) | DK413883A (da) |
| GB (1) | GB2127018B (da) |
| GR (1) | GR78989B (da) |
| HU (1) | HUT35274A (da) |
| IE (1) | IE55917B1 (da) |
| IL (1) | IL69667A0 (da) |
| NZ (1) | NZ205502A (da) |
| PH (1) | PH19760A (da) |
| ZA (1) | ZA836742B (da) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4820695A (en) * | 1982-09-13 | 1989-04-11 | Eli Lilly And Company | C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics |
| US4629786A (en) * | 1983-02-28 | 1986-12-16 | Eli Lilly And Company | C-20- and C-23 modified macrolide derivatives |
| IL71032A0 (en) * | 1983-02-28 | 1984-05-31 | Lilly Co Eli | C-20 and c-23-modified macrolide derivatives |
| GB8405087D0 (en) * | 1984-02-27 | 1984-04-04 | Omura S | Antibiotic |
| US4921947A (en) * | 1986-03-31 | 1990-05-01 | Eli Lilly And Company | Process for preparing macrolide derivatives |
| EP0262903A3 (en) * | 1986-09-29 | 1988-11-02 | Eli Lilly And Company | New acyl derivatives of 20-modified tylosin and desmycosin compounds |
| US4920103A (en) * | 1986-09-29 | 1990-04-24 | Eli Lilly And Company | Modifications of mycinose and 3-O-demethylmycinose in tylosin-type macrolides |
| US4820694A (en) * | 1986-09-29 | 1989-04-11 | Eli Lilly And Company | Modifications of 3-O-demethylmycinose in macrocin and lactenocin |
| SI8710674B (sl) * | 1987-04-14 | 1998-06-30 | Pliva | Postopek za pripravo 10,11,12,13-tetrahidro derivatov tilozina |
| ATE150757T1 (de) * | 1992-01-14 | 1997-04-15 | Zaidan Hojin Biseibutsu | 3,4'-didesoxymycaminosyltylonolid-derivate und herstellung davon |
| US5354708A (en) * | 1992-06-04 | 1994-10-11 | Taskar Nikhil R | Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine |
| TW226373B (da) * | 1992-07-15 | 1994-07-11 | Pfizer | |
| AU3121095A (en) * | 1994-09-22 | 1996-04-09 | Pfizer Inc. | Antibiotic macrolides |
| AU2014270353B2 (en) * | 2013-05-23 | 2018-09-20 | Elanco Animal Health Gmbh | Tylosin derivatives and method for preparation thereof |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1278441B (de) * | 1958-10-29 | 1968-09-26 | Lilly Co Eli | Verfahren zur Herstellung von Acylderivaten von Tylosin und Desmycosin und deren Salzen |
| US3178341A (en) * | 1960-06-27 | 1965-04-13 | Lilly Co Eli | Antibiotics tylosin and desmycosin and derivatives thereof |
| US3326759A (en) * | 1962-07-19 | 1967-06-20 | Lilly Co Eli | Antibiotics macrocin and lactenocin |
| JPS5321182A (en) * | 1976-08-10 | 1978-02-27 | Sanraku Inc | Antibiotic angolamycin derivatives and their preparation |
| GB1587685A (en) * | 1977-03-09 | 1981-04-08 | Microbial Chem Res Found | Macrolactone derivatives and their production |
| JPS53130686A (en) * | 1977-04-19 | 1978-11-14 | Toyo Jozo Co Ltd | 17-deformyl-17-thiazolidyl macrolide antibiotics |
| JPS53132584A (en) * | 1977-04-26 | 1978-11-18 | Toyo Jozo Co Ltd | 18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative |
| SE445739B (sv) * | 1978-09-14 | 1986-07-14 | Toyo Jozo Kk | 3", 4"-diacyltylosinderivat |
| JPS5655399A (en) * | 1979-09-19 | 1981-05-15 | Toyo Jozo Co Ltd | Deformyltylosin derivative |
| NL8004922A (nl) * | 1979-09-19 | 1981-03-23 | Toyo Jozo Kk | Deformyltylosinederivaten. |
| JPS5671099A (en) * | 1979-11-13 | 1981-06-13 | Toyo Jozo Co Ltd | 20-deoxodesmycosin |
| US4321361A (en) * | 1980-06-12 | 1982-03-23 | Eli Lilly And Company | Demycinosyltylosin and process for its production |
| US4279896A (en) * | 1980-06-23 | 1981-07-21 | Schering Corporation | Novel 20-imino macrolide antibacterial agents |
| US4349665A (en) * | 1980-06-27 | 1982-09-14 | Schering Corporation | Macrolide antibiotic complex |
| HU189519B (en) * | 1980-07-24 | 1986-07-28 | Eli Lilly And Co,Us | Process for preparing 2'''-o-demethyl-macrocin derivatives |
| US4299953A (en) * | 1980-07-29 | 1981-11-10 | Eli Lilly And Company | Mycarosyltylactone |
| US4304856A (en) * | 1980-11-10 | 1981-12-08 | Eli Lilly And Company | Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin |
| US4357325A (en) * | 1981-04-20 | 1982-11-02 | Eli Lilly And Company | Methods of controlling Pasteurella infections |
| US4401660A (en) | 1981-12-14 | 1983-08-30 | Eli Lilly And Company | Ester derivatives of 5-O-mycaminosyl tylonolide and method of using same |
| JPS58146595A (ja) * | 1982-02-25 | 1983-09-01 | Satoshi Omura | マクロライド系抗生物質 |
-
1982
- 1982-09-13 US US06/417,248 patent/US4443436A/en not_active Expired - Fee Related
-
1983
- 1983-09-05 AU AU18711/83A patent/AU565892B2/en not_active Ceased
- 1983-09-05 IL IL69667A patent/IL69667A0/xx unknown
- 1983-09-06 NZ NZ205502A patent/NZ205502A/en unknown
- 1983-09-07 GR GR72393A patent/GR78989B/el unknown
- 1983-09-07 PH PH29507A patent/PH19760A/en unknown
- 1983-09-08 GB GB08324045A patent/GB2127018B/en not_active Expired
- 1983-09-08 DE DE8686108251T patent/DE3381289D1/de not_active Expired - Lifetime
- 1983-09-08 EP EP86108251A patent/EP0203621B1/en not_active Expired - Lifetime
- 1983-09-08 EP EP83305240A patent/EP0104028B1/en not_active Expired
- 1983-09-08 DE DE8383305240T patent/DE3377576D1/de not_active Expired
- 1983-09-08 AT AT0320783A patent/AT381708B/de not_active IP Right Cessation
- 1983-09-12 ZA ZA836742A patent/ZA836742B/xx unknown
- 1983-09-12 CA CA000436450A patent/CA1229336A/en not_active Expired
- 1983-09-12 HU HU833166A patent/HUT35274A/hu unknown
- 1983-09-12 KR KR1019830004274A patent/KR850001952B1/ko not_active IP Right Cessation
- 1983-09-12 DK DK413883A patent/DK413883A/da not_active Application Discontinuation
- 1983-09-12 IE IE2132/83A patent/IE55917B1/xx unknown
- 1983-09-13 JP JP58169128A patent/JPS5973599A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| KR840005735A (ko) | 1984-11-15 |
| EP0203621B1 (en) | 1990-03-07 |
| IE55917B1 (en) | 1991-02-27 |
| EP0203621A1 (en) | 1986-12-03 |
| AU1871183A (en) | 1984-03-22 |
| ZA836742B (en) | 1984-04-25 |
| GB2127018B (en) | 1986-02-12 |
| AU565892B2 (en) | 1987-10-01 |
| EP0104028B1 (en) | 1988-08-03 |
| AT381708B (de) | 1986-11-25 |
| GB2127018A (en) | 1984-04-04 |
| GB8324045D0 (en) | 1983-10-12 |
| US4443436A (en) | 1984-04-17 |
| JPH0517240B2 (da) | 1993-03-08 |
| CA1229336A (en) | 1987-11-17 |
| DE3381289D1 (de) | 1990-04-12 |
| JPS5973599A (ja) | 1984-04-25 |
| GR78989B (da) | 1984-10-02 |
| IE832132L (en) | 1984-03-13 |
| PH19760A (en) | 1986-06-26 |
| NZ205502A (en) | 1986-03-14 |
| KR850001952B1 (ko) | 1985-12-31 |
| ATA320783A (de) | 1986-04-15 |
| IL69667A0 (en) | 1983-12-30 |
| DE3377576D1 (en) | 1988-09-08 |
| DK413883D0 (da) | 1983-09-12 |
| EP0104028A1 (en) | 1984-03-28 |
| HUT35274A (en) | 1985-06-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |