CS226747B2 - Method of preparing new benztriazols - Google Patents

Method of preparing new benztriazols

Info

Publication number
CS226747B2
CS226747B2 CS825592A CS559282A CS226747B2 CS 226747 B2 CS226747 B2 CS 226747B2 CS 825592 A CS825592 A CS 825592A CS 559282 A CS559282 A CS 559282A CS 226747 B2 CS226747 B2 CS 226747B2
Authority
CS
Czechoslovakia
Prior art keywords
methyl
dihydro
pyridazinone
amino
theory
Prior art date
Application number
CS825592A
Other languages
Czech (cs)
English (en)
Inventor
Norbert Dr Hauel
Volkhard Dr Austel
Joachim Dr Heider
Manfred Dr Reiffen
Willi Dr Diederen
Walter Dr Haarmann
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of CS226747B2 publication Critical patent/CS226747B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/04Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/16Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C07D249/18Benzotriazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS825592A 1981-07-25 1982-07-22 Method of preparing new benztriazols CS226747B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813129447 DE3129447A1 (de) 1981-07-25 1981-07-25 "neue benztriazole, ihre herstellung und ihre verwendung als arzneimittel"

Publications (1)

Publication Number Publication Date
CS226747B2 true CS226747B2 (en) 1984-04-16

Family

ID=6137768

Family Applications (1)

Application Number Title Priority Date Filing Date
CS825592A CS226747B2 (en) 1981-07-25 1982-07-22 Method of preparing new benztriazols

Country Status (27)

Country Link
US (1) US4616018A (ru)
EP (1) EP0071102B1 (ru)
JP (1) JPS5824582A (ru)
KR (1) KR880001476B1 (ru)
AR (1) AR230631A1 (ru)
AT (1) ATE16184T1 (ru)
AU (1) AU554184B2 (ru)
CA (1) CA1189076A (ru)
CS (1) CS226747B2 (ru)
DD (1) DD202564A5 (ru)
DE (2) DE3129447A1 (ru)
DK (1) DK331282A (ru)
ES (2) ES8308325A1 (ru)
FI (1) FI73994C (ru)
GB (1) GB2107703B (ru)
GR (1) GR76230B (ru)
HU (1) HU188585B (ru)
IE (1) IE53664B1 (ru)
IL (1) IL66385A (ru)
NO (1) NO159273C (ru)
NZ (1) NZ201364A (ru)
PH (1) PH19512A (ru)
PL (1) PL130643B1 (ru)
PT (1) PT75313B (ru)
SU (1) SU1179927A3 (ru)
YU (1) YU42783B (ru)
ZA (1) ZA825275B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8320005D0 (en) * 1983-07-25 1983-08-24 Fujisawa Pharmaceutical Co Benzothiazoline derivatives
DE3511110A1 (de) * 1985-03-27 1986-10-02 Dr. Karl Thomae Gmbh, 7950 Biberach Neue pyridazinone, ihre herstellung und diese verbindungen enthaltende arzneimittel
DE3734083A1 (de) * 1987-10-08 1989-04-20 Heumann Pharma Gmbh & Co Benzimidazole, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
ATE128135T1 (de) * 1988-07-11 1995-10-15 Akzo Nobel Nv Pyridazinon-derivate.
DE3934436A1 (de) * 1989-06-01 1991-04-18 Thomae Gmbh Dr K 2-hydroxy-n-propylamine, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung
CA2451699A1 (en) * 2001-06-26 2003-01-09 Beth Israel Deaconess Medical Center Compositions and methods for inhibiting platelet activation and thrombosis
GB201321740D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2516040C2 (de) * 1974-06-10 1984-12-20 Dr. Karl Thomae Gmbh, 7950 Biberach Benzimidazole, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
ES482789A0 (es) * 1978-08-25 1980-12-01 Thomae Gmbh Dr K Procedimiento para la preparacion de nuevos bencimidazoles sustituidos en posicion 5 o 6 con un anillo de piridazinona
DE2845220A1 (de) * 1978-10-17 1980-04-30 Yoshitomi Pharmaceutical Pyridazinon-derivate, ihre salze mit saeuren, verfahren zu ihrer herstellung und ihre verwendung bei der behandlung von thrombosen und hypertonie
US4258185A (en) * 1978-10-17 1981-03-24 Yoshitomi Pharmaceutical Industries, Ltd. Pyridazinone compounds

Also Published As

Publication number Publication date
PH19512A (en) 1986-05-14
PL130643B1 (en) 1984-08-31
IE821781L (en) 1983-01-25
FI822549A0 (fi) 1982-07-20
DE3267020D1 (en) 1985-11-28
PT75313A (de) 1982-08-01
ES514274A0 (es) 1983-08-16
ES8308325A1 (es) 1983-08-16
AU8637782A (en) 1983-02-03
DK331282A (da) 1983-01-26
AU554184B2 (en) 1986-08-14
ES519351A0 (es) 1983-11-01
EP0071102B1 (de) 1985-10-23
US4616018A (en) 1986-10-07
NO159273C (no) 1988-12-14
FI73994C (fi) 1987-12-10
FI822549L (fi) 1983-01-26
YU42783B (en) 1988-12-31
FI73994B (fi) 1987-08-31
GB2107703A (en) 1983-05-05
IL66385A (en) 1985-11-29
NO822119L (no) 1983-01-26
NO159273B (no) 1988-09-05
PL237601A1 (en) 1983-05-09
AR230631A1 (es) 1984-05-31
IL66385A0 (en) 1982-11-30
ATE16184T1 (de) 1985-11-15
YU159782A (en) 1984-08-31
HU188585B (en) 1986-04-28
ZA825275B (en) 1984-03-28
CA1189076A (en) 1985-06-18
KR880001476B1 (ko) 1988-08-13
NZ201364A (en) 1986-01-24
PT75313B (de) 1985-11-29
GR76230B (ru) 1984-08-04
DD202564A5 (de) 1983-09-21
JPS5824582A (ja) 1983-02-14
IE53664B1 (en) 1989-01-04
EP0071102A1 (de) 1983-02-09
DE3129447A1 (de) 1983-02-10
SU1179927A3 (ru) 1985-09-15
GB2107703B (en) 1985-06-12
ES8400744A1 (es) 1983-11-01
KR840000530A (ko) 1984-02-25

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