CS221801B2 - Method of praparation of the derivative of 4-deoxy-4-aminoerythromycine a - Google Patents

Method of praparation of the derivative of 4-deoxy-4-aminoerythromycine a Download PDF

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Publication number
CS221801B2
CS221801B2 CS78703A CS70378A CS221801B2 CS 221801 B2 CS221801 B2 CS 221801B2 CS 78703 A CS78703 A CS 78703A CS 70378 A CS70378 A CS 70378A CS 221801 B2 CS221801 B2 CS 221801B2
Authority
CS
Czechoslovakia
Prior art keywords
hydrogen
product
acid
solution
water
Prior art date
Application number
CS78703A
Other languages
Czech (cs)
English (en)
Inventor
Frank Ch Sciavolono
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/856,479 external-priority patent/US4150220A/en
Application filed by Pfizer filed Critical Pfizer
Publication of CS221801B2 publication Critical patent/CS221801B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS78703A 1977-02-04 1978-02-02 Method of praparation of the derivative of 4-deoxy-4-aminoerythromycine a CS221801B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76548077A 1977-02-04 1977-02-04
US05/856,479 US4150220A (en) 1977-02-04 1977-12-01 Semi-synthetic 4"-erythromycin A derivatives

Publications (1)

Publication Number Publication Date
CS221801B2 true CS221801B2 (en) 1983-04-29

Family

ID=27117613

Family Applications (1)

Application Number Title Priority Date Filing Date
CS78703A CS221801B2 (en) 1977-02-04 1978-02-02 Method of praparation of the derivative of 4-deoxy-4-aminoerythromycine a

Country Status (30)

Country Link
JP (1) JPS5827798B2 (xx)
AR (1) AR222147A1 (xx)
AU (1) AU501298B1 (xx)
BG (2) BG32718A3 (xx)
CA (1) CA1106367A (xx)
CH (1) CH628906A5 (xx)
CS (1) CS221801B2 (xx)
DD (1) DD140048A5 (xx)
DE (1) DE2804507C2 (xx)
DK (1) DK148036C (xx)
ES (2) ES466057A1 (xx)
FI (1) FI780354A (xx)
FR (2) FR2379550A1 (xx)
GB (2) GB1585316A (xx)
GR (1) GR68691B (xx)
HU (1) HU182559B (xx)
IE (1) IE46661B1 (xx)
IL (2) IL53968A0 (xx)
IT (1) IT1094209B (xx)
LU (1) LU79004A1 (xx)
NL (1) NL176174C (xx)
NO (2) NO146472C (xx)
NZ (1) NZ186385A (xx)
PH (2) PH14421A (xx)
PL (1) PL116228B1 (xx)
PT (1) PT67568B (xx)
RO (4) RO77345A (xx)
SE (2) SE445223B (xx)
SU (1) SU927122A3 (xx)
YU (3) YU40913B (xx)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4382085A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
HN1998000074A (es) * 1997-06-11 1999-01-08 Pfizer Prod Inc Derivados de macrolidos c-4 sustituidos
US6407074B1 (en) 1997-06-11 2002-06-18 Pfizer Inc C-4″-substituted macrolide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

Also Published As

Publication number Publication date
FR2385735B1 (xx) 1980-10-24
GR68691B (xx) 1982-02-01
FR2385735A1 (fr) 1978-10-27
NO146472B (no) 1982-06-28
RO81622A (ro) 1983-04-29
HU182559B (en) 1984-02-28
IT7820005A0 (it) 1978-02-03
ES472429A1 (es) 1979-04-01
YU40799B (en) 1986-06-30
DK51878A (da) 1978-08-05
PH14421A (en) 1981-07-10
NL176174B (nl) 1984-10-01
NO150484C (no) 1984-10-24
IL53968A0 (en) 1978-04-30
SE8300870L (sv) 1983-02-16
PT67568B (en) 1979-06-18
RO79687A7 (ro) 1982-08-17
SE445223B (sv) 1986-06-09
GB1585315A (en) 1981-02-25
IE780239L (en) 1978-08-04
RO81622B (ro) 1983-04-30
NL176174C (nl) 1985-03-01
PT67568A (en) 1978-02-01
AU501298B1 (en) 1979-06-14
BG33159A3 (en) 1982-12-15
YU227983A (en) 1984-04-30
IL61997A0 (en) 1981-02-27
SE457086B (sv) 1988-11-28
FR2379550A1 (fr) 1978-09-01
LU79004A1 (fr) 1979-09-06
YU40798B (en) 1986-06-30
PL204428A1 (pl) 1979-06-04
RO79686A7 (ro) 1982-08-17
YU40913B (en) 1986-08-31
ES466057A1 (es) 1978-10-01
FR2379550B1 (xx) 1980-07-04
IE46661B1 (en) 1983-08-24
CA1106367A (en) 1981-08-04
BG32718A3 (en) 1982-09-15
SE8300870D0 (sv) 1983-02-16
CH628906A5 (en) 1982-03-31
NO150484B (no) 1984-07-16
NO780389L (no) 1978-08-07
YU7378A (en) 1983-04-30
FI780354A (fi) 1978-08-05
DE2804507C2 (de) 1982-11-04
YU26583A (en) 1984-02-29
DD140048A5 (de) 1980-02-06
DE2804507A1 (de) 1978-08-10
GB1585316A (en) 1981-02-25
NO146472C (no) 1982-10-06
RO77345A (ro) 1981-08-17
DK148036C (da) 1985-07-15
NL7801262A (nl) 1978-08-08
DK148036B (da) 1985-02-11
SU927122A3 (ru) 1982-05-07
PL116228B1 (en) 1981-05-30
SE7800270L (sv) 1978-08-05
PH16675A (en) 1983-12-13
NO811913L (no) 1978-08-07
AR222147A1 (es) 1981-04-30
NZ186385A (en) 1980-10-08
IT1094209B (it) 1985-07-26
JPS5827798B2 (ja) 1983-06-11
JPS53101337A (en) 1978-09-04

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