CS216525B2 - Method of making the phenylpiperazine derivatives - Google Patents
Method of making the phenylpiperazine derivatives Download PDFInfo
- Publication number
- CS216525B2 CS216525B2 CS801368A CS136880A CS216525B2 CS 216525 B2 CS216525 B2 CS 216525B2 CS 801368 A CS801368 A CS 801368A CS 136880 A CS136880 A CS 136880A CS 216525 B2 CS216525 B2 CS 216525B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- compound
- group
- compounds
- formula
- piperazine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyridine Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Cookers (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
NL7901633 | 1979-03-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
CS216525B2 true CS216525B2 (en) | 1982-11-26 |
Family
ID=19832723
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS801368A CS216525B2 (en) | 1979-03-01 | 1980-02-28 | Method of making the phenylpiperazine derivatives |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0015615B1 (es) |
JP (1) | JPS55141478A (es) |
AT (1) | ATE2219T1 (es) |
AU (1) | AU532411B2 (es) |
CA (1) | CA1138461A (es) |
CS (1) | CS216525B2 (es) |
DD (1) | DD151408A5 (es) |
DE (1) | DE3061561D1 (es) |
DK (1) | DK84380A (es) |
ES (3) | ES8106898A1 (es) |
FI (1) | FI800588A (es) |
GR (1) | GR67005B (es) |
HU (1) | HU182070B (es) |
IE (1) | IE49526B1 (es) |
IL (1) | IL59489A (es) |
PH (1) | PH17025A (es) |
PL (1) | PL126161B1 (es) |
SU (1) | SU1039442A3 (es) |
YU (1) | YU54680A (es) |
ZA (1) | ZA801119B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL8005133A (nl) * | 1980-09-12 | 1982-04-01 | Duphar Int Res | Fenylpiperazinederivaten met antiagressieve werking. |
NL8005131A (nl) * | 1980-09-12 | 1982-04-01 | Duphar Int Res | Fenylpiperazinederivaten met analgetische werking. |
US4457931A (en) * | 1982-09-27 | 1984-07-03 | Selvi & C. S.P.A. | Piperazine derivatives with anticholinergic and/or antihistaminic activity |
JPH0660160B2 (ja) * | 1985-12-13 | 1994-08-10 | テルモ株式会社 | アミド誘導体およびこれを含有する抗アレルギ−剤 |
US5340812A (en) * | 1989-04-22 | 1994-08-23 | John Wyeth & Brother, Limited | Piperazine derivatives |
DK0395313T3 (da) * | 1989-04-22 | 2000-06-19 | American Home Prod | Tertiære alkyl-funktionaliserede piperazin-derivater |
US5382583A (en) * | 1989-04-22 | 1995-01-17 | John Wyeth & Brother, Limited | Piperazine derivatives |
FI102175B1 (fi) * | 1989-04-22 | 1998-10-30 | Wyeth John & Brother Ltd | Menetelmä terapeuttisesti käyttökelpoisten piperatsiinijohdannaisten valmistamiseksi |
DK203990D0 (da) * | 1990-08-24 | 1990-08-24 | Novo Nordisk As | Piperazinylderivater |
GB9200293D0 (en) * | 1992-01-08 | 1992-02-26 | Wyeth John & Brother Ltd | Piperazine derivatives |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2833770A (en) * | 1958-05-06 | Chj-chj | ||
US2722529A (en) * | 1955-11-01 | Amides of certain l-amevoalkyl-x-phenyl | ||
BE788280A (fr) * | 1971-09-04 | 1973-02-28 | Pfizer | Nouvelles 1-(3-trifluoro-methyl-phenyl)-4-((amido cyclique)- alkyl) piperazines et composition pharmaceutique les contenant |
GB1443598A (en) * | 1973-07-06 | 1976-07-21 | Acraf | 1- 3-acetylaminopropyl-4-2,5-dichlorophenyl-piperazine |
FR2306694A1 (fr) * | 1975-04-07 | 1976-11-05 | Parcor | Derives de la piperazine |
-
1980
- 1980-02-25 AU AU55848/80A patent/AU532411B2/en not_active Ceased
- 1980-02-27 FI FI800588A patent/FI800588A/fi not_active Application Discontinuation
- 1980-02-27 SU SU802890551A patent/SU1039442A3/ru active
- 1980-02-27 GR GR61296A patent/GR67005B/el unknown
- 1980-02-27 ZA ZA00801119A patent/ZA801119B/xx unknown
- 1980-02-27 ES ES488988A patent/ES8106898A1/es not_active Expired
- 1980-02-27 PL PL1980222294A patent/PL126161B1/pl unknown
- 1980-02-27 DK DK84380A patent/DK84380A/da not_active Application Discontinuation
- 1980-02-28 YU YU00546/80A patent/YU54680A/xx unknown
- 1980-02-28 CS CS801368A patent/CS216525B2/cs unknown
- 1980-02-28 PH PH23695A patent/PH17025A/en unknown
- 1980-02-28 IL IL59489A patent/IL59489A/xx unknown
- 1980-02-28 EP EP80200173A patent/EP0015615B1/en not_active Expired
- 1980-02-28 IE IE405/80A patent/IE49526B1/en unknown
- 1980-02-28 AT AT80200173T patent/ATE2219T1/de not_active IP Right Cessation
- 1980-02-28 DE DE8080200173T patent/DE3061561D1/de not_active Expired
- 1980-02-29 HU HU80474A patent/HU182070B/hu unknown
- 1980-02-29 CA CA000346735A patent/CA1138461A/en not_active Expired
- 1980-03-01 JP JP2466480A patent/JPS55141478A/ja active Pending
- 1980-03-03 DD DD80219413A patent/DD151408A5/de unknown
- 1980-09-16 ES ES495106A patent/ES495106A0/es active Granted
- 1980-09-16 ES ES495105A patent/ES495105A0/es active Granted
Also Published As
Publication number | Publication date |
---|---|
IE49526B1 (en) | 1985-10-16 |
AU532411B2 (en) | 1983-09-29 |
JPS55141478A (en) | 1980-11-05 |
ES488988A0 (es) | 1981-09-01 |
ATE2219T1 (de) | 1983-01-15 |
EP0015615B1 (en) | 1983-01-12 |
ES8200883A1 (es) | 1981-11-16 |
SU1039442A3 (ru) | 1983-08-30 |
AU5584880A (en) | 1980-09-04 |
CA1138461A (en) | 1982-12-28 |
IL59489A0 (en) | 1980-05-30 |
PH17025A (en) | 1984-05-17 |
EP0015615A1 (en) | 1980-09-17 |
GR67005B (es) | 1981-05-18 |
FI800588A (fi) | 1980-09-02 |
ES8106898A1 (es) | 1981-09-01 |
ES8200884A1 (es) | 1981-11-16 |
PL222294A1 (es) | 1980-12-01 |
DD151408A5 (de) | 1981-10-21 |
IE800405L (en) | 1980-09-01 |
YU54680A (en) | 1983-09-30 |
ES495105A0 (es) | 1981-11-16 |
DK84380A (da) | 1980-09-02 |
DE3061561D1 (en) | 1983-02-17 |
PL126161B1 (en) | 1983-07-30 |
HU182070B (en) | 1983-12-28 |
ZA801119B (en) | 1981-09-30 |
ES495106A0 (es) | 1981-11-16 |
IL59489A (en) | 1984-05-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
US5395839A (en) | Imidazopyridine derivatives and their use | |
HU184966B (en) | Process for producing phenyl-piperazine derivatives of anti-agression activity | |
US6852718B2 (en) | Phenylsulphonylipiperazinyl derivatives as 5-HT receptor ligands | |
JPS6040428B2 (ja) | 新規3−アリ−ル−2−オキサゾリジノン誘導体、その製法及び該誘導体を含有する抗抑うつ剤 | |
PT85304B (pt) | Processo para a preparacao de derivados d difenil-profilamina | |
CS216525B2 (en) | Method of making the phenylpiperazine derivatives | |
JPS60156671A (ja) | ジヒドロピリジン誘導体およびその製造法 | |
FI80448C (fi) | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara piperazinkarboxamidderivat. | |
CA1244431A (en) | Phenylpiperazine derivatives and process for producing the same | |
FR2539741A1 (fr) | Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent | |
DE68924221T2 (de) | Imidazolderivate. | |
US4109088A (en) | 2-(indenyloxymethyl) morpholine derivatives | |
CZ325196A3 (en) | Derivatives of hydroximic acid, pharmaceutical compositions containing thereof, process of their preparation and intermediates used in the preparation process | |
JPH0441149B2 (es) | ||
CS214841B2 (en) | Method of making the tetrahydrochinolines | |
JPH0451554B2 (es) | ||
DE69223422T2 (de) | Benzothiadiazinderivate | |
JPS6252740B2 (es) | ||
US4076717A (en) | Derivatives of 1-(3-cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxylic acid | |
US4059584A (en) | 2-Acylamino-3-[3-(dialkylamino)propyl]imidazo[4,5-b]pyridines | |
CZ357190A3 (en) | Dihydropyrimidothiazine derivatives, process of their preparation and pharmaceutical compositions containing thereof | |
CS270576B2 (en) | Method of substituted 1-phenoxy-3-amino-2-propanols production | |
EP0392233B1 (de) | Substituierte 1.2.3.4-Oxatriazolium-5-olate, Verfahren zu ihrer Herstellung und ihre Verwendung | |
JPS6017789B2 (ja) | 5−(ω−アミノアシル)−3−カルボアルコキシアミノ−10,11−ジヒドロ−5H−ジベンゾ−〔b,f〕−アゼピン、その塩及びそれらの製造方法 | |
FR2697253A1 (fr) | Dérivés de 2-aminopyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique. |