CS202066B2 - Method of preparing alpha-amino-phophonic acids - Google Patents

Method of preparing alpha-amino-phophonic acids Download PDF

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Publication number
CS202066B2
CS202066B2 CS773353A CS335377A CS202066B2 CS 202066 B2 CS202066 B2 CS 202066B2 CS 773353 A CS773353 A CS 773353A CS 335377 A CS335377 A CS 335377A CS 202066 B2 CS202066 B2 CS 202066B2
Authority
CS
Czechoslovakia
Prior art keywords
acid
formula
salts
converted
group
Prior art date
Application number
CS773353A
Other languages
Czech (cs)
English (en)
Inventor
John G Dingwall
Eric K Baylis
Colin D Campbell
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Priority to CS781917A priority Critical patent/CS202067B2/cs
Publication of CS202066B2 publication Critical patent/CS202066B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/48Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/58Pyridine rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CS773353A 1976-05-21 1977-05-20 Method of preparing alpha-amino-phophonic acids CS202066B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS781917A CS202067B2 (cs) 1976-05-21 1978-03-24 Způsob přípravy alfa-aminofosfinových kyselin

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB21000/76A GB1542938A (en) 1976-05-21 1976-05-21 Aminophosphonous acids and processes for their preparation

Publications (1)

Publication Number Publication Date
CS202066B2 true CS202066B2 (en) 1980-12-31

Family

ID=10155485

Family Applications (1)

Application Number Title Priority Date Filing Date
CS773353A CS202066B2 (en) 1976-05-21 1977-05-20 Method of preparing alpha-amino-phophonic acids

Country Status (29)

Country Link
US (1) US4147780A (ja)
JP (1) JPS52151128A (ja)
AR (2) AR219077A1 (ja)
AT (1) AT350585B (ja)
AU (1) AU516592B2 (ja)
BE (1) BE854843A (ja)
BG (2) BG28070A4 (ja)
CA (1) CA1081241A (ja)
CS (1) CS202066B2 (ja)
DD (1) DD131751A5 (ja)
DE (1) DE2722162A1 (ja)
DK (1) DK221477A (ja)
EG (1) EG12688A (ja)
ES (1) ES458931A1 (ja)
FI (1) FI771602A (ja)
FR (1) FR2360601A1 (ja)
GB (1) GB1542938A (ja)
IE (1) IE44904B1 (ja)
IL (1) IL52127A0 (ja)
NL (1) NL7705602A (ja)
NO (1) NO771770L (ja)
NZ (1) NZ184166A (ja)
OA (1) OA05666A (ja)
PH (1) PH14170A (ja)
PL (2) PL110527B1 (ja)
PT (1) PT66581B (ja)
SE (1) SE7705886L (ja)
SU (2) SU805948A3 (ja)
ZA (1) ZA773017B (ja)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002031B1 (en) * 1977-11-19 1982-02-03 Ciba-Geigy Ag Methods of inhibiting plant and combating weeds using alpha-aminoalkanephosphonous acids
EP0002039A1 (en) * 1977-11-19 1979-05-30 Ciba-Geigy Ag Phosphonous acid derivatives, processes for their preparation and their use in combating microorganisms
IL61985A0 (en) * 1980-02-01 1981-02-27 Sparamedica Ag Phosphinic and phosphonic acid derivatives,their manufacture and pharmaceutical compositions containing them
US4473561A (en) * 1981-04-17 1984-09-25 Sumitomo Chemical Company, Limited Fungicidal composition comprising alpha-substituted ethylphosphinic acids or their salts
US4466913A (en) * 1981-06-30 1984-08-21 Maiji Seika Kaisha Ltd. Phosphorus-containing compounds and process for producing the same
US4477391A (en) * 1981-08-14 1984-10-16 Collins James F Amino acid isomers, their production and their medicinal use
SE455259B (sv) * 1984-01-30 1988-07-04 Kenogard Ab Anvendning av vissa aminoalkanfosfonsyror for bekempning av svampsjukdomar hos vexter
US5189030A (en) * 1985-06-11 1993-02-23 Ciba-Geigy Corporation 1-amino-2-phenylethanephosphonic acids as microbiocides
US5099063A (en) * 1986-11-05 1992-03-24 Merck & Co., Inc. Certain phosphinic acid derivatives having antibacterial activity
US5143908A (en) * 1986-11-05 1992-09-01 Merck & Co., Inc. Antibacterial agents and potentiators of carbapenem antibiotics
US4761405A (en) * 1987-03-04 1988-08-02 Nova Pharmaceutical Corporation Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency
US5041644A (en) * 1987-07-06 1991-08-20 Merck & Co., Inc. Peptide derivatives of β-chloro-L(Z)-dehydro-glutamic acid
JPS6413097A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Phosphonic acid derivative
US5030732A (en) * 1988-03-03 1991-07-09 Merck & Co., Inc. Aminoethylphosphinic acid derivatives
US4962097A (en) * 1988-10-28 1990-10-09 Merck & Co., Inc. Method of treating bacterial infection with phosphorus containing DHP enzyme inhibitors
US5147867A (en) * 1988-10-28 1992-09-15 Merck & Co., Inc. Phosphorus containing enzyme inhibitors
US5145990A (en) * 1988-10-28 1992-09-08 Merck & Co., Inc. Phosphorous containing dhp enzyme inhibitors
US5179173A (en) * 1991-04-10 1993-01-12 Nalco Chemical Company Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom
FI963390A (fi) * 1996-08-30 1998-03-01 Khomutov Radii M Kasvinsuojeluaineet
IT201600098005A1 (it) * 2016-09-29 2018-03-29 Univ Degli Studi Roma La Sapienza Analoghi e derivati di amminoacidi dicarbossilici come antibatterici

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3160632A (en) * 1961-01-30 1964-12-08 Stauffer Chemical Co Aminomethylenephosphinic acids, salts thereof, and process for their production
CH475287A (de) * 1965-10-27 1969-07-15 Monsanto Co Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren
US3424788A (en) * 1967-07-24 1969-01-28 Armour & Co Aminophosphinic acids and salts useful as bacteriostats

Also Published As

Publication number Publication date
NO771770L (no) 1977-11-22
EG12688A (en) 1979-06-30
ATA361777A (de) 1978-11-15
FI771602A (ja) 1977-11-22
GB1542938A (en) 1979-03-28
CA1081241A (en) 1980-07-08
AU516592B2 (en) 1981-06-11
PL106608B1 (pl) 1980-01-31
SE7705886L (sv) 1977-11-22
DK221477A (da) 1977-11-22
IL52127A0 (en) 1977-07-31
ES458931A1 (es) 1978-03-01
AU2531977A (en) 1978-11-23
FR2360601B1 (ja) 1979-09-07
PT66581A (en) 1977-06-01
DE2722162A1 (de) 1977-12-01
PH14170A (en) 1981-03-19
IE44904B1 (en) 1982-05-05
NZ184166A (en) 1980-03-05
JPS52151128A (en) 1977-12-15
NL7705602A (nl) 1977-11-23
OA05666A (fr) 1981-05-31
PL198267A1 (pl) 1978-03-13
AR222464A1 (es) 1981-05-29
ZA773017B (en) 1978-04-26
PL110527B1 (en) 1980-07-31
AR219077A1 (es) 1980-07-31
AT350585B (de) 1979-06-11
US4147780A (en) 1979-04-03
BG27905A3 (en) 1980-01-15
SU795484A3 (ru) 1981-01-07
DD131751A5 (de) 1978-07-19
BG28070A4 (en) 1980-02-25
SU805948A3 (ru) 1981-02-15
BE854843A (fr) 1977-11-21
IE44904L (en) 1977-11-21
PT66581B (en) 1978-10-20
FR2360601A1 (fr) 1978-03-03

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