ES458931A1 - Procedimiento para preparar derivados de acidos fosfonosos. - Google Patents
Procedimiento para preparar derivados de acidos fosfonosos.Info
- Publication number
- ES458931A1 ES458931A1 ES458931A ES458931A ES458931A1 ES 458931 A1 ES458931 A1 ES 458931A1 ES 458931 A ES458931 A ES 458931A ES 458931 A ES458931 A ES 458931A ES 458931 A1 ES458931 A1 ES 458931A1
- Authority
- ES
- Spain
- Prior art keywords
- yeast
- amino
- phosphonous acids
- inhibiting bacteria
- phosphonous
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 241000894006 Bacteria Species 0.000 title abstract 2
- 240000004808 Saccharomyces cerevisiae Species 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title abstract 2
- 150000007513 acids Chemical class 0.000 title abstract 2
- 230000002401 inhibitory effect Effects 0.000 title 1
- XRBCRPZXSCBRTK-UHFFFAOYSA-N phosphonous acid Chemical class OPO XRBCRPZXSCBRTK-UHFFFAOYSA-N 0.000 abstract 2
- 244000052616 bacterial pathogen Species 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/48—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
Abstract
Procedimiento para preparar derivados de ácidos fosfonosos, de fórmula general I *** o la correspondiente forma zwitteriónica, en cuya fórmula R y R1, que pueden ser iguales o diferentes, representan hidrógeno, deuterio o un grupo alquilo inferior, alquenilo inferior, alquinilo inferior o cicloalquilo, un grupo arilo o un anillo heterocíclico de 3 a 7 miembros conteniendo uno o más átomos de oxígeno, nitrógeno o azufre y que puede estar fusionado a un anillo aromático, un grupo alquilo inferior sustituido por un radical alquilo con 6 o 10 átomos de carbono, un grupo alquilo inferior sustituido con un anillo heterocíclico de 3 a 7 miembros como anteriormente se ha definido o R y R1 juntas forman una cadena polimetileno C2-C7 interrumpida opcionalmente por un átomo de oxígeno , nitrógeno o azufre, y sus sales con ácidos o bases farmaceúticamente aceptables y todos sus isómeros ópticos con la condición de que R y R1 no pueden ser ambos hidrógeno.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB21000/76A GB1542938A (en) | 1976-05-21 | 1976-05-21 | Aminophosphonous acids and processes for their preparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES458931A1 true ES458931A1 (es) | 1978-03-01 |
Family
ID=10155485
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES458931A Expired ES458931A1 (es) | 1976-05-21 | 1977-05-19 | Procedimiento para preparar derivados de acidos fosfonosos. |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US4147780A (es) |
| JP (1) | JPS52151128A (es) |
| AR (2) | AR219077A1 (es) |
| AT (1) | AT350585B (es) |
| AU (1) | AU516592B2 (es) |
| BE (1) | BE854843A (es) |
| BG (2) | BG27905A3 (es) |
| CA (1) | CA1081241A (es) |
| CS (1) | CS202066B2 (es) |
| DD (1) | DD131751A5 (es) |
| DE (1) | DE2722162A1 (es) |
| DK (1) | DK221477A (es) |
| EG (1) | EG12688A (es) |
| ES (1) | ES458931A1 (es) |
| FI (1) | FI771602A (es) |
| FR (1) | FR2360601A1 (es) |
| GB (1) | GB1542938A (es) |
| IE (1) | IE44904B1 (es) |
| IL (1) | IL52127A0 (es) |
| NL (1) | NL7705602A (es) |
| NO (1) | NO771770L (es) |
| NZ (1) | NZ184166A (es) |
| OA (1) | OA05666A (es) |
| PH (1) | PH14170A (es) |
| PL (2) | PL110527B1 (es) |
| PT (1) | PT66581B (es) |
| SE (1) | SE7705886L (es) |
| SU (2) | SU805948A3 (es) |
| ZA (1) | ZA773017B (es) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0002039A1 (en) * | 1977-11-19 | 1979-05-30 | Ciba-Geigy Ag | Phosphonous acid derivatives, processes for their preparation and their use in combating microorganisms |
| DE2861609D1 (en) * | 1977-11-19 | 1982-03-11 | Ciba Geigy Ag | Methods of inhibiting plant and combating weeds using alpha-aminoalkanephosphonous acids |
| IL61985A0 (en) * | 1980-02-01 | 1981-02-27 | Sparamedica Ag | Phosphinic and phosphonic acid derivatives,their manufacture and pharmaceutical compositions containing them |
| US4473561A (en) * | 1981-04-17 | 1984-09-25 | Sumitomo Chemical Company, Limited | Fungicidal composition comprising alpha-substituted ethylphosphinic acids or their salts |
| US4466913A (en) * | 1981-06-30 | 1984-08-21 | Maiji Seika Kaisha Ltd. | Phosphorus-containing compounds and process for producing the same |
| US4477391A (en) * | 1981-08-14 | 1984-10-16 | Collins James F | Amino acid isomers, their production and their medicinal use |
| SE455259B (sv) * | 1984-01-30 | 1988-07-04 | Kenogard Ab | Anvendning av vissa aminoalkanfosfonsyror for bekempning av svampsjukdomar hos vexter |
| US5189030A (en) * | 1985-06-11 | 1993-02-23 | Ciba-Geigy Corporation | 1-amino-2-phenylethanephosphonic acids as microbiocides |
| US5143908A (en) * | 1986-11-05 | 1992-09-01 | Merck & Co., Inc. | Antibacterial agents and potentiators of carbapenem antibiotics |
| US5099063A (en) * | 1986-11-05 | 1992-03-24 | Merck & Co., Inc. | Certain phosphinic acid derivatives having antibacterial activity |
| US4761405A (en) * | 1987-03-04 | 1988-08-02 | Nova Pharmaceutical Corporation | Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency |
| US5041644A (en) * | 1987-07-06 | 1991-08-20 | Merck & Co., Inc. | Peptide derivatives of β-chloro-L(Z)-dehydro-glutamic acid |
| JPS6413097A (en) * | 1987-07-06 | 1989-01-17 | Mitsubishi Chem Ind | Phosphonic acid derivative |
| US5030732A (en) * | 1988-03-03 | 1991-07-09 | Merck & Co., Inc. | Aminoethylphosphinic acid derivatives |
| US4962097A (en) * | 1988-10-28 | 1990-10-09 | Merck & Co., Inc. | Method of treating bacterial infection with phosphorus containing DHP enzyme inhibitors |
| US5145990A (en) * | 1988-10-28 | 1992-09-08 | Merck & Co., Inc. | Phosphorous containing dhp enzyme inhibitors |
| US5147867A (en) * | 1988-10-28 | 1992-09-15 | Merck & Co., Inc. | Phosphorus containing enzyme inhibitors |
| US5179173A (en) * | 1991-04-10 | 1993-01-12 | Nalco Chemical Company | Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom |
| FI963390A (fi) * | 1996-08-30 | 1998-03-01 | Khomutov Radii M | Kasvinsuojeluaineet |
| IT201600098005A1 (it) * | 2016-09-29 | 2018-03-29 | Univ Degli Studi Roma La Sapienza | Analoghi e derivati di amminoacidi dicarbossilici come antibatterici |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3160632A (en) * | 1961-01-30 | 1964-12-08 | Stauffer Chemical Co | Aminomethylenephosphinic acids, salts thereof, and process for their production |
| CH475287A (de) * | 1965-10-27 | 1969-07-15 | Monsanto Co | Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren |
| US3424788A (en) * | 1967-07-24 | 1969-01-28 | Armour & Co | Aminophosphinic acids and salts useful as bacteriostats |
-
1976
- 1976-05-21 GB GB21000/76A patent/GB1542938A/en not_active Expired
-
1977
- 1977-05-14 EG EG293/77A patent/EG12688A/xx active
- 1977-05-17 DE DE19772722162 patent/DE2722162A1/de not_active Withdrawn
- 1977-05-18 SE SE7705886A patent/SE7705886L/xx unknown
- 1977-05-18 FR FR7715324A patent/FR2360601A1/fr active Granted
- 1977-05-19 IL IL52127A patent/IL52127A0/xx unknown
- 1977-05-19 FI FI771602A patent/FI771602A/fi not_active Application Discontinuation
- 1977-05-19 DD DD7700199017A patent/DD131751A5/xx unknown
- 1977-05-19 PH PH19791A patent/PH14170A/en unknown
- 1977-05-19 CA CA278,750A patent/CA1081241A/en not_active Expired
- 1977-05-19 BG BG7736361A patent/BG27905A3/xx unknown
- 1977-05-19 BG BG7737259A patent/BG28070A4/xx unknown
- 1977-05-19 ES ES458931A patent/ES458931A1/es not_active Expired
- 1977-05-20 SU SU772484356A patent/SU805948A3/ru active
- 1977-05-20 ZA ZA00773017A patent/ZA773017B/xx unknown
- 1977-05-20 AU AU25319/77A patent/AU516592B2/en not_active Expired
- 1977-05-20 DK DK221477A patent/DK221477A/da unknown
- 1977-05-20 NZ NZ184166A patent/NZ184166A/xx unknown
- 1977-05-20 AT AT361777A patent/AT350585B/de not_active IP Right Cessation
- 1977-05-20 PL PL1977198267A patent/PL110527B1/pl not_active IP Right Cessation
- 1977-05-20 PT PT66581A patent/PT66581B/pt unknown
- 1977-05-20 NO NO771770A patent/NO771770L/no unknown
- 1977-05-20 IE IE1036/77A patent/IE44904B1/en unknown
- 1977-05-20 NL NL7705602A patent/NL7705602A/xx not_active Application Discontinuation
- 1977-05-20 CS CS773353A patent/CS202066B2/cs unknown
- 1977-05-20 BE BE177743A patent/BE854843A/xx not_active IP Right Cessation
- 1977-05-20 PL PL1977209221A patent/PL106608B1/pl unknown
- 1977-05-21 JP JP5823477A patent/JPS52151128A/ja active Pending
- 1977-05-23 US US05/799,428 patent/US4147780A/en not_active Expired - Lifetime
- 1977-05-23 AR AR267742A patent/AR219077A1/es active
- 1977-05-23 OA OA56174A patent/OA05666A/xx unknown
-
1978
- 1978-04-17 AR AR271804A patent/AR222464A1/es active
- 1978-06-09 SU SU782623755A patent/SU795484A3/ru active
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