FR2360601A1 - Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments - Google Patents

Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments

Info

Publication number
FR2360601A1
FR2360601A1 FR7715324A FR7715324A FR2360601A1 FR 2360601 A1 FR2360601 A1 FR 2360601A1 FR 7715324 A FR7715324 A FR 7715324A FR 7715324 A FR7715324 A FR 7715324A FR 2360601 A1 FR2360601 A1 FR 2360601A1
Authority
FR
France
Prior art keywords
phosphoneous
acids
preparation
application
medicinal products
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7715324A
Other languages
English (en)
Other versions
FR2360601B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of FR2360601A1 publication Critical patent/FR2360601A1/fr
Application granted granted Critical
Publication of FR2360601B1 publication Critical patent/FR2360601B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/48—Phosphonous acids R—P(OH)2; Thiophosphonous acids including RHP(=O)(OH); Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings

Abstract

Les composés de l'invention répondent à la formule générale I :
FR7715324A 1976-05-21 1977-05-18 Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments Granted FR2360601A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB21000/76A GB1542938A (en) 1976-05-21 1976-05-21 Aminophosphonous acids and processes for their preparation

Publications (2)

Publication Number Publication Date
FR2360601A1 true FR2360601A1 (fr) 1978-03-03
FR2360601B1 FR2360601B1 (fr) 1979-09-07

Family

ID=10155485

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7715324A Granted FR2360601A1 (fr) 1976-05-21 1977-05-18 Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments

Country Status (29)

Country Link
US (1) US4147780A (fr)
JP (1) JPS52151128A (fr)
AR (2) AR219077A1 (fr)
AT (1) AT350585B (fr)
AU (1) AU516592B2 (fr)
BE (1) BE854843A (fr)
BG (2) BG28070A4 (fr)
CA (1) CA1081241A (fr)
CS (1) CS202066B2 (fr)
DD (1) DD131751A5 (fr)
DE (1) DE2722162A1 (fr)
DK (1) DK221477A (fr)
EG (1) EG12688A (fr)
ES (1) ES458931A1 (fr)
FI (1) FI771602A (fr)
FR (1) FR2360601A1 (fr)
GB (1) GB1542938A (fr)
IE (1) IE44904B1 (fr)
IL (1) IL52127A0 (fr)
NL (1) NL7705602A (fr)
NO (1) NO771770L (fr)
NZ (1) NZ184166A (fr)
OA (1) OA05666A (fr)
PH (1) PH14170A (fr)
PL (2) PL110527B1 (fr)
PT (1) PT66581B (fr)
SE (1) SE7705886L (fr)
SU (2) SU805948A3 (fr)
ZA (1) ZA773017B (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002031B1 (fr) * 1977-11-19 1982-02-03 Ciba-Geigy Ag Procédé pour inhiber la croissance des plantes et pour combattre les mauvaises herbes par utilisation des acides alpha-aminoalcanephosphoneux
EP0002039A1 (fr) * 1977-11-19 1979-05-30 Ciba-Geigy Ag Dérivés d'acides phosphoneux, procédés pour leur préparation et leur utilisation dans la lutte contre les micro-organismes
IL61985A0 (en) * 1980-02-01 1981-02-27 Sparamedica Ag Phosphinic and phosphonic acid derivatives,their manufacture and pharmaceutical compositions containing them
US4473561A (en) * 1981-04-17 1984-09-25 Sumitomo Chemical Company, Limited Fungicidal composition comprising alpha-substituted ethylphosphinic acids or their salts
US4466913A (en) * 1981-06-30 1984-08-21 Maiji Seika Kaisha Ltd. Phosphorus-containing compounds and process for producing the same
US4477391A (en) * 1981-08-14 1984-10-16 Collins James F Amino acid isomers, their production and their medicinal use
SE455259B (sv) * 1984-01-30 1988-07-04 Kenogard Ab Anvendning av vissa aminoalkanfosfonsyror for bekempning av svampsjukdomar hos vexter
US5189030A (en) * 1985-06-11 1993-02-23 Ciba-Geigy Corporation 1-amino-2-phenylethanephosphonic acids as microbiocides
US5143908A (en) * 1986-11-05 1992-09-01 Merck & Co., Inc. Antibacterial agents and potentiators of carbapenem antibiotics
US5099063A (en) * 1986-11-05 1992-03-24 Merck & Co., Inc. Certain phosphinic acid derivatives having antibacterial activity
US4761405A (en) * 1987-03-04 1988-08-02 Nova Pharmaceutical Corporation Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency
JPS6413097A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Phosphonic acid derivative
US5041644A (en) * 1987-07-06 1991-08-20 Merck & Co., Inc. Peptide derivatives of β-chloro-L(Z)-dehydro-glutamic acid
US5030732A (en) * 1988-03-03 1991-07-09 Merck & Co., Inc. Aminoethylphosphinic acid derivatives
US5147867A (en) * 1988-10-28 1992-09-15 Merck & Co., Inc. Phosphorus containing enzyme inhibitors
US5145990A (en) * 1988-10-28 1992-09-08 Merck & Co., Inc. Phosphorous containing dhp enzyme inhibitors
US4962097A (en) * 1988-10-28 1990-10-09 Merck & Co., Inc. Method of treating bacterial infection with phosphorus containing DHP enzyme inhibitors
US5179173A (en) * 1991-04-10 1993-01-12 Nalco Chemical Company Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom
FI963390A (fi) * 1996-08-30 1998-03-01 Khomutov Radii M Kasvinsuojeluaineet
IT201600098005A1 (it) * 2016-09-29 2018-03-29 Univ Degli Studi Roma La Sapienza Analoghi e derivati di amminoacidi dicarbossilici come antibatterici

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH475287A (de) * 1965-10-27 1969-07-15 Monsanto Co Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3160632A (en) * 1961-01-30 1964-12-08 Stauffer Chemical Co Aminomethylenephosphinic acids, salts thereof, and process for their production
US3424788A (en) * 1967-07-24 1969-01-28 Armour & Co Aminophosphinic acids and salts useful as bacteriostats

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH475287A (de) * 1965-10-27 1969-07-15 Monsanto Co Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren

Also Published As

Publication number Publication date
PH14170A (en) 1981-03-19
PL110527B1 (en) 1980-07-31
CA1081241A (fr) 1980-07-08
ZA773017B (en) 1978-04-26
NO771770L (no) 1977-11-22
EG12688A (en) 1979-06-30
FI771602A (fr) 1977-11-22
JPS52151128A (en) 1977-12-15
AU516592B2 (en) 1981-06-11
PL198267A1 (pl) 1978-03-13
GB1542938A (en) 1979-03-28
SE7705886L (sv) 1977-11-22
PL106608B1 (pl) 1980-01-31
ATA361777A (de) 1978-11-15
BE854843A (fr) 1977-11-21
AT350585B (de) 1979-06-11
PT66581A (en) 1977-06-01
AU2531977A (en) 1978-11-23
ES458931A1 (es) 1978-03-01
CS202066B2 (en) 1980-12-31
BG27905A3 (en) 1980-01-15
IE44904B1 (en) 1982-05-05
AR222464A1 (es) 1981-05-29
NZ184166A (en) 1980-03-05
FR2360601B1 (fr) 1979-09-07
IE44904L (en) 1977-11-21
OA05666A (fr) 1981-05-31
DE2722162A1 (de) 1977-12-01
NL7705602A (nl) 1977-11-23
IL52127A0 (en) 1977-07-31
DD131751A5 (de) 1978-07-19
PT66581B (en) 1978-10-20
SU795484A3 (ru) 1981-01-07
BG28070A4 (en) 1980-02-25
US4147780A (en) 1979-04-03
AR219077A1 (es) 1980-07-31
DK221477A (da) 1977-11-22
SU805948A3 (ru) 1981-02-15

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Legal Events

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