BE854843A - Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments - Google Patents

Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments

Info

Publication number
BE854843A
BE854843A BE177743A BE177743A BE854843A BE 854843 A BE854843 A BE 854843A BE 177743 A BE177743 A BE 177743A BE 177743 A BE177743 A BE 177743A BE 854843 A BE854843 A BE 854843A
Authority
BE
Belgium
Prior art keywords
phosphoneous
preparation
new
application
acid derivatives
Prior art date
Application number
BE177743A
Other languages
English (en)
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of BE854843A publication Critical patent/BE854843A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/48Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/58Pyridine rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
BE177743A 1976-05-21 1977-05-20 Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments BE854843A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB21000/76A GB1542938A (en) 1976-05-21 1976-05-21 Aminophosphonous acids and processes for their preparation

Publications (1)

Publication Number Publication Date
BE854843A true BE854843A (fr) 1977-11-21

Family

ID=10155485

Family Applications (1)

Application Number Title Priority Date Filing Date
BE177743A BE854843A (fr) 1976-05-21 1977-05-20 Nouveaux derives d'acides phosphoneux, leur preparation et leur application en tant que medicaments

Country Status (29)

Country Link
US (1) US4147780A (fr)
JP (1) JPS52151128A (fr)
AR (2) AR219077A1 (fr)
AT (1) AT350585B (fr)
AU (1) AU516592B2 (fr)
BE (1) BE854843A (fr)
BG (2) BG28070A4 (fr)
CA (1) CA1081241A (fr)
CS (1) CS202066B2 (fr)
DD (1) DD131751A5 (fr)
DE (1) DE2722162A1 (fr)
DK (1) DK221477A (fr)
EG (1) EG12688A (fr)
ES (1) ES458931A1 (fr)
FI (1) FI771602A (fr)
FR (1) FR2360601A1 (fr)
GB (1) GB1542938A (fr)
IE (1) IE44904B1 (fr)
IL (1) IL52127A0 (fr)
NL (1) NL7705602A (fr)
NO (1) NO771770L (fr)
NZ (1) NZ184166A (fr)
OA (1) OA05666A (fr)
PH (1) PH14170A (fr)
PL (2) PL106608B1 (fr)
PT (1) PT66581B (fr)
SE (1) SE7705886L (fr)
SU (2) SU805948A3 (fr)
ZA (1) ZA773017B (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002039A1 (fr) * 1977-11-19 1979-05-30 Ciba-Geigy Ag Dérivés d'acides phosphoneux, procédés pour leur préparation et leur utilisation dans la lutte contre les micro-organismes
EP0002031B1 (fr) * 1977-11-19 1982-02-03 Ciba-Geigy Ag Procédé pour inhiber la croissance des plantes et pour combattre les mauvaises herbes par utilisation des acides alpha-aminoalcanephosphoneux
IL61985A0 (en) * 1980-02-01 1981-02-27 Sparamedica Ag Phosphinic and phosphonic acid derivatives,their manufacture and pharmaceutical compositions containing them
US4473561A (en) * 1981-04-17 1984-09-25 Sumitomo Chemical Company, Limited Fungicidal composition comprising alpha-substituted ethylphosphinic acids or their salts
US4466913A (en) * 1981-06-30 1984-08-21 Maiji Seika Kaisha Ltd. Phosphorus-containing compounds and process for producing the same
US4477391A (en) * 1981-08-14 1984-10-16 Collins James F Amino acid isomers, their production and their medicinal use
SE455259B (sv) * 1984-01-30 1988-07-04 Kenogard Ab Anvendning av vissa aminoalkanfosfonsyror for bekempning av svampsjukdomar hos vexter
US5189030A (en) * 1985-06-11 1993-02-23 Ciba-Geigy Corporation 1-amino-2-phenylethanephosphonic acids as microbiocides
US5143908A (en) * 1986-11-05 1992-09-01 Merck & Co., Inc. Antibacterial agents and potentiators of carbapenem antibiotics
US5099063A (en) * 1986-11-05 1992-03-24 Merck & Co., Inc. Certain phosphinic acid derivatives having antibacterial activity
US4761405A (en) * 1987-03-04 1988-08-02 Nova Pharmaceutical Corporation Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency
JPS6413097A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Phosphonic acid derivative
US5041644A (en) * 1987-07-06 1991-08-20 Merck & Co., Inc. Peptide derivatives of β-chloro-L(Z)-dehydro-glutamic acid
US5030732A (en) * 1988-03-03 1991-07-09 Merck & Co., Inc. Aminoethylphosphinic acid derivatives
US5147867A (en) * 1988-10-28 1992-09-15 Merck & Co., Inc. Phosphorus containing enzyme inhibitors
US4962097A (en) * 1988-10-28 1990-10-09 Merck & Co., Inc. Method of treating bacterial infection with phosphorus containing DHP enzyme inhibitors
US5145990A (en) * 1988-10-28 1992-09-08 Merck & Co., Inc. Phosphorous containing dhp enzyme inhibitors
US5179173A (en) * 1991-04-10 1993-01-12 Nalco Chemical Company Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom
FI963390A (fi) * 1996-08-30 1998-03-01 Khomutov Radii M Kasvinsuojeluaineet
IT201600098005A1 (it) * 2016-09-29 2018-03-29 Univ Degli Studi Roma La Sapienza Analoghi e derivati di amminoacidi dicarbossilici come antibatterici

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3160632A (en) * 1961-01-30 1964-12-08 Stauffer Chemical Co Aminomethylenephosphinic acids, salts thereof, and process for their production
CH475287A (de) * 1965-10-27 1969-07-15 Monsanto Co Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren
US3424788A (en) * 1967-07-24 1969-01-28 Armour & Co Aminophosphinic acids and salts useful as bacteriostats

Also Published As

Publication number Publication date
CA1081241A (fr) 1980-07-08
ZA773017B (en) 1978-04-26
PT66581B (en) 1978-10-20
AU2531977A (en) 1978-11-23
AR222464A1 (es) 1981-05-29
NL7705602A (nl) 1977-11-23
ATA361777A (de) 1978-11-15
FR2360601A1 (fr) 1978-03-03
PT66581A (en) 1977-06-01
NO771770L (no) 1977-11-22
PL198267A1 (pl) 1978-03-13
PL106608B1 (pl) 1980-01-31
CS202066B2 (en) 1980-12-31
AT350585B (de) 1979-06-11
EG12688A (en) 1979-06-30
SE7705886L (sv) 1977-11-22
DK221477A (da) 1977-11-22
IE44904L (en) 1977-11-21
SU795484A3 (ru) 1981-01-07
FR2360601B1 (fr) 1979-09-07
BG28070A4 (en) 1980-02-25
PH14170A (en) 1981-03-19
IL52127A0 (en) 1977-07-31
PL110527B1 (en) 1980-07-31
US4147780A (en) 1979-04-03
IE44904B1 (en) 1982-05-05
ES458931A1 (es) 1978-03-01
BG27905A3 (en) 1980-01-15
AU516592B2 (en) 1981-06-11
SU805948A3 (ru) 1981-02-15
DE2722162A1 (de) 1977-12-01
GB1542938A (en) 1979-03-28
AR219077A1 (es) 1980-07-31
OA05666A (fr) 1981-05-31
JPS52151128A (en) 1977-12-15
DD131751A5 (de) 1978-07-19
NZ184166A (en) 1980-03-05
FI771602A (fr) 1977-11-22

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: CIBA-GEIGY A.G.

Effective date: 19920531