CS200205B2 - Method of producing aminocyclols - Google Patents

Method of producing aminocyclols Download PDF

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Publication number
CS200205B2
CS200205B2 CS77170A CS17077A CS200205B2 CS 200205 B2 CS200205 B2 CS 200205B2 CS 77170 A CS77170 A CS 77170A CS 17077 A CS17077 A CS 17077A CS 200205 B2 CS200205 B2 CS 200205B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
compounds
nitro
methylene chloride
methyl
Prior art date
Application number
CS77170A
Other languages
Czech (cs)
English (en)
Inventor
Paul Stadler
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of CS200205B2 publication Critical patent/CS200205B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/081—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS77170A 1976-01-12 1977-01-11 Method of producing aminocyclols CS200205B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH26976A CH619468A5 (ko) 1976-01-12 1976-01-12

Publications (1)

Publication Number Publication Date
CS200205B2 true CS200205B2 (en) 1980-08-29

Family

ID=4183149

Family Applications (1)

Application Number Title Priority Date Filing Date
CS77170A CS200205B2 (en) 1976-01-12 1977-01-11 Method of producing aminocyclols

Country Status (22)

Country Link
US (1) US4145549A (ko)
JP (1) JPS5287197A (ko)
AT (1) AT364817B (ko)
AU (1) AU512003B2 (ko)
BE (1) BE850304A (ko)
CA (1) CA1108128A (ko)
CH (1) CH619468A5 (ko)
CS (1) CS200205B2 (ko)
DE (1) DE2700234A1 (ko)
DK (1) DK150490C (ko)
ES (1) ES454917A1 (ko)
FI (1) FI62094C (ko)
FR (1) FR2337727A1 (ko)
GB (1) GB1571835A (ko)
HU (1) HU176871B (ko)
IE (1) IE44560B1 (ko)
NL (1) NL7700124A (ko)
NZ (1) NZ183045A (ko)
SE (1) SE434401B (ko)
SU (1) SU725565A3 (ko)
YU (1) YU39377B (ko)
ZA (1) ZA77151B (ko)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1584464A (en) * 1977-04-19 1981-02-11 Farmaceutici Italia Ergot alkaloids
JPS5423487U (ko) * 1977-07-19 1979-02-15
EP0003286B1 (de) * 1978-01-20 1982-03-24 Sandoz Ag Ergopeptidalkaloid-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
YU41110B (en) * 1978-07-19 1986-12-31 Lek Tovarna Farmacevtskih Process for preparing dextrorotatory ergot alcaloids acid addition salts
DE3303616A1 (de) * 1982-02-12 1983-08-25 Sandoz-Patent-GmbH, 7850 Lörrach Mutterkornalkaloide, verfahren zu deren herstellung sowie diese verbindungen enthaltende pharmazeutische zubereitungen
RU2266906C1 (ru) * 2004-04-29 2005-12-27 Общество с ограниченной ответственностью "Исследовательский Институт Химического Разнообразия" (ООО "Исследовательский Институт Химического Разнообразия") Анелированные карбамоилазагетероциклы, способы их получения (варианты), фармацевтическая композиция, фокусированная библиотека
US20080161324A1 (en) * 2006-09-14 2008-07-03 Johansen Lisa M Compositions and methods for treatment of viral diseases

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2533698A (en) * 1950-12-12 Urethanes containing the lysergic
CH507249A (de) * 1968-05-31 1971-05-15 Sandoz Ag Verfahren zur Herstellung von 2-Brom-a-ergokryptin
GB1298277A (en) * 1969-04-18 1972-11-29 Sandoz Ltd Preparation of ergot peptide alkaloids
JPS4735440A (ko) * 1971-03-29 1972-11-25
CH581136A5 (ko) * 1972-09-26 1976-10-29 Sandoz Ag
FI56386C (fi) * 1973-07-09 1980-01-10 Sandoz Ag Foerfarande foer framstaellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazin-derivat
CH587858A5 (ko) * 1973-11-28 1977-05-13 Sandoz Ag
DE2525962A1 (de) * 1974-06-21 1976-01-08 Sandoz Ag Neue heterocyclische verbindungen, ihre herstellung und verwendung
CH601321A5 (ko) * 1975-01-06 1978-07-14 Sandoz Ag

Also Published As

Publication number Publication date
HU176871B (en) 1981-05-28
ATA8777A (de) 1981-04-15
CA1108128A (en) 1981-09-01
SE434401B (sv) 1984-07-23
FI62094B (fi) 1982-07-30
DK150490C (da) 1987-10-19
FI62094C (fi) 1982-11-10
ZA77151B (en) 1978-08-30
FI770008A (ko) 1977-07-13
JPS5287197A (en) 1977-07-20
ES454917A1 (es) 1978-04-01
DK577A (da) 1977-07-13
FR2337727B1 (ko) 1980-04-30
GB1571835A (en) 1980-07-23
CH619468A5 (ko) 1980-09-30
AU2122877A (en) 1978-07-20
IE44560L (en) 1977-07-12
DK150490B (da) 1987-03-09
YU6277A (en) 1982-10-31
NZ183045A (en) 1979-03-16
FR2337727A1 (fr) 1977-08-05
AT364817B (de) 1981-11-25
BE850304A (fr) 1977-07-12
NL7700124A (nl) 1977-07-14
YU39377B (en) 1984-12-31
AU512003B2 (en) 1980-09-18
US4145549A (en) 1979-03-20
SU725565A3 (ru) 1980-03-30
DE2700234A1 (de) 1977-07-14
IE44560B1 (en) 1982-01-13

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