CS197285B2 - Process for preparing carboxyalkylacylaminoacids - Google Patents

Process for preparing carboxyalkylacylaminoacids Download PDF

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Publication number
CS197285B2
CS197285B2 CS77926A CS92677A CS197285B2 CS 197285 B2 CS197285 B2 CS 197285B2 CS 77926 A CS77926 A CS 77926A CS 92677 A CS92677 A CS 92677A CS 197285 B2 CS197285 B2 CS 197285B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
compound
proline
apos
reacted
Prior art date
Application number
CS77926A
Other languages
Czech (cs)
English (en)
Inventor
David W Cushman
Original Assignee
Ondetti Miguel A
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ondetti Miguel A, Squibb & Sons Inc filed Critical Ondetti Miguel A
Publication of CS197285B2 publication Critical patent/CS197285B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS77926A 1976-02-13 1977-02-11 Process for preparing carboxyalkylacylaminoacids CS197285B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/657,793 US4052511A (en) 1976-02-13 1976-02-13 Carboxyacylproline derivatives

Publications (1)

Publication Number Publication Date
CS197285B2 true CS197285B2 (en) 1980-04-30

Family

ID=24638684

Family Applications (1)

Application Number Title Priority Date Filing Date
CS77926A CS197285B2 (en) 1976-02-13 1977-02-11 Process for preparing carboxyalkylacylaminoacids

Country Status (23)

Country Link
US (3) US4052511A (no)
JP (1) JPS6058751B2 (no)
AT (1) AT366030B (no)
BE (1) BE851363A (no)
CA (1) CA1104059A (no)
CH (1) CH602633A5 (no)
CS (1) CS197285B2 (no)
DD (1) DD129651A5 (no)
DE (1) DE2704985A1 (no)
DK (1) DK59077A (no)
FR (1) FR2340933A1 (no)
GB (1) GB1570921A (no)
HU (1) HU177144B (no)
IE (1) IE45086B1 (no)
NL (1) NL167688C (no)
NO (1) NO145915C (no)
NZ (1) NZ183222A (no)
PH (1) PH12066A (no)
PL (1) PL106416B1 (no)
SE (1) SE426169B (no)
SU (1) SU694070A3 (no)
YU (1) YU33277A (no)
ZA (1) ZA77564B (no)

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Also Published As

Publication number Publication date
AT366030B (de) 1982-03-10
ATA96977A (de) 1981-07-15
NO145915C (no) 1982-06-23
FR2340933B1 (no) 1980-04-11
PH12066A (en) 1978-10-18
SE7701562L (sv) 1977-09-23
NO770465L (no) 1977-08-16
US4086338A (en) 1978-04-25
US4052511A (en) 1977-10-04
GB1570921A (en) 1980-07-09
NL167688C (nl) 1982-01-18
PL106416B1 (pl) 1979-12-31
JPS52100461A (en) 1977-08-23
DD129651A5 (de) 1978-02-01
IE45086L (en) 1977-08-13
US4128653A (en) 1978-12-05
FR2340933A1 (fr) 1977-09-09
SE426169B (sv) 1982-12-13
NL7701463A (nl) 1977-08-16
YU33277A (en) 1982-08-31
JPS6058751B2 (ja) 1985-12-21
DE2704985A1 (de) 1977-08-18
HU177144B (en) 1981-07-28
DK59077A (da) 1977-08-14
ZA77564B (en) 1977-12-28
BE851363A (fr) 1977-08-11
NL167688B (nl) 1981-08-17
IE45086B1 (en) 1982-06-16
SU694070A3 (ru) 1979-10-25
NO145915B (no) 1982-03-15
CA1104059A (en) 1981-06-30
CH602633A5 (no) 1978-07-31
PL195997A1 (pl) 1978-02-27
NZ183222A (en) 1979-07-11
AU2189877A (en) 1978-08-10

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