CS195744B2 - Method of producing new derivatives of imidazole - Google Patents

Method of producing new derivatives of imidazole Download PDF

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Publication number
CS195744B2
CS195744B2 CS767763A CS776376A CS195744B2 CS 195744 B2 CS195744 B2 CS 195744B2 CS 767763 A CS767763 A CS 767763A CS 776376 A CS776376 A CS 776376A CS 195744 B2 CS195744 B2 CS 195744B2
Authority
CS
Czechoslovakia
Prior art keywords
carbon atoms
alkyl
group
imidazole
formula
Prior art date
Application number
CS767763A
Other languages
Czech (cs)
English (en)
Inventor
David A Cox
Geoffrey E Gymer
Braham Shroot
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS195744B2 publication Critical patent/CS195744B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CS767763A 1975-12-04 1976-11-30 Method of producing new derivatives of imidazole CS195744B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49797/75A GB1511390A (en) 1975-12-04 1975-12-04 Imidazolylalkyl sulphide antifungal agents

Publications (1)

Publication Number Publication Date
CS195744B2 true CS195744B2 (en) 1980-02-29

Family

ID=10453567

Family Applications (1)

Application Number Title Priority Date Filing Date
CS767763A CS195744B2 (en) 1975-12-04 1976-11-30 Method of producing new derivatives of imidazole

Country Status (34)

Country Link
US (1) US4107314A (nl)
JP (1) JPS5277062A (nl)
AR (1) AR223634A1 (nl)
AT (1) AT354435B (nl)
AU (1) AU504085B2 (nl)
BE (1) BE849012A (nl)
BG (1) BG28261A3 (nl)
CA (1) CA1056380A (nl)
CH (1) CH599163A5 (nl)
CS (1) CS195744B2 (nl)
DD (1) DD127186A5 (nl)
DE (1) DE2654665C3 (nl)
DK (1) DK545076A (nl)
EG (1) EG12483A (nl)
ES (1) ES453867A1 (nl)
FI (1) FI62300C (nl)
FR (1) FR2333506A1 (nl)
GB (1) GB1511390A (nl)
GR (1) GR61774B (nl)
HU (1) HU177882B (nl)
IE (1) IE44105B1 (nl)
IL (1) IL50869A (nl)
LU (1) LU76326A1 (nl)
NL (1) NL165463C (nl)
NO (1) NO145791C (nl)
NZ (1) NZ182565A (nl)
PH (1) PH14175A (nl)
PL (1) PL104366B1 (nl)
PT (1) PT65904B (nl)
RO (1) RO72349A (nl)
SE (1) SE423544C (nl)
SU (1) SU635871A3 (nl)
YU (1) YU40157B (nl)
ZA (1) ZA766280B (nl)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0001654B1 (de) * 1977-10-13 1981-07-22 Siegfried Aktiengesellschaft Imidazolyläthyl-oxyalkoxy-Derivate und ihre Thio-Analoge, pharmazeutische Zubereitungen mit diesen Stoffen und Verfahren zu ihrer Herstellung
DE2756269A1 (de) * 1977-12-16 1979-06-21 Bayer Ag Azolylalkyl-pyridinyl-aether, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide
US4343805A (en) * 1978-12-16 1982-08-10 John Wyeth & Brother Limited Heterocyclic compounds
US4272545A (en) * 1979-02-02 1981-06-09 Syntex (U.S.A.) Inc. Derivatives of thienyl- and furyl-substituted N-butyl and N-phenyl imidazoles
US4307105A (en) 1979-07-05 1981-12-22 E. R. Squibb & Sons, Inc. Imidazolylethoxymethyl derivatives of thiazole
US4248881A (en) * 1979-12-20 1981-02-03 E. R. Squibb & Sons, Inc. Imidazolylethoxymethyl derivatives of pyrazole
CA1155853A (en) * 1980-06-06 1983-10-25 Joseph A. Martin Imidazole derivatives and preparation thereof
US4458079A (en) * 1980-08-08 1984-07-03 Bristol-Myers Company Sulfur-containing imidazoles
IN158970B (nl) * 1981-06-09 1987-02-28 Ici Plc
GB8308601D0 (en) * 1983-03-29 1983-05-05 Ici Plc Heterocyclic compounds
GB2161160B (en) * 1984-07-06 1989-05-24 Fisons Plc Heterocyclic sulphinyl compounds
US4661602A (en) * 1985-03-29 1987-04-28 G. D. Searle & Co. Substituted alkyl imidazole derivatives
US4628104A (en) * 1985-04-08 1986-12-09 G. D. Searle & Co. Imidazole ketone derivatives
US4761483A (en) * 1985-06-26 1988-08-02 G. D. Searle & Co. Chloro-substituted ketone imidazole derivatives
AT389874B (de) * 1988-04-29 1990-02-12 Agrolinz Agrarchemikalien Neue pyridyl-thio-ethylazole, verfahren zu deren herstellung und diese enthaltende fungizide mittel
US6545163B1 (en) * 1995-10-02 2003-04-08 Napp Technologies Process to prepare 1-aryl-2-(1-imidazolyl) alkyl ethers and thioethers
DE10130706A1 (de) 2001-06-26 2003-01-02 Bayer Ag Thiazine und Thiazole als Materialschutzmittel

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU557755A3 (ru) * 1968-08-19 1977-05-05 Янссен Фармасьютика Н.В. (Фирма) Способ получени производных имидазола
GB1475271A (en) * 1975-04-30 1977-06-01 Pfizer Ltd 1-aryl-2-1-imidazolyl-alkyl ethers and thioethers and their use as antifungal agents

Also Published As

Publication number Publication date
IL50869A (en) 1980-06-30
DE2654665B2 (de) 1981-05-07
NL165463C (nl) 1981-04-15
RO72349A (ro) 1981-08-30
ZA766280B (en) 1977-09-28
NO145791B (no) 1982-02-22
NO764134L (nl) 1977-06-07
EG12483A (en) 1979-03-31
FI763471A (nl) 1977-06-05
CH599163A5 (nl) 1978-05-12
US4107314A (en) 1978-08-15
IE44105B1 (en) 1981-08-12
SU635871A3 (ru) 1978-11-30
PH14175A (en) 1981-03-19
NZ182565A (en) 1978-04-03
ES453867A1 (es) 1977-11-01
DE2654665C3 (de) 1982-04-22
JPS5745438B2 (nl) 1982-09-28
NL165463B (nl) 1980-11-17
BG28261A3 (en) 1980-03-25
SE423544C (sv) 1986-09-08
PT65904A (fr) 1976-12-01
GR61774B (en) 1979-01-16
YU281676A (en) 1982-10-31
DK545076A (da) 1977-06-05
NO145791C (no) 1982-06-02
FR2333506A1 (fr) 1977-07-01
PT65904B (fr) 1978-07-05
AU1968876A (en) 1978-05-25
JPS5277062A (en) 1977-06-29
SE7613615L (sv) 1977-06-05
AT354435B (de) 1979-01-10
LU76326A1 (nl) 1978-07-10
AU504085B2 (en) 1979-10-04
HU177882B (en) 1982-01-28
SE423544B (sv) 1982-05-10
ATA889476A (de) 1979-06-15
IE44105L (en) 1977-06-04
PL104366B1 (pl) 1979-08-31
AR223634A1 (es) 1981-09-15
FR2333506B1 (nl) 1980-11-07
YU40157B (en) 1985-08-31
BE849012A (fr) 1977-06-02
IL50869A0 (en) 1977-01-31
FI62300C (fi) 1982-12-10
FI62300B (fi) 1982-08-31
GB1511390A (en) 1978-05-17
DD127186A5 (nl) 1977-09-07
NL7613425A (nl) 1977-06-07
DE2654665A1 (de) 1977-06-08
CA1056380A (en) 1979-06-12

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