CO7160002A2 - Métodos para preparar triazolopiridinas sustituidas - Google Patents

Métodos para preparar triazolopiridinas sustituidas

Info

Publication number
CO7160002A2
CO7160002A2 CO15004251A CO15004251A CO7160002A2 CO 7160002 A2 CO7160002 A2 CO 7160002A2 CO 15004251 A CO15004251 A CO 15004251A CO 15004251 A CO15004251 A CO 15004251A CO 7160002 A2 CO7160002 A2 CO 7160002A2
Authority
CO
Colombia
Prior art keywords
methods
preparing substituted
substituted triazolopyridines
preparing
triazolopyridines
Prior art date
Application number
CO15004251A
Other languages
English (en)
Spanish (es)
Inventor
Volker Klaus Schulze
Franz Josef Mais
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CO7160002A2 publication Critical patent/CO7160002A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CO15004251A 2012-07-10 2015-01-09 Métodos para preparar triazolopiridinas sustituidas CO7160002A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12175640 2012-07-10
EP12185590 2012-09-24
EP13170585 2013-06-05

Publications (1)

Publication Number Publication Date
CO7160002A2 true CO7160002A2 (es) 2015-01-15

Family

ID=48793197

Family Applications (1)

Application Number Title Priority Date Filing Date
CO15004251A CO7160002A2 (es) 2012-07-10 2015-01-09 Métodos para preparar triazolopiridinas sustituidas

Country Status (24)

Country Link
US (1) US9388177B2 (OSRAM)
EP (1) EP2872506A1 (OSRAM)
JP (1) JP6238979B2 (OSRAM)
KR (1) KR20150040845A (OSRAM)
CN (1) CN104603136B (OSRAM)
AP (1) AP3778A (OSRAM)
AU (1) AU2013289381A1 (OSRAM)
BR (1) BR112015000308A2 (OSRAM)
CA (1) CA2878481A1 (OSRAM)
CL (1) CL2015000038A1 (OSRAM)
CO (1) CO7160002A2 (OSRAM)
CR (1) CR20150006A (OSRAM)
DO (1) DOP2015000007A (OSRAM)
EA (1) EA027544B1 (OSRAM)
HK (1) HK1206731A1 (OSRAM)
IL (1) IL236265A (OSRAM)
IN (1) IN2015DN00085A (OSRAM)
MX (1) MX2015000348A (OSRAM)
NZ (1) NZ703020A (OSRAM)
PE (1) PE20150354A1 (OSRAM)
PH (1) PH12015500061A1 (OSRAM)
SG (1) SG11201408419QA (OSRAM)
TN (1) TN2015000008A1 (OSRAM)
WO (1) WO2014009219A1 (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105431435A (zh) * 2013-06-07 2016-03-23 拜耳制药股份公司 具有作为mps-1抑制剂的活性的取代的三唑并吡啶类
TN2015000545A1 (en) * 2013-06-11 2017-04-06 Bayer Pharma AG Prodrug derivatives of substituted triazolopyridines
US20160128988A1 (en) 2013-06-11 2016-05-12 Bayer Pharma Aktiengesellschaft Combinations for the treatment of cancer comprising a mps-1 kinase inhibitor and a mitotic inhibitor
EP3283642B1 (en) 2015-04-17 2023-10-11 Netherlands Translational Research Center Holding B.V. Prognostic biomarkers for ttk inhibitor chemotherapy
TW201800408A (zh) 2016-06-15 2018-01-01 拜耳製藥公司 Mps-1抑制劑

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050009812A1 (en) * 2001-10-05 2005-01-13 Takuya Seko Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
MXPA06013250A (es) * 2004-05-14 2007-02-28 Abbott Lab Inhibidores de quinasa como agentes terapeuticos.
UA89503C2 (uk) * 2004-09-13 2010-02-10 Х. Луннбек А/С Заміщені похідні аніліну
BRPI0516819A (pt) * 2004-10-07 2008-09-23 Warner Lambert Co derivados de triazolopiridina e agentes antibacterianos
US20060194823A1 (en) * 2004-12-22 2006-08-31 Georg Kettschau Sulfonamido-macrocycles as Tie2 inhibitors and the salts thereof, a pharmaceutical composition comprising these compounds, the method of preparing and the use thereof
CN101516883A (zh) * 2006-06-06 2009-08-26 先灵公司 作为蛋白激酶抑制剂的咪唑并吡嗪化合物
EP1870416A1 (en) * 2006-06-21 2007-12-26 Bayer Schering Pharma Aktiengesellschaft Sulphonamido-macrocycles as tie2 inhibitors
EP2057158B8 (en) 2006-08-30 2015-09-30 Cellzome Limited Triazole derivatives as kinase inhibitors
JO3598B1 (ar) * 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
CA2693232A1 (en) 2007-07-18 2009-01-22 Novartis Ag Bicyclic heteroaryl compounds and their use as kinase inhibitors
EP2212326A1 (en) 2007-08-23 2010-08-04 AstraZeneca AB 2-anilinopurin-8-ones as inhibitors of ttk/mps1 for the treatment of proliferative disorders
EA201070328A1 (ru) 2007-08-31 2010-08-30 Мерк Сероно С.А. Соединения триазолопиридина и их применение в качестве ингибиторов ask
GB0719803D0 (en) 2007-10-10 2007-11-21 Cancer Rec Tech Ltd Therapeutic compounds and their use
GB0724342D0 (en) * 2007-12-13 2008-01-30 Prolysis Ltd Anitbacterial compositions
WO2009137322A2 (en) * 2008-05-05 2009-11-12 The Trustees Of The University Of Pennsylvania Processes for the preparation of biphenyl compounds
WO2009155527A2 (en) * 2008-06-19 2009-12-23 Progenics Pharmaceuticals, Inc. Phosphatidylinositol 3 kinase inhibitors
EP2396324A1 (en) 2009-02-13 2011-12-21 Fovea Pharmaceuticals Ý1, 2, 4¨triazolo ý1, 5 -a¨pyridines as kinase inhibitors
EP2424537B1 (en) 2009-04-29 2015-07-08 Bayer Intellectual Property GmbH Substituted imidazoquinoxalines
WO2010141360A1 (en) * 2009-06-05 2010-12-09 Merck Sharp & Dohme Corp. Biaryl benzotriazole derivatives
EP2438066A2 (en) * 2009-06-05 2012-04-11 Cephalon, Inc. PREPARATION AND USES OF 1,2,4-TRIAZOLO [1,5a]PYRIDINE DERIVATIVES
EP2473498A1 (en) 2009-09-04 2012-07-11 Bayer Pharma Aktiengesellschaft Substituted aminoquinoxalines as tyrosine threonine kinase inhibitors
EP2343294A1 (en) * 2009-11-30 2011-07-13 Bayer Schering Pharma AG Substituted triazolopyridines
EP2343295A1 (en) * 2009-11-30 2011-07-13 Bayer Schering Pharma AG Triazolopyridine derivates
EP2343297A1 (en) * 2009-11-30 2011-07-13 Bayer Schering Pharma AG Triazolopyridines
UY33452A (es) * 2010-06-16 2012-01-31 Bayer Schering Pharma Ag Triazolopiridinas sustituidas
WO2012044567A2 (en) * 2010-09-30 2012-04-05 Merck Sharp & Dohme Corp. Imidazole derivatives
CA2833657A1 (en) * 2011-04-21 2012-10-26 Bayer Intellectual Property Gmbh Triazolopyridines
WO2012160029A1 (en) * 2011-05-23 2012-11-29 Bayer Intellectual Property Gmbh Substituted triazolopyridines
UA112096C2 (uk) * 2011-12-12 2016-07-25 Байєр Інтеллектуал Проперті Гмбх Заміщені триазолопіридини та їх застосування як інгібіторів ttk

Also Published As

Publication number Publication date
CN104603136B (zh) 2017-06-27
MX2015000348A (es) 2015-04-14
AP2014008177A0 (en) 2014-12-31
AU2013289381A1 (en) 2015-01-22
SG11201408419QA (en) 2015-01-29
US20150148542A1 (en) 2015-05-28
DOP2015000007A (es) 2015-02-15
TN2015000008A1 (en) 2016-06-29
AP3778A (en) 2016-08-31
EA027544B1 (ru) 2017-08-31
PE20150354A1 (es) 2015-03-21
IL236265A0 (en) 2015-02-26
CL2015000038A1 (es) 2015-03-13
NZ703020A (en) 2017-08-25
CA2878481A1 (en) 2014-01-16
JP2015523372A (ja) 2015-08-13
WO2014009219A1 (en) 2014-01-16
HK1206731A1 (en) 2016-01-15
EP2872506A1 (en) 2015-05-20
IN2015DN00085A (OSRAM) 2015-05-29
US9388177B2 (en) 2016-07-12
KR20150040845A (ko) 2015-04-15
CR20150006A (es) 2015-02-16
PH12015500061A1 (en) 2015-03-02
BR112015000308A2 (pt) 2017-06-27
CN104603136A (zh) 2015-05-06
EA201590116A1 (ru) 2015-07-30
JP6238979B2 (ja) 2017-11-29
IL236265A (en) 2017-07-31

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