MX2007004179A - Derivados de triazolpiridina como agentes antibacterianos. - Google Patents

Derivados de triazolpiridina como agentes antibacterianos.

Info

Publication number
MX2007004179A
MX2007004179A MX2007004179A MX2007004179A MX2007004179A MX 2007004179 A MX2007004179 A MX 2007004179A MX 2007004179 A MX2007004179 A MX 2007004179A MX 2007004179 A MX2007004179 A MX 2007004179A MX 2007004179 A MX2007004179 A MX 2007004179A
Authority
MX
Mexico
Prior art keywords
antibacterial agents
triazolopyridine derivatives
triazolopyridine
derivatives
antimicrobials
Prior art date
Application number
MX2007004179A
Other languages
English (en)
Inventor
Chris Limberakis
Richard John Sciotti
Jeremy Tyson Starr
Huifen Chen
David Charles Donnell Butler
Vishnumurthy Ramachandra Hegde
Ravindra Madhukar Rasne
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of MX2007004179A publication Critical patent/MX2007004179A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Abstract

La presente invencion se refiere a una nueva clase de derivador de triazolopiridina, a su uso como antimicrobianos, y a agentes farmaceuticos que contienen estos compuestos.
MX2007004179A 2004-10-07 2005-09-23 Derivados de triazolpiridina como agentes antibacterianos. MX2007004179A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US61693104P 2004-10-07 2004-10-07
US71059205P 2005-08-24 2005-08-24
PCT/IB2005/003112 WO2006038116A2 (en) 2004-10-07 2005-09-23 Triazolopyridine derivatives as antibacterial agents

Publications (1)

Publication Number Publication Date
MX2007004179A true MX2007004179A (es) 2007-06-07

Family

ID=35998551

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007004179A MX2007004179A (es) 2004-10-07 2005-09-23 Derivados de triazolpiridina como agentes antibacterianos.

Country Status (7)

Country Link
US (1) US7524860B2 (es)
EP (1) EP1799680A2 (es)
JP (1) JP2008515874A (es)
BR (1) BRPI0516819A (es)
CA (1) CA2582482A1 (es)
MX (1) MX2007004179A (es)
WO (1) WO2006038116A2 (es)

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WO2008125111A1 (en) * 2007-04-16 2008-10-23 Leo Pharma A/S Triazolopyridines as phosphodiesterase inhibitors for treatment of dermal diseases
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US8119658B2 (en) 2007-10-01 2012-02-21 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
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CA2727036C (en) 2008-06-20 2017-03-21 Genentech, Inc. Triazolopyridine jak inhibitor compounds and methods
JPWO2009157423A1 (ja) 2008-06-24 2011-12-15 財団法人乙卯研究所 縮合環を有するオキサゾリジノン誘導体
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WO2010010187A1 (en) * 2008-07-25 2010-01-28 Galapagos Nv Novel compounds useful for the treatment of degenerative and inflammatory diseases
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WO2010010189A1 (en) * 2008-07-25 2010-01-28 Galapagos Nv Novel compounds useful for the treatment of degenerative and inflammatory diseases
WO2010010184A1 (en) * 2008-07-25 2010-01-28 Galapagos Nv [1, 2, 4] triazolo [1, 5-a] pyridines as jak inhibitors
TWI453207B (zh) 2008-09-08 2014-09-21 Signal Pharm Llc 胺基三唑并吡啶，其組合物及使用其之治療方法
WO2010057877A1 (en) * 2008-11-18 2010-05-27 Cellzome Limited 7-pyridinyl- or phenyl- substituted triazolo [1, 5 -a] pyridines as pi3k inhibitors
WO2010092015A1 (en) 2009-02-10 2010-08-19 Cellzome Limited Urea triazololo [1, 5-a] pyridine derivatives as pi3k inhibitors
CA2763900A1 (en) 2009-06-05 2010-12-09 Cephalon, Inc. Preparation and uses of 1,2,4-triazolo [1,5a] pyridine derivatives
JO3030B1 (ar) 2009-06-26 2016-09-05 Galapagos Nv مركب جديد مفيد لمعالجة الامراض التنكسية والالتهابات
TWI462920B (zh) 2009-06-26 2014-12-01 葛萊伯格有限公司 用於治療退化性及發炎疾病之新穎化合物
EP2343297A1 (en) 2009-11-30 2011-07-13 Bayer Schering Pharma AG Triazolopyridines
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BR112012024705A2 (pt) 2010-03-31 2016-06-07 Actelion Pharmaceuticals Ltd derivados antibacterianos de isoquinolin-3-ilureia
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CN106488915B (zh) 2014-02-13 2020-10-02 因赛特公司 作为lsd1抑制剂的环丙胺
US9527835B2 (en) 2014-02-13 2016-12-27 Incyte Corporation Cyclopropylamines as LSD1 inhibitors
EP3392244A1 (en) 2014-02-13 2018-10-24 Incyte Corporation Cyclopropylamines as lsd1 inhibitors
EP3626713B1 (en) 2014-02-13 2021-09-29 Incyte Corporation Cyclopropylamines for use as lsd1 inhibitors
US9695168B2 (en) 2014-07-10 2017-07-04 Incyte Corporation Substituted imidazo[1,5-α]pyridines and imidazo[1,5-α]pyrazines as LSD1 inhibitors
WO2016007727A1 (en) 2014-07-10 2016-01-14 Incyte Corporation Triazolopyridines and triazolopyrazines as lsd1 inhibitors
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US9695167B2 (en) 2014-07-10 2017-07-04 Incyte Corporation Substituted triazolo[1,5-a]pyridines and triazolo[1,5-a]pyrazines as LSD1 inhibitors
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EA035534B1 (ru) 2015-08-12 2020-06-30 Инсайт Корпорейшн Соли ингибитора lsd1
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WO2004014908A1 (en) 2002-08-13 2004-02-19 Warner-Lambert Company Llc Heterobicylcic metalloproteinase inhibitors

Also Published As

Publication number Publication date
CA2582482A1 (en) 2006-04-13
WO2006038116A2 (en) 2006-04-13
WO2006038116A3 (en) 2006-07-13
BRPI0516819A (pt) 2008-09-23
JP2008515874A (ja) 2008-05-15
US20080021059A1 (en) 2008-01-24
US7524860B2 (en) 2009-04-28
EP1799680A2 (en) 2007-06-27

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