CO6241154A2 - "compuestos novedosos con accion agonista o antagonista del receptor 1 vainilloide 1 (vr1/trpv1)\" - Google Patents

"compuestos novedosos con accion agonista o antagonista del receptor 1 vainilloide 1 (vr1/trpv1)\"

Info

Publication number
CO6241154A2
CO6241154A2 CO09118505A CO09118505A CO6241154A2 CO 6241154 A2 CO6241154 A2 CO 6241154A2 CO 09118505 A CO09118505 A CO 09118505A CO 09118505 A CO09118505 A CO 09118505A CO 6241154 A2 CO6241154 A2 CO 6241154A2
Authority
CO
Colombia
Prior art keywords
vainilloide
trpv1
agonist
receiver
new compounds
Prior art date
Application number
CO09118505A
Other languages
English (en)
Spanish (es)
Inventor
Robert Frank
Gregor Bahrenberg
Thomas Christoph
Klaus Schiene
Vry Jean N De
Derek Saunders
Bernard Sundermann
Jeewoo Lee
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102007018149A external-priority patent/DE102007018149A1/de
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of CO6241154A2 publication Critical patent/CO6241154A2/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
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  • Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
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CO09118505A 2007-04-16 2009-10-22 "compuestos novedosos con accion agonista o antagonista del receptor 1 vainilloide 1 (vr1/trpv1)\" CO6241154A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102007018149A DE102007018149A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
EP2008002997 2008-04-15
US12/103,667 US8084484B2 (en) 2007-04-16 2008-04-15 Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions

Publications (1)

Publication Number Publication Date
CO6241154A2 true CO6241154A2 (es) 2011-01-20

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Application Number Title Priority Date Filing Date
CO09118505A CO6241154A2 (es) 2007-04-16 2009-10-22 "compuestos novedosos con accion agonista o antagonista del receptor 1 vainilloide 1 (vr1/trpv1)\"

Country Status (14)

Country Link
JP (1) JP2010523727A (OSRAM)
KR (1) KR20100016593A (OSRAM)
CN (1) CN101679370A (OSRAM)
AU (1) AU2008238250B2 (OSRAM)
BR (1) BRPI0810035A2 (OSRAM)
CA (1) CA2683461A1 (OSRAM)
CO (1) CO6241154A2 (OSRAM)
EC (1) ECSP099692A (OSRAM)
IL (1) IL201505A0 (OSRAM)
MX (1) MX2009011149A (OSRAM)
NZ (1) NZ580411A (OSRAM)
RU (1) RU2498982C2 (OSRAM)
WO (1) WO2008125342A2 (OSRAM)
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RU2498982C2 (ru) 2013-11-20
WO2008125342A2 (de) 2008-10-23
BRPI0810035A2 (pt) 2016-07-26
KR20100016593A (ko) 2010-02-12
AU2008238250B2 (en) 2013-01-24
IL201505A0 (en) 2010-05-31
JP2010523727A (ja) 2010-07-15
AU2008238250A1 (en) 2008-10-23
ZA200907099B (en) 2013-03-27
WO2008125342A3 (de) 2009-01-15
CA2683461A1 (en) 2008-10-23
NZ580411A (en) 2012-06-29
CN101679370A (zh) 2010-03-24
MX2009011149A (es) 2009-10-30
ECSP099692A (es) 2009-11-30
RU2009142023A (ru) 2011-05-27

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