CO5700758A2 - Proceso para la preparacion de amino alcoholes sustituidos - Google Patents

Proceso para la preparacion de amino alcoholes sustituidos

Info

Publication number
CO5700758A2
CO5700758A2 CO06055464A CO06055464A CO5700758A2 CO 5700758 A2 CO5700758 A2 CO 5700758A2 CO 06055464 A CO06055464 A CO 06055464A CO 06055464 A CO06055464 A CO 06055464A CO 5700758 A2 CO5700758 A2 CO 5700758A2
Authority
CO
Colombia
Prior art keywords
preparation
amino substituted
atoms
substituted alcohols
alkyl
Prior art date
Application number
CO06055464A
Other languages
English (en)
Inventor
Yanzhong Wu
Arkadiy Rubezhov
Jean Schmid
Jay Thomas Afragola
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of CO5700758A2 publication Critical patent/CO5700758A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/04Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/02Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/04Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
    • C07C215/06Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
    • C07C215/08Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with only one hydroxy group and one amino group bound to the carbon skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

1.- Un proceso para la preparación de una aminoalcohol sustituido de la fórmula HO-(CH2)n-NR1R2 en donde R1 y R2 son cada uno independientemente H o alquilo C1-C3; o R1 y R2 cuando se toman opcionalmente junto con el átomo de nitrógeno el cual está cada uno unido forman un anillo heterocíclico saturado de 4 a 6 miembros que tiene 1-2 átomos de nitrógeno y 0-1 átomos de oxígeno o 0-1 átomos de azufre, y opcionalmente sustituido con R3; n es un entero de 2 a 7; R3 es alquilo C1-C3; que comprende la reacción de un alcohol de la fórmula HO-(CH2)n-X, donde X es Cl, Br o I, con una amina NHR1R2 en agua como solvente en un rango de temperatura de aproximadamente 20°C a aproximadamente 90°C.
CO06055464A 2003-12-08 2006-06-08 Proceso para la preparacion de amino alcoholes sustituidos CO5700758A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52793003P 2003-12-08 2003-12-08

Publications (1)

Publication Number Publication Date
CO5700758A2 true CO5700758A2 (es) 2006-11-30

Family

ID=34676795

Family Applications (1)

Application Number Title Priority Date Filing Date
CO06055464A CO5700758A2 (es) 2003-12-08 2006-06-08 Proceso para la preparacion de amino alcoholes sustituidos

Country Status (21)

Country Link
US (1) US7521552B2 (es)
EP (1) EP1692091A2 (es)
JP (1) JP2007513186A (es)
KR (1) KR20060127402A (es)
CN (1) CN1890244A (es)
AR (1) AR046873A1 (es)
AU (1) AU2004297245A1 (es)
BR (1) BRPI0417442A (es)
CA (1) CA2546907A1 (es)
CO (1) CO5700758A2 (es)
EC (1) ECSP066598A (es)
GT (1) GT200400256A (es)
HN (1) HN2004000518A (es)
IL (1) IL176019A0 (es)
NO (1) NO20062647L (es)
PA (1) PA8619501A1 (es)
PE (1) PE20050672A1 (es)
RU (1) RU2006117985A (es)
TW (1) TW200524843A (es)
WO (1) WO2005056514A2 (es)
ZA (1) ZA200604685B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010052181A2 (de) * 2008-11-05 2010-05-14 Basf Se Verfahren zur herstellung von n,n-substituierten-3-aminopropan-1-olen
CN101784016A (zh) * 2009-01-16 2010-07-21 鸿富锦精密工业(深圳)有限公司 在数码相框上实现发送邮件的方法及系统
CZ301920B6 (cs) * 2009-06-16 2010-07-28 Zentiva, K. S. Zpusob výroby (S)-4-methylamino-3-(3,4-dichlorfenyl)butan-1-olu
US8658829B2 (en) * 2010-02-08 2014-02-25 Ndsu Research Foundation Method of producing polyalkylated oligoalkylenepolyamines
KR101675440B1 (ko) * 2014-10-14 2016-11-15 한국화학연구원 광학 활성 3-클로로-1-아릴프로판-1-올 유도체로부터 3-아미노-1-아릴프로판-1-올 유도체의 제조방법

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1018868B (de) * 1954-11-06 1957-11-07 Rhone Poulenc Sa Verfahren zur Herstellung von Phenthiazinderivaten
GB783289A (en) 1954-11-12 1957-09-18 Rhone Poulenc Sa New phenthiazine derivatives and processes for their preparation
US4874785A (en) * 1985-10-01 1989-10-17 Ethyl Corporation Quaternary ammonium compounds
ES2244183T3 (es) * 1998-03-23 2005-12-01 Basf Aktiengesellschaft 6-(2-halo-4-alcoxifenil)-triazolpirimidinas fungicidas.
CA2419238A1 (en) * 2000-08-16 2002-02-21 University Of Alberta Non-pressurized methods for the preparation of conjugated solid supports for boronic acids

Also Published As

Publication number Publication date
HN2004000518A (es) 2007-03-26
GT200400256A (es) 2005-08-18
TW200524843A (en) 2005-08-01
PE20050672A1 (es) 2005-10-24
BRPI0417442A (pt) 2007-03-13
RU2006117985A (ru) 2008-01-20
AU2004297245A1 (en) 2005-06-23
US20050124806A1 (en) 2005-06-09
NO20062647L (no) 2006-09-06
IL176019A0 (en) 2006-10-05
JP2007513186A (ja) 2007-05-24
AR046873A1 (es) 2005-12-28
ZA200604685B (en) 2009-03-25
PA8619501A1 (es) 2005-08-10
US7521552B2 (en) 2009-04-21
EP1692091A2 (en) 2006-08-23
WO2005056514A2 (en) 2005-06-23
WO2005056514A3 (en) 2005-08-11
CA2546907A1 (en) 2005-06-23
CN1890244A (zh) 2007-01-03
ECSP066598A (es) 2006-10-25
KR20060127402A (ko) 2006-12-12

Similar Documents

Publication Publication Date Title
CO5700758A2 (es) Proceso para la preparacion de amino alcoholes sustituidos
CO5631432A2 (es) Derivados de n-[fenil(piepidin-2-il)metil]benzamida, su preparacion y su aplicacion en terapeutica
AR049401A1 (es) Aza-biciclononanos
PE20030762A1 (es) Compuestos heterociclicos como antagonistas nk1
PE20030890A1 (es) Cumarinas utiles como biomarcadores
DK1385926T3 (da) Smöreoliesammensætning der omfatter en tilsætningsstofkombination af en carboxylsyre og en amin som antirustmiddel
CO6140053A2 (es) Proceso para fabricar 2-amino-5-halobenzamidas 3-sustituidas
AR068538A1 (es) Compuesto heterociclico de 5 miembros con actividad supresora de la secrecion de acido
ES2271615T3 (es) N-aril-2-oxazolidinona-5-carboxamidas y sus derivados y su uso como antibacterianos.
AR045868A1 (es) Proceso para preparar compuestos de ocarbamoilo en presencia de grupo amina activa
EA200300777A1 (ru) N-фенпропилциклопентил-замещенные производные глутарамида в качестве nep ингибиторов для fsad
BRPI0510335A (pt) composto heterocìclico
AR052915A1 (es) Derivados de pirrolidin y piperidin acetileno
AR059517A1 (es) N- sulfonilacion selectiva de alcoholes sustituidos con 2- aminotrifluoralquilo
CO5690598A2 (es) 6-[(sustituido)fenil]triazolopirimidinas como agentes anticancer
AR123584A2 (es) Procesos y compuestos intermediarios para la preparación de derivados de 2-carboxamida-cicloamino-urea
CO5631434A2 (es) Derivados de piridina-carboxamida y su uso como plaguicidas
GB1046506A (en) Guanidine compounds and process for their manufacture
AR054121A1 (es) Compuestos de fenilpiridilpiperazina, procedimiento de preparacion, composiciones farmaceuticas que los contienen, y usos farmacologicos como antagonistas de receptores histaminergicos h3
ECSP066606A (es) Proceso para la preparación de inhibidores de tubulina
PE20011137A1 (es) Inhibidores de las metaloproteasas que contienen cadenas laterales heterociclicas n-sustituidas
AR053722A2 (es) Procedimiento para preparar secretagogos de hormonas del crecimiento y poliformo de los compuestos obtenidos
AR046041A1 (es) Procedimiento para la preparacion de compuestos heterociclicos n-amino sustituidos
AR058171A1 (es) Procesos para la preparacion de derivados de ciclopropilamida
PE20230110A1 (es) Procesos para la preparacion de un inhibidor de cinasa

Legal Events

Date Code Title Description
FC Application refused