ECSP066598A - Proceso para la preparación de amino alcoholes sustituidos - Google Patents
Proceso para la preparación de amino alcoholes sustituidosInfo
- Publication number
- ECSP066598A ECSP066598A EC2006006598A ECSP066598A ECSP066598A EC SP066598 A ECSP066598 A EC SP066598A EC 2006006598 A EC2006006598 A EC 2006006598A EC SP066598 A ECSP066598 A EC SP066598A EC SP066598 A ECSP066598 A EC SP066598A
- Authority
- EC
- Ecuador
- Prior art keywords
- preparation
- amino substituted
- substituted alcohols
- haloalcohols
- useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
- C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
- C07C215/08—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with only one hydroxy group and one amino group bound to the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Se suministra un proceso para la preparación de amino alcoholes sustituidos HO-(CH2)n-NR1R2 de haloalcoholes HO-(CH2)n-X, donde X es Cl, Br, o I, mediante la reacción con una amina HNR1R2, en agua como solvente a temperatura en el rango de aproximadamente 20°C a aproximadamente 90°C opcionalmente en la presencia de una cantidad catalítica de unos yoduros metálicos fuente de yoduro. Los haloalcoholes son útiles en la preparación de compuestos 6-[fenilo(sustituido)]-triazolopirimidina que son útiles en el tratamiento de cáncer.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52793003P | 2003-12-08 | 2003-12-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP066598A true ECSP066598A (es) | 2006-10-25 |
Family
ID=34676795
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2006006598A ECSP066598A (es) | 2003-12-08 | 2006-06-02 | Proceso para la preparación de amino alcoholes sustituidos |
Country Status (21)
Country | Link |
---|---|
US (1) | US7521552B2 (es) |
EP (1) | EP1692091A2 (es) |
JP (1) | JP2007513186A (es) |
KR (1) | KR20060127402A (es) |
CN (1) | CN1890244A (es) |
AR (1) | AR046873A1 (es) |
AU (1) | AU2004297245A1 (es) |
BR (1) | BRPI0417442A (es) |
CA (1) | CA2546907A1 (es) |
CO (1) | CO5700758A2 (es) |
EC (1) | ECSP066598A (es) |
GT (1) | GT200400256A (es) |
HN (1) | HN2004000518A (es) |
IL (1) | IL176019A0 (es) |
NO (1) | NO20062647L (es) |
PA (1) | PA8619501A1 (es) |
PE (1) | PE20050672A1 (es) |
RU (1) | RU2006117985A (es) |
TW (1) | TW200524843A (es) |
WO (1) | WO2005056514A2 (es) |
ZA (1) | ZA200604685B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102203054B (zh) * | 2008-11-05 | 2014-07-30 | 巴斯夫欧洲公司 | 生产n,n-取代的3-氨基丙-1-醇的方法 |
CN101784016A (zh) * | 2009-01-16 | 2010-07-21 | 鸿富锦精密工业(深圳)有限公司 | 在数码相框上实现发送邮件的方法及系统 |
CZ2009385A3 (cs) * | 2009-06-16 | 2010-07-28 | Zentiva, K. S. | Zpusob výroby (S)-4-methylamino-3-(3,4-dichlorfenyl)butan-1-olu |
WO2011097490A1 (en) * | 2010-02-08 | 2011-08-11 | Ndsu Research Foundation | Method of producing polyalkylated oligoalkylenepolyamines |
KR101675440B1 (ko) * | 2014-10-14 | 2016-11-15 | 한국화학연구원 | 광학 활성 3-클로로-1-아릴프로판-1-올 유도체로부터 3-아미노-1-아릴프로판-1-올 유도체의 제조방법 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1018868B (de) * | 1954-11-06 | 1957-11-07 | Rhone Poulenc Sa | Verfahren zur Herstellung von Phenthiazinderivaten |
GB783289A (en) | 1954-11-12 | 1957-09-18 | Rhone Poulenc Sa | New phenthiazine derivatives and processes for their preparation |
US4874785A (en) * | 1985-10-01 | 1989-10-17 | Ethyl Corporation | Quaternary ammonium compounds |
CA2324154C (en) * | 1998-03-23 | 2008-03-18 | American Cyanamid Company | Fungicidal 6-(2-halo-4-alkoxyphenyl)-triazolopyrimidines |
CA2419238A1 (en) * | 2000-08-16 | 2002-02-21 | University Of Alberta | Non-pressurized methods for the preparation of conjugated solid supports for boronic acids |
-
2004
- 2004-12-03 TW TW093137288A patent/TW200524843A/zh unknown
- 2004-12-06 HN HN2004000518A patent/HN2004000518A/es unknown
- 2004-12-06 GT GT200400256A patent/GT200400256A/es unknown
- 2004-12-07 WO PCT/US2004/040855 patent/WO2005056514A2/en active Application Filing
- 2004-12-07 RU RU2006117985/04A patent/RU2006117985A/ru not_active Application Discontinuation
- 2004-12-07 AR ARP040104568A patent/AR046873A1/es not_active Application Discontinuation
- 2004-12-07 KR KR1020067011097A patent/KR20060127402A/ko not_active Application Discontinuation
- 2004-12-07 BR BRPI0417442-9A patent/BRPI0417442A/pt not_active IP Right Cessation
- 2004-12-07 CA CA002546907A patent/CA2546907A1/en not_active Abandoned
- 2004-12-07 PA PA20048619501A patent/PA8619501A1/es unknown
- 2004-12-07 EP EP04813204A patent/EP1692091A2/en not_active Withdrawn
- 2004-12-07 PE PE2004001202A patent/PE20050672A1/es not_active Application Discontinuation
- 2004-12-07 AU AU2004297245A patent/AU2004297245A1/en not_active Withdrawn
- 2004-12-07 JP JP2006542868A patent/JP2007513186A/ja not_active Withdrawn
- 2004-12-07 CN CNA2004800362789A patent/CN1890244A/zh active Pending
- 2004-12-08 US US11/006,936 patent/US7521552B2/en not_active Expired - Fee Related
-
2006
- 2006-05-30 IL IL176019A patent/IL176019A0/en unknown
- 2006-06-02 EC EC2006006598A patent/ECSP066598A/es unknown
- 2006-06-07 ZA ZA200604685A patent/ZA200604685B/xx unknown
- 2006-06-08 CO CO06055464A patent/CO5700758A2/es not_active Application Discontinuation
- 2006-06-08 NO NO20062647A patent/NO20062647L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
KR20060127402A (ko) | 2006-12-12 |
NO20062647L (no) | 2006-09-06 |
GT200400256A (es) | 2005-08-18 |
PE20050672A1 (es) | 2005-10-24 |
RU2006117985A (ru) | 2008-01-20 |
CO5700758A2 (es) | 2006-11-30 |
IL176019A0 (en) | 2006-10-05 |
JP2007513186A (ja) | 2007-05-24 |
CA2546907A1 (en) | 2005-06-23 |
EP1692091A2 (en) | 2006-08-23 |
AU2004297245A1 (en) | 2005-06-23 |
US7521552B2 (en) | 2009-04-21 |
HN2004000518A (es) | 2007-03-26 |
AR046873A1 (es) | 2005-12-28 |
CN1890244A (zh) | 2007-01-03 |
WO2005056514A3 (en) | 2005-08-11 |
BRPI0417442A (pt) | 2007-03-13 |
US20050124806A1 (en) | 2005-06-09 |
WO2005056514A2 (en) | 2005-06-23 |
PA8619501A1 (es) | 2005-08-10 |
ZA200604685B (en) | 2009-03-25 |
TW200524843A (en) | 2005-08-01 |
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