PA8619501A1 - Proceso para la preparacion de aminoalcoholes sustituidos - Google Patents

Proceso para la preparacion de aminoalcoholes sustituidos

Info

Publication number
PA8619501A1
PA8619501A1 PA20048619501A PA8619501A PA8619501A1 PA 8619501 A1 PA8619501 A1 PA 8619501A1 PA 20048619501 A PA20048619501 A PA 20048619501A PA 8619501 A PA8619501 A PA 8619501A PA 8619501 A1 PA8619501 A1 PA 8619501A1
Authority
PA
Panama
Prior art keywords
preparation
aminoalcoholes
substituted
haloalcoholes
useful
Prior art date
Application number
PA20048619501A
Other languages
English (en)
Inventor
Yanzhong Wu
Arkadiy Rubezhov
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of PA8619501A1 publication Critical patent/PA8619501A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
    • C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
    • C07C215/08—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with only one hydroxy group and one amino group bound to the carbon skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

SE PROVEE UN PROCESO PARA LA PREPARACION DE AMINOALCOHOLES SUSTITUIDOS HO-(CH2)N-NR1R2 A PARTIR DE HALOALCOHOLES HO-(CH2)N-X, DONDE X ES CL, Br O I, MEDIANTE REACCION CON UNA AMINA HNR1R2, EN AGUA COMO SOLVENTE A UN RANGO DE TEMPERATURA DE APROXIMADAMENTE 90°C OPCIONALMENTE EN PRESENCIA DE UNA CANTIDAD CATALITICA DE YODUROS METALICOS COMO FUENTE DE YODURO. LOS HALOALCOHOLES SON UTILES EN LA PREPARACION DE COMPUESTOS DE 6-[FENIL(SUSTITUIDO)]-TRIAZOLOPIRIMIDINA LOS CUALES SON UTILES EN EL TRATAMIENTO DEL CANCER.
PA20048619501A 2003-12-08 2004-12-07 Proceso para la preparacion de aminoalcoholes sustituidos PA8619501A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52793003P 2003-12-08 2003-12-08

Publications (1)

Publication Number Publication Date
PA8619501A1 true PA8619501A1 (es) 2005-08-10

Family

ID=34676795

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20048619501A PA8619501A1 (es) 2003-12-08 2004-12-07 Proceso para la preparacion de aminoalcoholes sustituidos

Country Status (21)

Country Link
US (1) US7521552B2 (es)
EP (1) EP1692091A2 (es)
JP (1) JP2007513186A (es)
KR (1) KR20060127402A (es)
CN (1) CN1890244A (es)
AR (1) AR046873A1 (es)
AU (1) AU2004297245A1 (es)
BR (1) BRPI0417442A (es)
CA (1) CA2546907A1 (es)
CO (1) CO5700758A2 (es)
EC (1) ECSP066598A (es)
GT (1) GT200400256A (es)
HN (1) HN2004000518A (es)
IL (1) IL176019A0 (es)
NO (1) NO20062647L (es)
PA (1) PA8619501A1 (es)
PE (1) PE20050672A1 (es)
RU (1) RU2006117985A (es)
TW (1) TW200524843A (es)
WO (1) WO2005056514A2 (es)
ZA (1) ZA200604685B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8536377B2 (en) * 2008-11-05 2013-09-17 Basf Se Method for producing N,N-substituted-3-aminopropan-1-ols
CN101784016A (zh) * 2009-01-16 2010-07-21 鸿富锦精密工业（深圳）有限公司 在数码相框上实现发送邮件的方法及系统
CZ2009385A3 (cs) * 2009-06-16 2010-07-28 Zentiva, K. S. Zpusob výroby (S)-4-methylamino-3-(3,4-dichlorfenyl)butan-1-olu
JP2013518901A (ja) * 2010-02-08 2013-05-23 エヌディーエスユー リサーチ ファウンデーション ポリアルキル化オリゴアルキレンポリアミンを生成する方法
KR101675440B1 (ko) * 2014-10-14 2016-11-15 한국화학연구원 광학 활성 3-클로로-1-아릴프로판-1-올 유도체로부터 3-아미노-1-아릴프로판-1-올 유도체의 제조방법

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1018868B (de) * 1954-11-06 1957-11-07 Rhone Poulenc Sa Verfahren zur Herstellung von Phenthiazinderivaten
GB783289A (en) 1954-11-12 1957-09-18 Rhone Poulenc Sa New phenthiazine derivatives and processes for their preparation
US4874785A (en) * 1985-10-01 1989-10-17 Ethyl Corporation Quaternary ammonium compounds
WO1999048893A1 (en) * 1998-03-23 1999-09-30 American Cyanamid Company Fungicidal 6-(2-halo-4-alkoxyphenyl)-triazolopyrimidines
CA2419238A1 (en) * 2000-08-16 2002-02-21 University Of Alberta Non-pressurized methods for the preparation of conjugated solid supports for boronic acids

Also Published As

Publication number Publication date
JP2007513186A (ja) 2007-05-24
BRPI0417442A (pt) 2007-03-13
KR20060127402A (ko) 2006-12-12
AU2004297245A1 (en) 2005-06-23
ZA200604685B (en) 2009-03-25
CA2546907A1 (en) 2005-06-23
HN2004000518A (es) 2007-03-26
NO20062647L (no) 2006-09-06
US7521552B2 (en) 2009-04-21
WO2005056514A3 (en) 2005-08-11
ECSP066598A (es) 2006-10-25
EP1692091A2 (en) 2006-08-23
CO5700758A2 (es) 2006-11-30
IL176019A0 (en) 2006-10-05
CN1890244A (zh) 2007-01-03
PE20050672A1 (es) 2005-10-24
RU2006117985A (ru) 2008-01-20
TW200524843A (en) 2005-08-01
US20050124806A1 (en) 2005-06-09
AR046873A1 (es) 2005-12-28
GT200400256A (es) 2005-08-18
WO2005056514A2 (en) 2005-06-23

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