AR046873A1 - Proceso para la preparacion de aminoalcoholes sustituidos - Google Patents
Proceso para la preparacion de aminoalcoholes sustituidosInfo
- Publication number
- AR046873A1 AR046873A1 ARP040104568A ARP040104568A AR046873A1 AR 046873 A1 AR046873 A1 AR 046873A1 AR P040104568 A ARP040104568 A AR P040104568A AR P040104568 A ARP040104568 A AR P040104568A AR 046873 A1 AR046873 A1 AR 046873A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- substituted
- atoms
- aminoalcoholes
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
- C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
- C07C215/08—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with only one hydroxy group and one amino group bound to the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Los haloalcoholes son útiles en la preparación de compuestos de 6-[fenil](sustituido)]-triazolopirimidina los cuales son útiles en el tratamiento del cáncer. Reivindicación 1: Un proceso para la preparación de un aminoalcohol sustituido de la fórmula HO-(CH2)n-NR1R2 en donde R1 y R2 son cada uno independientemente H o alquilo C1-3, o R1 y R2 cuando opcionalmente son tomados en forma conjunta con el átomo de N al cual cada uno está unido forman un anillo heterocíclico saturado de 4 a 6 miembros que tiene 1-2 átomos de N y 0-1 átomos de O o 0-1 átomos de S, y opcionalmente con R3; n es un número entero de 2 a 7; R3 es alquilo C1-3; el cual comprende la reacción de un haloalcohol de la fórmula HO-(CH2)n-X en donde X es Cl, Br, o I, con una amina NHR1R2, en agua como solvente a un rango de temperatura entre aproximadamente 20sC y aproximadamente 90sC.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US52793003P | 2003-12-08 | 2003-12-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR046873A1 true AR046873A1 (es) | 2005-12-28 |
Family
ID=34676795
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP040104568A AR046873A1 (es) | 2003-12-08 | 2004-12-07 | Proceso para la preparacion de aminoalcoholes sustituidos |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US7521552B2 (es) |
| EP (1) | EP1692091A2 (es) |
| JP (1) | JP2007513186A (es) |
| KR (1) | KR20060127402A (es) |
| CN (1) | CN1890244A (es) |
| AR (1) | AR046873A1 (es) |
| AU (1) | AU2004297245A1 (es) |
| BR (1) | BRPI0417442A (es) |
| CA (1) | CA2546907A1 (es) |
| CO (1) | CO5700758A2 (es) |
| EC (1) | ECSP066598A (es) |
| GT (1) | GT200400256A (es) |
| HN (1) | HN2004000518A (es) |
| IL (1) | IL176019A0 (es) |
| NO (1) | NO20062647L (es) |
| PA (1) | PA8619501A1 (es) |
| PE (1) | PE20050672A1 (es) |
| RU (1) | RU2006117985A (es) |
| TW (1) | TW200524843A (es) |
| WO (1) | WO2005056514A2 (es) |
| ZA (1) | ZA200604685B (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2590457T3 (es) * | 2008-11-05 | 2016-11-22 | Basf Se | Procedimiento para la producción de 3-aminopropano-1-oles N,N-sustituidos |
| CN101784016A (zh) * | 2009-01-16 | 2010-07-21 | 鸿富锦精密工业（深圳）有限公司 | 在数码相框上实现发送邮件的方法及系统 |
| CZ2009385A3 (cs) * | 2009-06-16 | 2010-07-28 | Zentiva, K. S. | Zpusob výroby (S)-4-methylamino-3-(3,4-dichlorfenyl)butan-1-olu |
| WO2011097490A1 (en) * | 2010-02-08 | 2011-08-11 | Ndsu Research Foundation | Method of producing polyalkylated oligoalkylenepolyamines |
| KR101675440B1 (ko) * | 2014-10-14 | 2016-11-15 | 한국화학연구원 | 광학 활성 3-클로로-1-아릴프로판-1-올 유도체로부터 3-아미노-1-아릴프로판-1-올 유도체의 제조방법 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1018868B (de) * | 1954-11-06 | 1957-11-07 | Rhone Poulenc Sa | Verfahren zur Herstellung von Phenthiazinderivaten |
| GB783289A (en) | 1954-11-12 | 1957-09-18 | Rhone Poulenc Sa | New phenthiazine derivatives and processes for their preparation |
| US4874785A (en) * | 1985-10-01 | 1989-10-17 | Ethyl Corporation | Quaternary ammonium compounds |
| CN100339378C (zh) * | 1998-03-23 | 2007-09-26 | 巴斯福股份公司 | 杀真菌的6－(2－卤代－4－烷氧基苯基)－三唑并嘧啶 |
| AU2001287399A1 (en) * | 2000-08-16 | 2002-02-25 | University Of Alberta | Non-pressurized methods for the preparation of conjugated solid supports for boronic acids |
-
2004
- 2004-12-03 TW TW093137288A patent/TW200524843A/zh unknown
- 2004-12-06 HN HN2004000518A patent/HN2004000518A/es unknown
- 2004-12-06 GT GT200400256A patent/GT200400256A/es unknown
- 2004-12-07 PE PE2004001202A patent/PE20050672A1/es not_active Application Discontinuation
- 2004-12-07 PA PA20048619501A patent/PA8619501A1/es unknown
- 2004-12-07 JP JP2006542868A patent/JP2007513186A/ja not_active Withdrawn
- 2004-12-07 WO PCT/US2004/040855 patent/WO2005056514A2/en active Application Filing
- 2004-12-07 CN CNA2004800362789A patent/CN1890244A/zh active Pending
- 2004-12-07 AU AU2004297245A patent/AU2004297245A1/en not_active Withdrawn
- 2004-12-07 BR BRPI0417442-9A patent/BRPI0417442A/pt not_active IP Right Cessation
- 2004-12-07 EP EP04813204A patent/EP1692091A2/en not_active Withdrawn
- 2004-12-07 KR KR1020067011097A patent/KR20060127402A/ko not_active Application Discontinuation
- 2004-12-07 CA CA002546907A patent/CA2546907A1/en not_active Abandoned
- 2004-12-07 AR ARP040104568A patent/AR046873A1/es not_active Application Discontinuation
- 2004-12-07 RU RU2006117985/04A patent/RU2006117985A/ru not_active Application Discontinuation
- 2004-12-08 US US11/006,936 patent/US7521552B2/en not_active Expired - Fee Related
-
2006
- 2006-05-30 IL IL176019A patent/IL176019A0/en unknown
- 2006-06-02 EC EC2006006598A patent/ECSP066598A/es unknown
- 2006-06-07 ZA ZA200604685A patent/ZA200604685B/xx unknown
- 2006-06-08 NO NO20062647A patent/NO20062647L/no not_active Application Discontinuation
- 2006-06-08 CO CO06055464A patent/CO5700758A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2006117985A (ru) | 2008-01-20 |
| CA2546907A1 (en) | 2005-06-23 |
| PA8619501A1 (es) | 2005-08-10 |
| CO5700758A2 (es) | 2006-11-30 |
| ECSP066598A (es) | 2006-10-25 |
| PE20050672A1 (es) | 2005-10-24 |
| CN1890244A (zh) | 2007-01-03 |
| BRPI0417442A (pt) | 2007-03-13 |
| HN2004000518A (es) | 2007-03-26 |
| US20050124806A1 (en) | 2005-06-09 |
| TW200524843A (en) | 2005-08-01 |
| JP2007513186A (ja) | 2007-05-24 |
| ZA200604685B (en) | 2009-03-25 |
| IL176019A0 (en) | 2006-10-05 |
| KR20060127402A (ko) | 2006-12-12 |
| US7521552B2 (en) | 2009-04-21 |
| NO20062647L (no) | 2006-09-06 |
| WO2005056514A3 (en) | 2005-08-11 |
| AU2004297245A1 (en) | 2005-06-23 |
| WO2005056514A2 (en) | 2005-06-23 |
| EP1692091A2 (en) | 2006-08-23 |
| GT200400256A (es) | 2005-08-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |