CO2021005140A2 - Formas mórficas de los inhibidores del factor d del complemento - Google Patents

Formas mórficas de los inhibidores del factor d del complemento

Info

Publication number
CO2021005140A2
CO2021005140A2 CONC2021/0005140A CO2021005140A CO2021005140A2 CO 2021005140 A2 CO2021005140 A2 CO 2021005140A2 CO 2021005140 A CO2021005140 A CO 2021005140A CO 2021005140 A2 CO2021005140 A2 CO 2021005140A2
Authority
CO
Colombia
Prior art keywords
complement factor
inhibitors
morphic forms
forms
morphic
Prior art date
Application number
CONC2021/0005140A
Other languages
English (en)
Spanish (es)
Inventor
Avinash Phadke
Akihiro Hashimoto
Mark Andres
Original Assignee
Achillion Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Achillion Pharmaceuticals Inc filed Critical Achillion Pharmaceuticals Inc
Publication of CO2021005140A2 publication Critical patent/CO2021005140A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
CONC2021/0005140A 2018-09-25 2021-04-22 Formas mórficas de los inhibidores del factor d del complemento CO2021005140A2 (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862736294P 2018-09-25 2018-09-25
US201862757565P 2018-11-08 2018-11-08
US201862760520P 2018-11-13 2018-11-13
US201962796776P 2019-01-25 2019-01-25
PCT/US2019/053012 WO2020069024A1 (en) 2018-09-25 2019-09-25 Morphic forms of complement factor d inhibitors

Publications (1)

Publication Number Publication Date
CO2021005140A2 true CO2021005140A2 (es) 2021-04-30

Family

ID=69949508

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2021/0005140A CO2021005140A2 (es) 2018-09-25 2021-04-22 Formas mórficas de los inhibidores del factor d del complemento

Country Status (11)

Country Link
US (1) US11807627B2 (enExample)
EP (1) EP3856164B1 (enExample)
JP (1) JP2022502500A (enExample)
KR (1) KR20210093855A (enExample)
CN (1) CN112996497A (enExample)
AU (1) AU2019346464A1 (enExample)
BR (1) BR112021005506A2 (enExample)
CA (1) CA3114039A1 (enExample)
CO (1) CO2021005140A2 (enExample)
MX (1) MX2021003425A (enExample)
WO (1) WO2020069024A1 (enExample)

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