CN1747929B - 趋化因子i-tac或sdf-1结合于ccxckr2受体的抑制剂 - Google Patents

趋化因子i-tac或sdf-1结合于ccxckr2受体的抑制剂 Download PDF

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CN1747929B
CN1747929B CN2003801097644A CN200380109764A CN1747929B CN 1747929 B CN1747929 B CN 1747929B CN 2003801097644 A CN2003801097644 A CN 2003801097644A CN 200380109764 A CN200380109764 A CN 200380109764A CN 1747929 B CN1747929 B CN 1747929B
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methyl
phenyl
substituted
allyl
unsubstituted
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CN1747929A (zh
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A·梅利基安
J·博恩斯
B·E·麦克马斯特
T·沙尔
J·J·赖特
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Chemocentryx Inc
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    • A61P35/00—Antineoplastic agents
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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CN2003801097644A 2002-12-20 2003-12-22 趋化因子i-tac或sdf-1结合于ccxckr2受体的抑制剂 Expired - Lifetime CN1747929B (zh)

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Application Number Priority Date Filing Date Title
US43491202P 2002-12-20 2002-12-20
US60/434,912 2002-12-20
US51615103P 2003-10-30 2003-10-30
US60/516,151 2003-10-30
PCT/US2003/041024 WO2004058705A2 (en) 2002-12-20 2003-12-22 Inhibitors of the binding of chemokines i-tac or sdf-1 to the ccxckr2 receptor

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CN1747929A CN1747929A (zh) 2006-03-15
CN1747929B true CN1747929B (zh) 2010-04-28

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AT (1) ATE427933T1 (https=)
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US7253007B2 (en) 2001-11-30 2007-08-07 Chemocentryx, Inc. Compositions and methods for detecting and treating diseases and conditions related to chemokine receptors
ATE427933T1 (de) * 2002-12-20 2009-04-15 Chemocentryx Inc Inhibitoren der bindungder chemokine i-tac bzw. sdf-1 an den ccxckr2-rezeptor
SI1638933T1 (sl) 2003-06-17 2008-10-31 Pfizer Derivati N-pirolidin-3-il-amida kot inhibitorji ponovnega privzema serotonina in noradrenalina
EP1715892A4 (en) * 2004-02-03 2008-07-09 Chemocentryx Inc METHODS AND COMPOSITIONS FOR MODULATING ANGIOGENESIS
WO2006038989A1 (en) * 2004-09-29 2006-04-13 Chemocentryx, Inc. Substituted arylamides
WO2006116319A2 (en) * 2005-04-21 2006-11-02 Chemocentryx, Inc. Reagents that bind ccx-ckr2
EP1909575A2 (en) * 2005-06-29 2008-04-16 ChemoCentryx Inc Substituted n-cinnamyl benzamides
DE602006018057D1 (de) * 2005-11-10 2010-12-16 Chemocentryx Inc Substituierte chinolone und verwendungsverfahren
EA028604B1 (ru) * 2013-05-30 2017-12-29 Идорсиа Фармасьютиклз Лтд. Модуляторы рецептора cxcr7
ES2732437T3 (es) * 2014-12-01 2019-11-22 Idorsia Pharmaceuticals Ltd Moduladores del receptor de CXCR7

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ATE427933T1 (de) 2009-04-15
US20100144720A1 (en) 2010-06-10
WO2004058705B1 (en) 2004-09-30
MXPA05006507A (es) 2006-02-17
AU2003300293A1 (en) 2004-07-22
WO2004058705A2 (en) 2004-07-15
KR20050109920A (ko) 2005-11-22
AU2003300293B8 (en) 2010-01-14
US7649011B2 (en) 2010-01-19
US20040171655A1 (en) 2004-09-02
CA2511242A1 (en) 2004-07-15
EP1606251A2 (en) 2005-12-21
JP2006515854A (ja) 2006-06-08
CN1747929A (zh) 2006-03-15
KR101061352B1 (ko) 2011-08-31
EP1606251B1 (en) 2009-04-08
JP4870357B2 (ja) 2012-02-08
ES2323528T3 (es) 2009-07-20
CA2511242C (en) 2010-01-12
AU2003300293B2 (en) 2009-12-17
WO2004058705A3 (en) 2004-08-19
DE60327106D1 (de) 2009-05-20

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