CN109476641B - Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 - Google Patents

Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 Download PDF

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CN109476641B
CN109476641B CN201780045651.4A CN201780045651A CN109476641B CN 109476641 B CN109476641 B CN 109476641B CN 201780045651 A CN201780045651 A CN 201780045651A CN 109476641 B CN109476641 B CN 109476641B
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cancer
mmol
compound
methyl
formula
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CN109476641A (zh
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P·西尔
S·布朗纳
F·A·罗梅罗
S·马格努森
V·H-W·徐
J·瓦伊
K·W·赖
F·王
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Genentech Inc
Constellation Pharmaceuticals Inc
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Constellation Pharmaceuticals Inc
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CN201780045651.4A 2016-05-24 2017-05-24 Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 Active CN109476641B (zh)

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WO2017205536A2 (en) 2016-05-24 2017-11-30 Genentech, Inc. Therapeutic compounds and uses thereof
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CN110573501B (zh) * 2017-06-30 2023-09-29 北京泰德制药股份有限公司 Rho相关蛋白激酶抑制剂、包含其的药物组合物及其制备方法和用途
WO2019000683A1 (zh) 2017-06-30 2019-01-03 北京泰德制药股份有限公司 Rho相关蛋白激酶抑制剂、包含其的药物组合物及其制备方法和用途
TWI846350B (zh) 2017-09-15 2024-06-21 美商佛瑪治療公司 作為ＣＢＰ／ｐ３００抑制劑之四氫－咪唑並喹啉化合物
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