HK1243072A1 - 布羅莫結構域抑制劑及其用途 - Google Patents

布羅莫結構域抑制劑及其用途

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Publication number
HK1243072A1
HK1243072A1 HK18102568.8A HK18102568A HK1243072A1 HK 1243072 A1 HK1243072 A1 HK 1243072A1 HK 18102568 A HK18102568 A HK 18102568A HK 1243072 A1 HK1243072 A1 HK 1243072A1
Authority
HK
Hong Kong
Prior art keywords
bromodomain inhibitors
bromodomain
inhibitors
Prior art date
Application number
HK18102568.8A
Other languages
English (en)
Inventor
Brian K Albrecht
Steven F Bellon
Daniel J Burdick
Alexandre Cote
Terry Crawford
Les A Dakin
Tsui Vickie Hsiao-Wei
Michael Charles Hewitt
Yves Leblanc
Steven R Magnuson
Christopher G Nasveschuk
F Anthony Romero
Yong Tang
Alexander M Taylor
Shumei Wang
Original Assignee
基因泰克公司
星座製藥股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 基因泰克公司, 星座製藥股份有限公司 filed Critical 基因泰克公司
Publication of HK1243072A1 publication Critical patent/HK1243072A1/zh

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
HK18102568.8A 2014-11-10 2018-02-22 布羅莫結構域抑制劑及其用途 HK1243072A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462077711P 2014-11-10 2014-11-10
PCT/US2015/059997 WO2016077375A1 (en) 2014-11-10 2015-11-10 Bromodomain inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
HK1243072A1 true HK1243072A1 (zh) 2018-07-06

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
HK18102568.8A HK1243072A1 (zh) 2014-11-10 2018-02-22 布羅莫結構域抑制劑及其用途

Country Status (6)

Country Link
US (1) US10258603B2 (zh)
EP (1) EP3218376B1 (zh)
JP (1) JP6639497B2 (zh)
CN (1) CN107108613B (zh)
HK (1) HK1243072A1 (zh)
WO (1) WO2016077375A1 (zh)

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US10258603B2 (en) 2019-04-16
CN107108613A (zh) 2017-08-29
JP2017533250A (ja) 2017-11-09
JP6639497B2 (ja) 2020-02-05
WO2016077375A1 (en) 2016-05-19
EP3218376A1 (en) 2017-09-20
US20170340604A1 (en) 2017-11-30
EP3218376B1 (en) 2019-12-25
CN107108613B (zh) 2020-02-25

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