CN108355111A - 一种治疗子宫颈癌的药物及其制备方法 - Google Patents
一种治疗子宫颈癌的药物及其制备方法 Download PDFInfo
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Abstract
本发明公开了一种治疗子宫颈癌的药物及其制备方法,其是由土茯苓、贯众、苦参、地榆、牛膝、栀子、黄柏、薏苡仁、黄芪、女贞子、枸杞子、枳壳、莪术、白花蛇舌草、白茅根、当归、昆布、海藻、蚤休、山慈姑、香附、柴胡、全蝎、续断、半枝莲、白芍、茯苓、升麻、生地黄、玄参、沉香、延胡索按一定重量配比制备而成,本发明药物具有凉血止血,清热解毒,行气破血,消积止痛,理气解郁,止痛调经的功能,用于治疗子宫颈癌见效快、疗效好,不复发。
Description
技术领域
本发明涉及一种治疗子宫颈癌的药物及其制备方法,属中药领域。
背景技术
子宫颈癌是最常见的妇科恶性肿瘤。原位癌高发年龄为30~35岁,浸润癌为45~55岁,近年来其发病有年轻化的趋势。近几十年宫颈细胞学筛查的普遍应用,使子宫颈癌和癌前病变得以早期发现和治疗,子宫颈癌的发病率和死亡率已有明显下降。由于西药治疗副作用大,因此人们对有效治疗子宫颈癌的中药药物存在极大的需求,至今为止,还没有发现关于本发明的有关报道。
发明内容
本发明人依据中医理论的研究和临床试验的反复验证,终于找到了有效治疗子宫颈癌的药物,从而完成了本发明。
本发明的目的就是提供一种有效治疗子宫颈癌的中药组合药物。
本发明的另一目的就是提供了该中药组合药物的制备方法。
本发明药物是选择土茯苓、贯众、苦参、地榆、牛膝、栀子、黄柏、薏苡仁、黄芪、女贞子、枸杞子、枳壳、莪术、白花蛇舌草、白茅根、当归、昆布、海藻、蚤休、山慈姑、香附、柴胡、全蝎、续断、半枝莲、白芍、茯苓、升麻、生地黄、玄参、沉香、延胡索进行组合制备的,将这些药物组合使得各药物功效产生协同作用,从而能够有效治疗子宫颈癌。其中选用土茯苓是因为其性味甘淡,平,入肝、胃经,有解毒,除湿,利关节的功能,治梅毒,淋浊,筋骨挛痛,脚气,疔疮,痈肿,瘰疬。选用贯众是因为其性味苦,凉,入肝、胃经,有杀蛔、绦、蛲虫,清热,解毒,凉血,止血的功能,治风热感冒,湿热癍疹,吐血,衄血,肠风便血,血痢,血崩,带下。选用苦参是因为其性味苦,寒,入肝、肾、大肠、小肠经,有清热,燥湿,杀虫的功能,治热毒血痢,肠风下血,黄疸,赤白带下,小儿肺炎,疳积,急性扁桃体炎,痔漏,脱肛,皮肤瘙痒,阴疮湿痒,瘰疬,烫伤。选用地榆是因为其性味苦酸、寒。入肝、大肠经。凉血止血,清热解毒。治吐血,衄血,血痢,崩溃,肠风,痔漏,痈肿,湿疹,金疮,烧伤。选用牛膝是因为其性味甘苦酸,平,入肝、肾经,生用散瘀血,消痈肿的功能,治淋病,尿血,经闭,癥瘕,难产,胞衣不下,产后瘀血腹痛,喉痹,痈肿,跌打损伤,熟用补肝肾,强筋骨,治腰膝骨痛,四肢拘挛,痿痹。选用栀子是因为其性味苦,寒,入心、肝、肺、胃经,有清热,泻火,凉血的功能,治热病虚烦不眠,黄疸,淋病,消渴,目赤,咽痛,吐血,衄血,血痢,尿血,热毒疮疡,扭伤肿痛。选用黄柏是因为其性味苦,寒,入肺、胃、肾经,有滋阴降火,润燥滑肠的功能,治烦热消渴,骨蒸劳热,肺热咳嗽,大便燥结,小便不利。选用薏苡仁是因为其性味甘淡,凉,入脾、肺、肾经,有健脾,补肺,清热,湿的功能,治泄泻,湿痹,筋脉拘挛,屈伸不利,水肿,脚气,肺痿,肺痈,肠痈,淋浊,白带。选用黄芪是因为其性味甘,微温,入肺、脾经,生用有益卫固表,利水消肿,托毒,生肌的功能,治自汗,盗汗,血痹,浮肿,痈疽不溃或溃久敛;炙用有补中益气的功能,治内伤劳倦,脾虚泄泻,脱肛,气虚血脱,崩带及一切气衰血虚之症。选用女贞子是因为其性味苦甘,平,入肝、肾经,有补肝肾,强腰膝的功能,治阴虚内热,头晕,目花耳鸣,腰膝酸软,须发早白。选用枸杞子是因为其性味甘,平,有滋肾,润肺,补肝,明目的功能,治肝肾阴亏,腰膝酸软,头晕目眩,目昏多泪,虚劳咳嗽,消渴,遗精。选用枳壳是因为其性味苦辛,凉,入肺、脾、大肠经,有破气,行痰,消积的功能,治胸膈痰滞,胸痞,胁胀,食积,噫气,呕逆,下痢后重,脱肛,子宫脱垂。选用莪术是因为其性味辛、苦,温,归肝、脾经,有行气破血,消积止痛的功能,治癥瘕痞块,瘀血经闭,食积肛痛,跌打肿痛,早期宫颈癌。选用白花蛇舌草是因为其性味苦甘,寒,入心、肝、脾三经,有清热,利湿,解毒的功能,治肺热喘咳,扁桃体炎,咽喉炎,阑尾炎,痢疾,黄疸,盆腔炎,附件炎,痈肿疔疮,毒蛇咬伤。选用白茅根是因为其性味甘、寒,入肺、胃、小肠经,有凉血,止血,清热,利尿的功能,治热病烦渴,吐血,衄血,肺热喘急,胃热哕逆,淋病,小便不利,水肿,黄疸。选用当归是因为其性味甘辛,温,入心、肝、脾经,有补血和血,调经止痛,润燥滑肠的功能,治月经不调,经闭腹痛,癥瘕结聚,崩漏,血虚头痛,眩晕,痿痹,肠燥难便,赤痢后重,痈疽疮疡,金疮,跌扑损伤。选用昆布是因为其性味咸,寒,入胃经,有软坚,行水的功能,治瘰疬,瘿瘤,噎膈,水肿,睾丸肿痛,带下。选用海藻是因为其性味苦咸,寒,入肺、脾、肾经,有软坚,消痰,利水,泄热的功能,治瘰疬,瘿瘤,积聚,水肿,脚气,睾丸肿痛。选用蚤休是因为其性味苦辛,寒,有毒,入心、肝经,有清热解毒,平喘止咳,熄风定惊的功能,治痈肿,疔疮,瘰疬,喉痹,慢性气管炎,小儿惊风抽搐,蛇虫咬伤。选用山慈姑是因为其性味甘微辛,寒,入肝、脾经,有消肿,散结,化痰,解毒的功能,治痈疽疔肿,瘰疬,喉痹肿痛,蛇、虫、狂犬伤。选用香附是因为其性味辛微苦干,平,入肝、三焦经,有理气解郁,止痛调经的功能,治肝胃不和,气郁不舒,胸腹胁肋胀痛,痰饮痞满,月经不调,崩漏带下。选用柴胡是因为其性味苦,凉,入肝、胆经,有和解表里,疏肝,升阳的功能,治寒热往来,胸满胁痛,口苦耳聋,头痛目眩,疟疾,下利脱肛,月经不调,子宫下垂。选用全蝎是因为其性味咸辛,平,有毒,入足厥阴经,有祛风,止痉,通络,解毒的功能,治惊风抽搐,癫癎,中风、半身不遂、口眼喎斜,偏头痛,风湿痹痛,破伤风,淋巴结结核,风疹疮肿。选用续断是因为其性味苦辛,微温,入肝、肾经,有补肝肾,续筋骨,调血脉的功能,治腰背酸痛,足膝无力,胎漏,崩漏,带下,遗精,跌打损伤,金疮,痔漏,痈疽疮肿。选用半枝莲是因为其性味苦,寒,有清热,解毒的功能,治咽喉肿痛,烫伤,跌打损伤,湿疮。选用白芍是因为其性味苦酸,凉,入肝、脾经,有养血柔肝,缓中止痛,敛阴收汗的功能,治胸腹胁肋疼痛,泻痢腹痛,自汗盗汗,阴虚发热,月经不调,崩漏,带下。选用茯苓是因为其性味甘淡,平,入心、脾、肺经,有渗湿利水,益脾和胃,宁心安神的功能,治小便不利水肿胀痛,痰饮咳逆,呕哕,泄泻,遗精,淋浊,惊悸,健忘。选用升麻是因为其性味甘辛微苦,凉,入肺、脾、胃经,有升阳,发表,透疹,解毒的功能,治时气疫劳,头痛寒热,喉痛,口疮疤,斑疹不透,中气下陷,久泻久痢,脱肛,妇女崩带,子宫下坠,痈肿疮毒。选用生地黄是因为其性味甘,寒,归心、肝、肾经,有清热凉血,养阴,生津的功能,治热病烦渴,阴虚内热,骨蒸劳热,内热消渴,吐血,衄血,发斑发疹。选用玄参是因为其性味苦咸,凉,入肺、肾经,有滋阴,降火,除烦,解毒的功能,治热病烦渴,发斑,骨蒸劳热,夜寐不宁,自汗盗汗,津伤便秘,吐血衄血,咽喉肿痛,痈肿,瘰疬。选用沉香是因为其性味辛苦,入肾、脾、胃经,有降气温中,暖肾纳气的功能,治气逆喘息,呕吐呃逆,脘腹胀痛,腰膝虚冷,大肠虚秘,小便气淋,男子精冷。选用延胡索是因为其性味辛苦,温,入肝、胃经,有活血,散瘀,理气,止痛的功能,治心腹腰膝诸痛,月经不调,癥瘕,崩中,产后血晕,恶露不尽,跌打损伤。
具体实施方式
本发明组分的药物用量也是发明人经过大量摸索总结得出的,各组分的用量在下述重量范围内都具有较好的疗效:
土茯苓25-35克,贯众15-25克,苦参15-25克,地榆15-25克,牛膝10-20克,栀子5-15克,黄柏5-15克,薏苡仁15-25克,黄芪15-25克,女贞子15-25克,枸杞子10-20克,枳壳5-15克,莪术10-20克,白花蛇舌草25-35克,白茅根15-25克,当归10-20克,昆布15-25克,海藻15-25克,蚤休10-20克,山慈姑10-20克,香附10-20克,柴胡5-15克,全蝎4-8克,续断15-25克,半枝莲15-25克,白芍10-20克,茯苓10-20克,升麻15-25克,生地黄10-20克,玄参10-20克,沉香4-8克,延胡索10-20克。
优选为:
土茯苓30克,贯众20克,苦参20克,地榆20克,牛膝15克,栀子10克,黄柏10克,薏苡仁20克,黄芪20克,女贞子20克,枸杞子15克,枳壳10克,莪术15克,白花蛇舌草30克,白茅根20克,当归15克,昆布20克,海藻20克,蚤休15克,山慈姑15克,香附15克,柴胡10克,全蝎6克,续断20克,半枝莲20克,白芍15克,茯苓15克,升麻20克,生地黄15克,玄参15克,沉香6克,延胡索15克。
本发明药物的制备方法如下
一、备料
1、土茯苓:用水浸漂,夏季每日换水1次,春、秋每2日换水1次,冬季可3日换水1次,防止发臭,以泡透为度,捞出切片,及时干燥;
2、贯众:用清水稍浸,取出,早晚各洒水一次,润软,切片,晒干;
3、苦参:拣净杂质,除去残茎,洗净泥土,用水浸泡,捞出,润透,切片,晒干;
4、地榆:拣去杂质,用水洗净,稍浸泡,润透,切成厚片,晒干;
5、牛膝:拣去杂质,洗净,润软,去芦,切段,晒干;
6、栀子:筛去灰屑,拣去杂质,碾碎过筛或剪去两端;
7、黄柏:拣去杂质,用水洗净,捞出,润透,切片或切丝,晒干;
8、薏苡仁:取原药材,除去残留皮壳、杂质;
9、黄芪:拣净杂质,除去残留的根头和空心较大的根,用水浸泡,捞出,润透后及时切片,晒干;
10、女贞子:拣去杂质,洗净,晒干;
11、枸杞子:簸净杂质,摘去残留的梗和蒂;
12、枳壳:除去瓤、核,冼净,稍浸,捞出,润软,以手能捏对折为度,切片,晾干;
13、莪术:取原药材,除去杂质,大小分档,洗净,略浸泡,取出,润透,切薄片,干燥,筛去碎屑;
14、白花蛇舌草:取原药材,除去杂质,抢水洗净,稍晾,切段,干燥,筛去灰屑;
15、白茅根:拣净杂质,洗净,微润,切段,晒干,簸净碎屑;
16、当归:拣去杂质,洗净,闷润,稍晾,切片晒干;
17、昆布:拣去杂质,用水漂净,切成宽丝,晾干;
18、海藻:拣去杂质,用水略漂,稍晾,切段,晒干;
19、蚤休:秋季采挖,除去须根,洗净,干燥;
20、山慈姑:除尽须根,洗净,清水浸泡2-4小时,取出润透,切片,晒干;
21、香附:拣去杂质,碾成碎粒,簸去细毛及细末;
22、柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,晒干;
23、全蝎:清水漂去盐质,晒干,或微火焙用;
24、续断:洗净泥沙,除去残留根头,润透后切片晒干,筛去屑;
25、半枝莲:除去杂质,洗净,稍润,切段,干燥;
26、白芍:拣去杂质,分开大小个,用水浸泡至八成透,捞出,晒晾,润至内外湿度均匀,切片,干燥;
27、茯苓:用水浸泡,洗净捞出,闷透后,切片,晒干;
28、升麻:拣去杂质,略泡洗净,捞出,润透,切片,晒干;、
29、生地黄:取原药材,除去杂质,洗净,稍润,切厚片,干燥,筛去碎屑;
30、玄参:拣净杂质,除去芦头,洗净润透,切片,晾干;
31、沉香:刷净,劈成小块,用时捣碎或研成细粉;
32、延胡索:拣去杂质,用水浸泡,洗净,晒晾,润至内外湿度均匀,切片或打碎。
二、制备
1、将所述重量的土茯苓、贯众、苦参、地榆、牛膝、栀子、黄柏、薏苡仁、黄芪、女贞子、枸杞子、枳壳、莪术、白花蛇舌草、白茅根、当归、昆布、海藻、蚤休、山慈姑、香附、柴胡、全蝎、续断、半枝莲、白芍、茯苓、升麻、生地黄、玄参、沉香、延胡索放入煎药容器内,加水8倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
2、将过滤的药渣加水6倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
3、将两次煎煮液混合搅拌均匀,分为4剂服用。
组方中贯众有杀蛔、绦、蛲虫,清热,解毒,凉血,止血的功能为君药;地榆有凉血止血,清热解毒的功能;莪术有行气破血,消积止痛的功能,二者为臣药,三味药共同发挥凉血止血,清热解毒,行气破血,消积止痛的作用,治疗子宫颈癌效力全面,且以凉血止血,清热解毒,行气破血为主可治本,当归有补血和血,调经止痛,润燥滑肠的功能为佐药,香附有理气解郁,止痛调经的功能为使药,与下余诸药是治标。
本发明药物具有凉血止血,清热解毒,行气破血,消积止痛,理气解郁,止痛调经的功能,用于治疗子宫颈癌,疗程短、见效快、治愈后不复发。
以下通过试验例来进一步阐述本发明所述药物的有益效果,这些试验例包括本发明药物的动物毒性试验报告和临床疗效观察资料。
[试验例1]本发明药物的动物毒性试验报告:
取家兔30只,雌雄兼用,体重2.0—2.5kg,分两组,每组15只,其中一组为超剂量试验组,另一组为正常量试验组。超常量组为20ml/kg,正常量为10ml/kg,给药方式为灌胃法给药,每天两次,连服7天,每天观察给药反应,结果表明二组家兔活动、饮食正常,药物无不良毒副作用。
[试验例2]本发明药物的临床疗效观察
1、一般资料
收治子宫颈癌门诊患者共33例。
2、诊断标准
子宫颈癌早期多为接触性出血;中晚期为不规则阴道流血。出血量根据病灶大小、侵及间质内血管情况而不同,若侵袭大血管可引起大出血。年轻患者也可表现为经期延长、经量增多;老年患者常为绝经后不规则阴道流血。一般外生型较早出现阴道出血症状,出血量多;内生型较晚出现该症状。
3、治疗方法
选用上述药剂,给患者服用,每次服用1剂,每天早、晚各服1次,30天为一个疗程,连续服用3个疗程。
4、疗效评定标准
显效:子宫颈癌症状消失,三年未复发;
好转:子宫颈癌症状明显好转,不规则流血、接触性流血量及次数减少,逐步恢复正常;
无效:达不到好转标准者。
5、治疗结果(见下表)
在上述治疗中,用本发明药物治疗子宫颈癌患者33例,结果显效28例,显效率为84.8%,好转3例,好转率为9.1%,无效2例,总有效率为93.9%。
Claims (3)
1.一种治疗子宫颈癌的药物,其特征在于:它是由下列重量范围内的原料药制成:
土茯苓25-35克,贯众15-25克,苦参15-25克,地榆15-25克,牛膝10-20克,栀子5-15克,黄柏5-15克,薏苡仁15-25克,黄芪15-25克,女贞子15-25克,枸杞子10-20克,枳壳5-15克,莪术10-20克,白花蛇舌草25-35克,白茅根15-25克,当归10-20克,昆布15-25克,海藻15-25克,蚤休10-20克,山慈姑10-20克,香附10-20克,柴胡5-15克,全蝎4-8克,续断15-25克,半枝莲15-25克,白芍10-20克,茯苓10-20克,升麻15-25克,生地黄10-20克,玄参10-20克,沉香4-8克,延胡索10-20克。
2.根据权利要求1所述的药物,其中各原料药的用量为:
土茯苓30克,贯众20克,苦参20克,地榆20克,牛膝15克,栀子10克,黄柏10克,薏苡仁20克,黄芪20克,女贞子20克,枸杞子15克,枳壳10克,莪术15克,白花蛇舌草30克,白茅根20克,当归15克,昆布20克,海藻20克,蚤休15克,山慈姑15克,香附15克,柴胡10克,全蝎6克,续断20克,半枝莲20克,白芍15克,茯苓15克,升麻20克,生地黄15克,玄参15克,沉香6克,延胡索15克。
3.根据权利要求1或2所述药物的制备方法,它包括下列步骤:
(一)备料
(1)土茯苓:用水浸漂,夏季每日换水1次,春、秋每2日换水1次,冬季可3日换水1次,防止发臭,以泡透为度,捞出切片,及时干燥;
(2)贯众:用清水稍浸,取出,早晚各洒水一次,润软,切片,晒干;
(3)苦参:拣净杂质,除去残茎,洗净泥土,用水浸泡,捞出,润透,切片,晒干;
(4)地榆:拣去杂质,用水洗净,稍浸泡,润透,切成厚片,晒干;
(5)牛膝:拣去杂质,洗净,润软,去芦,切段,晒干;
(6)栀子:筛去灰屑,拣去杂质,碾碎过筛或剪去两端;
(7)黄柏:拣去杂质,用水洗净,捞出,润透,切片或切丝,晒干;
(8)薏苡仁:取原药材,除去残留皮壳、杂质;
(9)黄芪:拣净杂质,除去残留的根头和空心较大的根,用水浸泡,捞出,润透后及时切片,晒干;
(10)女贞子:拣去杂质,洗净,晒干;
(11)枸杞子:簸净杂质,摘去残留的梗和蒂;
(12)枳壳:除去瓤、核,冼净,稍浸,捞出,润软,以手能捏对折为度,切片,晾干;
(13)莪术:取原药材,除去杂质,大小分档,洗净,略浸泡,取出,润透,切薄片,干燥,筛去碎屑;
(14)白花蛇舌草:取原药材,除去杂质,抢水洗净,稍晾,切段,干燥,筛去灰屑;
(15)白茅根:拣净杂质,洗净,微润,切段,晒干,簸净碎屑;
(16)当归:拣去杂质,洗净,闷润,稍晾,切片晒干;
(17)昆布:拣去杂质,用水漂净,切成宽丝,晾干;
(18)海藻:拣去杂质,用水略漂,稍晾,切段,晒干;
(19)蚤休:秋季采挖,除去须根,洗净,干燥;
(20)山慈姑:除尽须根,洗净,清水浸泡2-4小时,取出润透,切片,晒干;
(21)香附:拣去杂质,碾成碎粒,簸去细毛及细末;
(22)柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,晒干;
(23)全蝎:清水漂去盐质,晒干,或微火焙用;
(24)续断:洗净泥沙,除去残留根头,润透后切片晒干,筛去屑;
(25)半枝莲:除去杂质,洗净,稍润,切段,干燥;
(26)白芍:拣去杂质,分开大小个,用水浸泡至八成透,捞出,晒晾,润至内外湿度均匀,切片,干燥;
(27)茯苓:用水浸泡,洗净捞出,闷透后,切片,晒干;
(28)升麻:拣去杂质,略泡洗净,捞出,润透,切片,晒干;、
(29)生地黄:取原药材,除去杂质,洗净,稍润,切厚片,干燥,筛去碎屑;
(30)玄参:拣净杂质,除去芦头,洗净润透,切片,晾干;
(31)沉香:刷净,劈成小块,用时捣碎或研成细粉;
(32)延胡索:拣去杂质,用水浸泡,洗净,晒晾,润至内外湿度均匀,切片或打碎;
(二)制备
(1)将所述重量的土茯苓、贯众、苦参、地榆、牛膝、栀子、黄柏、薏苡仁、黄芪、女贞子、枸杞子、枳壳、莪术、白花蛇舌草、白茅根、当归、昆布、海藻、蚤休、山慈姑、香附、柴胡、全蝎、续断、半枝莲、白芍、茯苓、升麻、生地黄、玄参、沉香、延胡索放入煎药容器内,加水8倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
(2)将过滤的药渣加水6倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
(3)将两次煎煮液混合搅拌均匀,分为4剂服用。
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