CN104662018B - 取代的杂双环化合物、组合物及其医疗应用 - Google Patents

取代的杂双环化合物、组合物及其医疗应用 Download PDF

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Publication number
CN104662018B
CN104662018B CN201380019452.8A CN201380019452A CN104662018B CN 104662018 B CN104662018 B CN 104662018B CN 201380019452 A CN201380019452 A CN 201380019452A CN 104662018 B CN104662018 B CN 104662018B
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phenyl
pyrrolo
methyl
dihydro
cyclopropyl
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CN104662018A (zh
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M·塔卡
S·考尔
D·布尼亚
K·穆克蒂亚
S·库尔海德
Y·穆努特
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Eurofins Advinus Ltd
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Advinus Therapeutics Pvt Ltd
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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  • Health & Medical Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Immunology (AREA)
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  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
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  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN201380019452.8A 2012-04-20 2013-04-18 取代的杂双环化合物、组合物及其医疗应用 Expired - Fee Related CN104662018B (zh)

Applications Claiming Priority (3)

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IN1573/CHE/2012 2012-04-20
IN1573CH2012 IN2012CH01573A (enExample) 2012-04-20 2013-04-18
PCT/IN2013/000259 WO2013157022A1 (en) 2012-04-20 2013-04-18 Substituted hetero-bicyclic compounds, compositions and medicinal applications thereof

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CN104662018A CN104662018A (zh) 2015-05-27
CN104662018B true CN104662018B (zh) 2017-10-24

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US (1) US9233983B2 (enExample)
EP (1) EP2838898B1 (enExample)
JP (1) JP6182593B2 (enExample)
CN (1) CN104662018B (enExample)
AU (1) AU2013250726B2 (enExample)
CA (1) CA2869954C (enExample)
IL (1) IL235146A (enExample)
IN (1) IN2012CH01573A (enExample)
WO (1) WO2013157022A1 (enExample)
ZA (1) ZA201407341B (enExample)

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