CN103269724A - 生产F-18标记的β-淀粉样蛋白配体的方法 - Google Patents
生产F-18标记的β-淀粉样蛋白配体的方法 Download PDFInfo
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- CN103269724A CN103269724A CN201180027675XA CN201180027675A CN103269724A CN 103269724 A CN103269724 A CN 103269724A CN 201180027675X A CN201180027675X A CN 201180027675XA CN 201180027675 A CN201180027675 A CN 201180027675A CN 103269724 A CN103269724 A CN 103269724A
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- C07C217/78—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
- C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
- C07C217/82—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring
- C07C217/84—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
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- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
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- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
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- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
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- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
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- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
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- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
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Abstract
Description
Claims (13)
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Cited By (2)
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CN105612583A (zh) * | 2013-10-18 | 2016-05-25 | 通用电气健康护理有限公司 | 密闭蒸发系统 |
CN109867591A (zh) * | 2019-03-12 | 2019-06-11 | 浙江大学 | 18f标记的aie荧光/pet双模态探针及其制备方法和应用 |
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CN103328011A (zh) * | 2010-06-04 | 2013-09-25 | 皮拉马影像股份公司 | 生产F-18标记的β-淀粉样蛋白配体的方法 |
SG185782A1 (en) | 2010-06-04 | 2013-01-30 | Piramal Imaging Sa | Method for production of f-18 labeled amyloid beta ligands |
US11504430B2 (en) * | 2010-12-29 | 2022-11-22 | Ge Healthcare Limited | Eluent solution |
PL2723394T3 (pl) | 2011-06-21 | 2018-11-30 | Piramal Imaging Sa | Preparaty fluorowanego stylbenu odpowiednie do zastosowań w obrazowaniu PET |
BR112014009013A2 (pt) * | 2011-10-19 | 2017-05-02 | Piramal Imaging Sa | método melhorado para a produção de ligandos aß rotulados por f-18 |
KR101326000B1 (ko) * | 2012-01-30 | 2013-11-07 | 재단법인 아산사회복지재단 | 수소이온 농도가 조절된 플루오린-18의 용리액 제조 및 이를 이용한 플루오린-18의 표지방법 |
DK3538161T3 (da) * | 2016-11-08 | 2022-09-05 | Univ California | Fremgangsmåder til flerdosissyntese af [F-18]FDDNP til kliniske indstillinger |
JP7241013B2 (ja) * | 2017-03-17 | 2023-03-16 | 日本メジフィジックス株式会社 | イオフルパンの製造方法 |
EA202091767A1 (ru) * | 2018-01-24 | 2021-02-16 | Ац Иммуне Са | Новый способ получения визуализирующего соединения |
WO2024107620A1 (en) * | 2022-11-14 | 2024-05-23 | Eli Lilly And Company | Polymorphic forms of florbetapir precursor av-105 |
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PT1999109E (pt) | 2006-03-30 | 2012-03-16 | Univ Pennsylvania | Derivados de estirilpiridina e sua utilização para ligação e obtenção de imagens de placas amilóides |
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