CN102875441A - Ppar活性化合物 - Google Patents

Ppar活性化合物 Download PDF

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Publication number
CN102875441A
CN102875441A CN2012103274659A CN201210327465A CN102875441A CN 102875441 A CN102875441 A CN 102875441A CN 2012103274659 A CN2012103274659 A CN 2012103274659A CN 201210327465 A CN201210327465 A CN 201210327465A CN 102875441 A CN102875441 A CN 102875441A
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Prior art keywords
indol
propionic acid
benzenesulfonyl
methoxyl group
compound
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CN2012103274659A
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Chinese (zh)
Inventor
J·阿罗尔德
D·R·阿尔蒂
C·赫特
P·N·易卜拉欣
H·克鲁普克
J·林
M·V·米尔本
W·王
C·张
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Plexxikon Inc
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Plexxikon Inc
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Publication of CN102875441A publication Critical patent/CN102875441A/zh
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    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • C04B35/63Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
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    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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CN2012103274659A 2003-07-17 2004-07-16 Ppar活性化合物 Pending CN102875441A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US48852303P 2003-07-17 2003-07-17
US60/488,523 2003-07-17
US55299404P 2004-03-12 2004-03-12
US60/552,994 2004-03-12

Related Parent Applications (1)

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CNA200480025050XA Division CN1845898A (zh) 2003-07-17 2004-07-16 Ppar活性化合物

Publications (1)

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CN102875441A true CN102875441A (zh) 2013-01-16

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CN2012103274659A Pending CN102875441A (zh) 2003-07-17 2004-07-16 Ppar活性化合物

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US (5) US7202266B2 (US07476746-20090113-C00133.png)
EP (1) EP1648867B1 (US07476746-20090113-C00133.png)
JP (1) JP4845730B2 (US07476746-20090113-C00133.png)
KR (2) KR101415503B1 (US07476746-20090113-C00133.png)
CN (1) CN102875441A (US07476746-20090113-C00133.png)
AU (1) AU2004259738B2 (US07476746-20090113-C00133.png)
BR (1) BRPI0412684A (US07476746-20090113-C00133.png)
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IL (1) IL173079A (US07476746-20090113-C00133.png)
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UA (1) UA88767C2 (US07476746-20090113-C00133.png)
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Cited By (1)

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CN115504925A (zh) * 2021-06-22 2022-12-23 广东药科大学 一类新型ppar激动剂、其制备方法及其作为药物的用途

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