CN102838546B - 作为5-ht2a血清素受体调节剂用于治疗与其相关病症的吡唑衍生物 - Google Patents

作为5-ht2a血清素受体调节剂用于治疗与其相关病症的吡唑衍生物 Download PDF

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Publication number
CN102838546B
CN102838546B CN201210300858.0A CN201210300858A CN102838546B CN 102838546 B CN102838546 B CN 102838546B CN 201210300858 A CN201210300858 A CN 201210300858A CN 102838546 B CN102838546 B CN 102838546B
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base
phenyl
compound
piperazine
pyrazoles
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CN102838546A (zh
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熊易峰
马丁.C.谢里耶
金孙.卡洛琳.蔡
彼得.I.多莎
布莱恩.M.史密斯
索尼娅.斯特拉-普莱内特
布雷特.厄尔曼
布拉德利.蒂加登
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Arena Pharmaceuticals Inc
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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CN201210300858.0A 2006-10-03 2007-10-02 作为5-ht2a血清素受体调节剂用于治疗与其相关病症的吡唑衍生物 Expired - Fee Related CN102838546B (zh)

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US84907006P 2006-10-03 2006-10-03
US60/849,070 2006-10-03
CN2007800371033A CN101611013B (zh) 2006-10-03 2007-10-02 作为5-ht2a血清素受体调节剂用于治疗与其相关病症的吡唑衍生物

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CN102838546B true CN102838546B (zh) 2015-07-15

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CN2007800371033A Expired - Fee Related CN101611013B (zh) 2006-10-03 2007-10-02 作为5-ht2a血清素受体调节剂用于治疗与其相关病症的吡唑衍生物

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US (6) US9434692B2 (https=)
EP (1) EP2066641B1 (https=)
JP (2) JP5346292B2 (https=)
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AR (1) AR063100A1 (https=)
AU (1) AU2007305235C1 (https=)
CA (1) CA2664398C (https=)
CL (1) CL2007002859A1 (https=)
ES (1) ES2494846T3 (https=)
JO (1) JO2954B1 (https=)
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