CN102089304A - 作为m3毒蕈碱性受体拮抗剂的奎宁环衍生物 - Google Patents

作为m3毒蕈碱性受体拮抗剂的奎宁环衍生物 Download PDF

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Publication number
CN102089304A
CN102089304A CN2008801303428A CN200880130342A CN102089304A CN 102089304 A CN102089304 A CN 102089304A CN 2008801303428 A CN2008801303428 A CN 2008801303428A CN 200880130342 A CN200880130342 A CN 200880130342A CN 102089304 A CN102089304 A CN 102089304A
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China
Prior art keywords
phenyl
bicyclo
cycloheptanecarbonyloxy
azonium
octane
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Pending
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CN2008801303428A
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Chinese (zh)
Inventor
罗南.L.福特
安德鲁.N.马瑟
安东尼奥.梅特
理查德.J.布尔
伊莉莎白.A.斯基德莫尔
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Pulmagen Therapeutics Synergy Ltd
AstraZeneca AB
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Pulmagen Therapeutics Synergy Ltd
AstraZeneca AB
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Application filed by Pulmagen Therapeutics Synergy Ltd, AstraZeneca AB filed Critical Pulmagen Therapeutics Synergy Ltd
Publication of CN102089304A publication Critical patent/CN102089304A/zh
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CN2008801303428A 2008-05-13 2008-05-13 作为m3毒蕈碱性受体拮抗剂的奎宁环衍生物 Pending CN102089304A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/GB2008/001647 WO2009138707A1 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
CN102089304A true CN102089304A (zh) 2011-06-08

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US (2) US8329729B2 (enExample)
EP (1) EP2300464A1 (enExample)
JP (1) JP4837800B2 (enExample)
CN (1) CN102089304A (enExample)
AU (1) AU2008356409B2 (enExample)
BR (1) BRPI0822693A2 (enExample)
CA (1) CA2723981A1 (enExample)
CL (1) CL2009001137A1 (enExample)
EA (1) EA017627B1 (enExample)
EC (1) ECSP10010606A (enExample)
HN (1) HN2010002403A (enExample)
IL (1) IL209126A0 (enExample)
MX (1) MX2010012189A (enExample)
NI (1) NI201000195A (enExample)
NZ (1) NZ589091A (enExample)
WO (1) WO2009138707A1 (enExample)
ZA (1) ZA201007988B (enExample)

Cited By (2)

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Publication number Priority date Publication date Assignee Title
CN103265478A (zh) * 2013-05-20 2013-08-28 中国人民解放军第二军医大学 巯基烟酸类化合物及其制备方法
CN114716380A (zh) * 2022-04-01 2022-07-08 新乡医学院 一种高效相转移催化的4-取代吡唑酮类化合物不对称氟化方法

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EP2300464A1 (en) 2008-05-13 2011-03-30 AstraZeneca AB Quinuclidine derivatives as muscarinic m3 receptor antagonists
KR20110010725A (ko) * 2008-05-13 2011-02-07 아스트라제네카 아베 무스카린성 수용체 길항제 및 β２­아드레날린수용체 효능제를 포함하는 제약 생성물
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
WO2025171311A1 (en) * 2024-02-09 2025-08-14 University Of Florida Research Foundation, Incorporated Aryl and pyridyl amide pesticides and compositions thereof

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