ZA201007988B - Quinuclidine derivatives as muscarinic m3 receptor antagonists - Google Patents

Quinuclidine derivatives as muscarinic m3 receptor antagonists

Info

Publication number
ZA201007988B
ZA201007988B ZA2010/07988A ZA201007988A ZA201007988B ZA 201007988 B ZA201007988 B ZA 201007988B ZA 2010/07988 A ZA2010/07988 A ZA 2010/07988A ZA 201007988 A ZA201007988 A ZA 201007988A ZA 201007988 B ZA201007988 B ZA 201007988B
Authority
ZA
South Africa
Prior art keywords
muscarinic
receptor antagonists
quinuclidine derivatives
quinuclidine
derivatives
Prior art date
Application number
ZA2010/07988A
Other languages
English (en)
Inventor
Elizabeth Anne Skidmore
Andrew Nigel Mather
Rhonan Lee Ford
Antonio Mete
Richard James Bull
Original Assignee
Pulmagen Therapeutics (Synergy) Ltd
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pulmagen Therapeutics (Synergy) Ltd, Astrazeneca Ab filed Critical Pulmagen Therapeutics (Synergy) Ltd
Publication of ZA201007988B publication Critical patent/ZA201007988B/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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ZA2010/07988A 2008-05-13 2010-11-08 Quinuclidine derivatives as muscarinic m3 receptor antagonists ZA201007988B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/GB2008/001647 WO2009138707A1 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
ZA201007988B true ZA201007988B (en) 2011-07-27

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US (2) US8329729B2 (enExample)
EP (1) EP2300464A1 (enExample)
JP (1) JP4837800B2 (enExample)
CN (1) CN102089304A (enExample)
AU (1) AU2008356409B2 (enExample)
BR (1) BRPI0822693A2 (enExample)
CA (1) CA2723981A1 (enExample)
CL (1) CL2009001137A1 (enExample)
EA (1) EA017627B1 (enExample)
EC (1) ECSP10010606A (enExample)
HN (1) HN2010002403A (enExample)
IL (1) IL209126A0 (enExample)
MX (1) MX2010012189A (enExample)
NI (1) NI201000195A (enExample)
NZ (1) NZ589091A (enExample)
WO (1) WO2009138707A1 (enExample)
ZA (1) ZA201007988B (enExample)

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CN102908624A (zh) * 2008-05-13 2013-02-06 阿斯利康(瑞典)有限公司 包含毒蕈碱性受体拮抗剂和β2-肾上腺素受体激动剂的药物产品
JP4837800B2 (ja) 2008-05-13 2011-12-14 アストラゼネカ・アクチエボラーグ ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
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CN103265478B (zh) * 2013-05-20 2015-09-30 中国人民解放军第二军医大学 巯基烟酸类化合物及其制备方法
CN114716380B (zh) * 2022-04-01 2024-06-21 新乡医学院 一种相转移催化的4-取代吡唑酮类化合物不对称氟化方法
WO2025171311A1 (en) * 2024-02-09 2025-08-14 University Of Florida Research Foundation, Incorporated Aryl and pyridyl amide pesticides and compositions thereof

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AU2008356409B2 (en) 2012-01-19
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WO2009138707A9 (en) 2010-01-28
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CL2009001137A1 (es) 2009-11-27
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EA017627B1 (ru) 2013-01-30
NZ589091A (en) 2011-07-29
IL209126A0 (en) 2011-01-31
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US8329729B2 (en) 2012-12-11
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CA2723981A1 (en) 2009-11-19
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EA201001645A1 (ru) 2011-06-30
HN2010002403A (es) 2013-01-28

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