BRPI0822693A2 - Derivados de quinuclidina como antagonistas do receptor muscarínico m3 - Google Patents

Derivados de quinuclidina como antagonistas do receptor muscarínico m3

Info

Publication number
BRPI0822693A2
BRPI0822693A2 BRPI0822693-8A BRPI0822693A BRPI0822693A2 BR PI0822693 A2 BRPI0822693 A2 BR PI0822693A2 BR PI0822693 A BRPI0822693 A BR PI0822693A BR PI0822693 A2 BRPI0822693 A2 BR PI0822693A2
Authority
BR
Brazil
Prior art keywords
receptor antagonists
muscarinic receptor
quinuclidine derivatives
quinuclidine
derivatives
Prior art date
Application number
BRPI0822693-8A
Other languages
English (en)
Portuguese (pt)
Inventor
Rhonan Lee Ford
Andrew Nigel Mather
Antonio Mete
Richard James Bull
Elizabeth Anne Skidmore
Original Assignee
Astrazeneca Ab
Pulmagen Therapeutics Synergy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab, Pulmagen Therapeutics Synergy filed Critical Astrazeneca Ab
Publication of BRPI0822693A2 publication Critical patent/BRPI0822693A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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BRPI0822693-8A 2008-05-13 2008-05-13 Derivados de quinuclidina como antagonistas do receptor muscarínico m3 BRPI0822693A2 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/GB2008/001647 WO2009138707A1 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
BRPI0822693A2 true BRPI0822693A2 (pt) 2015-07-07

Family

ID=40361403

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0822693-8A BRPI0822693A2 (pt) 2008-05-13 2008-05-13 Derivados de quinuclidina como antagonistas do receptor muscarínico m3

Country Status (17)

Country Link
US (2) US8329729B2 (enExample)
EP (1) EP2300464A1 (enExample)
JP (1) JP4837800B2 (enExample)
CN (1) CN102089304A (enExample)
AU (1) AU2008356409B2 (enExample)
BR (1) BRPI0822693A2 (enExample)
CA (1) CA2723981A1 (enExample)
CL (1) CL2009001137A1 (enExample)
EA (1) EA017627B1 (enExample)
EC (1) ECSP10010606A (enExample)
HN (1) HN2010002403A (enExample)
IL (1) IL209126A0 (enExample)
MX (1) MX2010012189A (enExample)
NI (1) NI201000195A (enExample)
NZ (1) NZ589091A (enExample)
WO (1) WO2009138707A1 (enExample)
ZA (1) ZA201007988B (enExample)

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TW200825084A (en) * 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
MX2010012019A (es) * 2008-05-13 2011-03-04 Astrazeneca Ab Producto farmaceutico que comprende un antagonista receptor muscarinico y un agonista de adrenoceptor beta2.
JP4837800B2 (ja) 2008-05-13 2011-12-14 アストラゼネカ・アクチエボラーグ ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
CN103265478B (zh) * 2013-05-20 2015-09-30 中国人民解放军第二军医大学 巯基烟酸类化合物及其制备方法
CN114716380B (zh) * 2022-04-01 2024-06-21 新乡医学院 一种相转移催化的4-取代吡唑酮类化合物不对称氟化方法
WO2025171311A1 (en) * 2024-02-09 2025-08-14 University Of Florida Research Foundation, Incorporated Aryl and pyridyl amide pesticides and compositions thereof

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FR2155927A1 (en) 1971-10-15 1973-05-25 Synthelabo 1-phenylcyclo hexane carboxylic acid esters - with antispasmodic and anticholinergic activity
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FR2208649A1 (en) 1972-12-01 1974-06-28 Synthelabo 1-(2-Thienyl)cycloalkane carboxylic ester salts - with spasmolytic and anticholinergic activity
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US20110172237A1 (en) 2011-07-14
CA2723981A1 (en) 2009-11-19
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US20130030001A1 (en) 2013-01-31
AU2008356409B2 (en) 2012-01-19
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CN102089304A (zh) 2011-06-08
AU2008356409A1 (en) 2009-11-19
WO2009138707A1 (en) 2009-11-19
EA201001645A1 (ru) 2011-06-30
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EA017627B1 (ru) 2013-01-30
CL2009001137A1 (es) 2009-11-27

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