JP4837800B2 - ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体 - Google Patents

ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体 Download PDF

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JP4837800B2
JP4837800B2 JP2011508991A JP2011508991A JP4837800B2 JP 4837800 B2 JP4837800 B2 JP 4837800B2 JP 2011508991 A JP2011508991 A JP 2011508991A JP 2011508991 A JP2011508991 A JP 2011508991A JP 4837800 B2 JP4837800 B2 JP 4837800B2
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phenyl
bicyclo
cycloheptanecarbonyloxy
azonia
methyl
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JP2011520853A5 (enExample
JP2011520853A (ja
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ローナン・リー・フォード
アンドリュー・ナイジェル・メーザー
アントニオ・メーテ
リチャード・ジェイムズ・ブル
エリザベス・アン・スキッドモア
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Pulmagen Therapeutics Synergy Ltd
AstraZeneca AB
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Pulmagen Therapeutics Synergy Ltd
AstraZeneca AB
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    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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JP2011508991A 2008-05-13 2008-05-13 ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体 Expired - Fee Related JP4837800B2 (ja)

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PCT/GB2008/001647 WO2009138707A1 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as muscarinic m3 receptor antagonists

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JP2011520853A5 JP2011520853A5 (enExample) 2011-09-29
JP4837800B2 true JP4837800B2 (ja) 2011-12-14

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CN (1) CN102089304A (enExample)
AU (1) AU2008356409B2 (enExample)
BR (1) BRPI0822693A2 (enExample)
CA (1) CA2723981A1 (enExample)
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US5807670A (en) * 1995-08-14 1998-09-15 Abbott Laboratories Detection of hepatitis GB virus genotypes
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
NZ589091A (en) 2008-05-13 2011-07-29 Astrazeneca Ab Quinuclidine derivatives as muscarinic m3 receptor antagonists
CN102908624A (zh) * 2008-05-13 2013-02-06 阿斯利康(瑞典)有限公司 包含毒蕈碱性受体拮抗剂和β2-肾上腺素受体激动剂的药物产品
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
CN103265478B (zh) * 2013-05-20 2015-09-30 中国人民解放军第二军医大学 巯基烟酸类化合物及其制备方法
CN114716380B (zh) * 2022-04-01 2024-06-21 新乡医学院 一种相转移催化的4-取代吡唑酮类化合物不对称氟化方法
WO2025171311A1 (en) * 2024-02-09 2025-08-14 University Of Florida Research Foundation, Incorporated Aryl and pyridyl amide pesticides and compositions thereof

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CL2009001137A1 (es) 2009-11-27
EA201001645A1 (ru) 2011-06-30
CA2723981A1 (en) 2009-11-19
CN102089304A (zh) 2011-06-08
HN2010002403A (es) 2013-01-28
ZA201007988B (en) 2011-07-27
MX2010012189A (es) 2011-03-02
NZ589091A (en) 2011-07-29
AU2008356409A1 (en) 2009-11-19
AU2008356409B2 (en) 2012-01-19
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US8329729B2 (en) 2012-12-11
US20110172237A1 (en) 2011-07-14
IL209126A0 (en) 2011-01-31
EP2300464A1 (en) 2011-03-30
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JP2011520853A (ja) 2011-07-21
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