CN101518517B - 药物剂量逐渐增加的剂型 - Google Patents
药物剂量逐渐增加的剂型 Download PDFInfo
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- CN101518517B CN101518517B CN200910129895.8A CN200910129895A CN101518517B CN 101518517 B CN101518517 B CN 101518517B CN 200910129895 A CN200910129895 A CN 200910129895A CN 101518517 B CN101518517 B CN 101518517B
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- MLICVSDCCDDWMD-KVVVOXFISA-M potassium;(z)-octadec-9-enoate Chemical compound [K+].CCCCCCCC\C=C/CCCCCCCC([O-])=O MLICVSDCCDDWMD-KVVVOXFISA-M 0.000 description 1
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- KWGRBVOPPLSCSI-WCBMZHEXSA-N pseudoephedrine Chemical compound CN[C@@H](C)[C@@H](O)C1=CC=CC=C1 KWGRBVOPPLSCSI-WCBMZHEXSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2328696P | 1996-08-16 | 1996-08-16 | |
| US60/023,286 | 1996-08-16 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB97197439XA Division CN100484518C (zh) | 1996-08-16 | 1997-08-08 | 药物剂量逐渐增加的剂型 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN101518517A CN101518517A (zh) | 2009-09-02 |
| CN101518517B true CN101518517B (zh) | 2014-11-26 |
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB97197439XA Expired - Lifetime CN100484518C (zh) | 1996-08-16 | 1997-08-08 | 药物剂量逐渐增加的剂型 |
| CN200910129895.8A Expired - Lifetime CN101518517B (zh) | 1996-08-16 | 1997-08-08 | 药物剂量逐渐增加的剂型 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB97197439XA Expired - Lifetime CN100484518C (zh) | 1996-08-16 | 1997-08-08 | 药物剂量逐渐增加的剂型 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0957899B1 (enExample) |
| JP (1) | JP4393587B2 (enExample) |
| CN (2) | CN100484518C (enExample) |
| AT (1) | ATE234602T1 (enExample) |
| AU (1) | AU3909597A (enExample) |
| CA (1) | CA2263558A1 (enExample) |
| CY (1) | CY2475B1 (enExample) |
| DE (1) | DE69720055T2 (enExample) |
| DK (1) | DK0957899T3 (enExample) |
| ES (1) | ES2194210T3 (enExample) |
| PT (1) | PT957899E (enExample) |
| WO (1) | WO1998006380A2 (enExample) |
| ZA (1) | ZA977254B (enExample) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6440457B1 (en) | 1993-05-27 | 2002-08-27 | Alza Corporation | Method of administering antidepressant dosage form |
| US5837284A (en) | 1995-12-04 | 1998-11-17 | Mehta; Atul M. | Delivery of multiple doses of medications |
| EP1690531A3 (en) * | 1996-09-30 | 2010-01-20 | Alza Corporation | Dosage form and method for administering drug |
| EP0932388B1 (en) * | 1996-09-30 | 2006-03-29 | Alza Corporation | Dosage form and method for administering drug |
| US6919373B1 (en) | 1996-11-12 | 2005-07-19 | Alza Corporation | Methods and devices for providing prolonged drug therapy |
| CN1182839C (zh) * | 1996-11-25 | 2005-01-05 | 阿尔萨公司 | 递增剂量的剂型 |
| US6962997B1 (en) | 1997-05-22 | 2005-11-08 | Celgene Corporation | Process and intermediates for resolving piperidyl acetamide steroisomers |
| DE69920689T2 (de) * | 1998-06-03 | 2005-02-24 | Alza Corp., Mountain View | Vorrichtungen zum Aufrechterhalten eines gewünschten therapeutischen Medikamenteneffekts über einen verlängerten Therapiezeitraum |
| AU2012232984B2 (en) * | 1998-06-03 | 2015-10-29 | Alza Corporation | Methods and devices for providing prolonged drug therapy |
| KR100827254B1 (ko) * | 1998-06-03 | 2008-05-07 | 알자 코포레이션 | 연장된 약물 치료를 제공하기 위한 방법 및 장치 |
| KR100890537B1 (ko) * | 1998-06-03 | 2009-03-27 | 알자 코포레이션 | 연장된 약물 치료를 제공하기 위한 방법 및 장치 |
| AU2004200938B2 (en) * | 1998-06-03 | 2006-09-14 | Alza Corporation | Methods and devices for providing prolonged drug therapy |
| HU230454B1 (hu) | 1998-11-02 | 2016-07-28 | Alkermes Pharma Ireland Limited | Metilfenidátot tartalmazó módosított felszabadulású sokszemcsés készítmény |
| US6673367B1 (en) * | 1998-12-17 | 2004-01-06 | Euro-Celtique, S.A. | Controlled/modified release oral methylphenidate formulations |
| US6419960B1 (en) | 1998-12-17 | 2002-07-16 | Euro-Celtique S.A. | Controlled release formulations having rapid onset and rapid decline of effective plasma drug concentrations |
| US6217904B1 (en) | 1999-04-06 | 2001-04-17 | Pharmaquest Ltd. | Pharmaceutical dosage form for pulsatile delivery of d-threo-methylphenidate and a second CNS stimulant |
| JP2004508278A (ja) * | 2000-01-20 | 2004-03-18 | デルシス ファーマシューティカル コーポレイション | 多段薬物投与形態 |
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| JP2006507305A (ja) * | 2002-10-31 | 2006-03-02 | アルザ・コーポレーシヨン | 液体製剤の上昇型放出を提供する剤形 |
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| US20070259033A1 (en) * | 2003-09-26 | 2007-11-08 | Evangeline Cruz | Controlled release formulations exhibiting an ascending rate of release |
| US8541026B2 (en) | 2004-09-24 | 2013-09-24 | Abbvie Inc. | Sustained release formulations of opioid and nonopioid analgesics |
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| WO2015001488A1 (en) | 2013-07-01 | 2015-01-08 | Ranbaxy Laboratories Limited | Extended-release tablets of paliperidone and processes of preparation thereof |
| CA2936748C (en) | 2014-10-31 | 2017-08-08 | Purdue Pharma | Methods and compositions particularly for treatment of attention deficit disorder |
| MX2018007977A (es) * | 2015-12-31 | 2018-11-09 | Cadila Healthcare Ltd | Forma farmaceutica osmotica de liberacion extendida que contiene una carga de clorhidrato de metilfenidato alta. |
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| US4915954A (en) * | 1987-09-03 | 1990-04-10 | Alza Corporation | Dosage form for delivering a drug at two different rates |
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| US4327725A (en) * | 1980-11-25 | 1982-05-04 | Alza Corporation | Osmotic device with hydrogel driving member |
| US4842867A (en) * | 1986-05-09 | 1989-06-27 | Alza Corporation | Pulsed drug delivery of doxylamine |
| GB2206046B (en) * | 1987-06-25 | 1991-04-03 | Alza Corp | Multi-unit delivery system |
| US4874388A (en) * | 1987-06-25 | 1989-10-17 | Alza Corporation | Multi-layer delivery system |
| US4814181A (en) * | 1987-09-03 | 1989-03-21 | Alza Corporation | Dosage form comprising fast agent delivery followed by slow agent delivery |
| US5017381A (en) * | 1990-05-02 | 1991-05-21 | Alza Corporation | Multi-unit pulsatile delivery system |
| PT621032E (pt) * | 1993-04-23 | 2001-01-31 | Novartis Ag | Dispositivo de distribuicao de libertacao controlada de farmaco |
| GB9402203D0 (en) * | 1994-02-04 | 1994-03-30 | Smithkline Beecham Plc | Pharmaceutical formulation |
-
1997
- 1997-08-08 WO PCT/US1997/013816 patent/WO1998006380A2/en not_active Ceased
- 1997-08-08 AT AT97936421T patent/ATE234602T1/de active
- 1997-08-08 EP EP97936421A patent/EP0957899B1/en not_active Expired - Lifetime
- 1997-08-08 JP JP50984198A patent/JP4393587B2/ja not_active Expired - Lifetime
- 1997-08-08 DE DE69720055T patent/DE69720055T2/de not_active Expired - Lifetime
- 1997-08-08 DK DK97936421T patent/DK0957899T3/da active
- 1997-08-08 AU AU39095/97A patent/AU3909597A/en not_active Abandoned
- 1997-08-08 PT PT97936421T patent/PT957899E/pt unknown
- 1997-08-08 CN CNB97197439XA patent/CN100484518C/zh not_active Expired - Lifetime
- 1997-08-08 CN CN200910129895.8A patent/CN101518517B/zh not_active Expired - Lifetime
- 1997-08-08 ES ES97936421T patent/ES2194210T3/es not_active Expired - Lifetime
- 1997-08-08 CA CA002263558A patent/CA2263558A1/en not_active Abandoned
- 1997-08-13 ZA ZA9707254A patent/ZA977254B/xx unknown
-
2004
- 2004-08-27 CY CY0400067A patent/CY2475B1/xx unknown
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4915954A (en) * | 1987-09-03 | 1990-04-10 | Alza Corporation | Dosage form for delivering a drug at two different rates |
Also Published As
| Publication number | Publication date |
|---|---|
| ATE234602T1 (de) | 2003-04-15 |
| DK0957899T3 (da) | 2003-04-22 |
| ES2194210T3 (es) | 2003-11-16 |
| WO1998006380A3 (en) | 1998-05-14 |
| AU3909597A (en) | 1998-03-06 |
| EP0957899A2 (en) | 1999-11-24 |
| JP4393587B2 (ja) | 2010-01-06 |
| ZA977254B (en) | 1998-05-11 |
| CN101518517A (zh) | 2009-09-02 |
| PT957899E (pt) | 2003-07-31 |
| HK1137355A1 (zh) | 2010-07-30 |
| CN100484518C (zh) | 2009-05-06 |
| CN1228691A (zh) | 1999-09-15 |
| DE69720055T2 (de) | 2003-09-11 |
| DE69720055D1 (de) | 2003-04-24 |
| JP2000516610A (ja) | 2000-12-12 |
| HK1021886A1 (zh) | 2000-07-14 |
| EP0957899B1 (en) | 2003-03-19 |
| WO1998006380A2 (en) | 1998-02-19 |
| CY2475B1 (en) | 2005-06-03 |
| CA2263558A1 (en) | 1998-02-19 |
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