CN101506167A - 病毒聚合酶抑制剂 - Google Patents

病毒聚合酶抑制剂 Download PDF

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Publication number
CN101506167A
CN101506167A CNA2007800306227A CN200780030622A CN101506167A CN 101506167 A CN101506167 A CN 101506167A CN A2007800306227 A CNA2007800306227 A CN A2007800306227A CN 200780030622 A CN200780030622 A CN 200780030622A CN 101506167 A CN101506167 A CN 101506167A
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alkyl
het
compound
independently
cycloalkyl
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Chinese (zh)
Inventor
皮埃尔·L·博利厄
勒内·库洛姆比
古尔雷兹·法扎尔
西尔维·古勒特
马丁·波伊里尔
琼·兰考特
蒂莫西·斯坦默斯
邦克哈姆·萨沃内卡姆
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Boehringer Ingelheim International GmbH
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Boehringer Ingelheim International GmbH
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Publication of CN101506167A publication Critical patent/CN101506167A/zh
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/63—One oxygen atom
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CN103130709B (zh) * 2011-11-22 2017-04-12 常州亚邦制药有限公司 具有抗hiv活性的3‑氨基丙酸哌啶酰胺类化合物，合成方法及用途
CN103601671A (zh) * 2013-10-22 2014-02-26 上海泰坦科技股份有限公司 碘代三氟甲基吡啶的制备方法

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