CH629823A5 - Derives steroides substitues en 11beta et leur procede de preparation. - Google Patents

Derives steroides substitues en 11beta et leur procede de preparation. Download PDF

Info

Publication number
CH629823A5
CH629823A5 CH38978A CH38978A CH629823A5 CH 629823 A5 CH629823 A5 CH 629823A5 CH 38978 A CH38978 A CH 38978A CH 38978 A CH38978 A CH 38978A CH 629823 A5 CH629823 A5 CH 629823A5
Authority
CH
Switzerland
Prior art keywords
radical
carbon atoms
formula
group
compounds
Prior art date
Application number
CH38978A
Other languages
English (en)
French (fr)
Inventor
Jean Georges Teutsch
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of CH629823A5 publication Critical patent/CH629823A5/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/006—Ketals at position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
CH38978A 1977-01-13 1978-01-13 Derives steroides substitues en 11beta et leur procede de preparation. CH629823A5 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7700857A FR2377417A1 (fr) 1977-01-13 1977-01-13 Nouveaux derives steroides substitues en 11b, ainsi que leur procede de preparation

Publications (1)

Publication Number Publication Date
CH629823A5 true CH629823A5 (fr) 1982-05-14

Family

ID=9185436

Family Applications (1)

Application Number Title Priority Date Filing Date
CH38978A CH629823A5 (fr) 1977-01-13 1978-01-13 Derives steroides substitues en 11beta et leur procede de preparation.

Country Status (14)

Country Link
US (1) US4147695A (US07413550-20080819-C00001.png)
JP (1) JPS5390253A (US07413550-20080819-C00001.png)
BE (1) BE862868A (US07413550-20080819-C00001.png)
CA (1) CA1122971A (US07413550-20080819-C00001.png)
CH (1) CH629823A5 (US07413550-20080819-C00001.png)
DE (1) DE2801415A1 (US07413550-20080819-C00001.png)
DK (1) DK164324C (US07413550-20080819-C00001.png)
FR (1) FR2377417A1 (US07413550-20080819-C00001.png)
GB (1) GB1595131A (US07413550-20080819-C00001.png)
HU (1) HU175290B (US07413550-20080819-C00001.png)
IE (1) IE46300B1 (US07413550-20080819-C00001.png)
LU (1) LU78860A1 (US07413550-20080819-C00001.png)
NL (1) NL7800365A (US07413550-20080819-C00001.png)
SE (1) SE440780B (US07413550-20080819-C00001.png)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE23167T1 (de) * 1981-01-09 1986-11-15 Roussel Uclaf In stellung 11 substituierte steroidzwischenprodukte und verfahren zu ihrer herstellung.
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1 (fr) * 1982-03-01 1986-02-14 Roussel Uclaf Nouveaux produits derives de la structure 3-ceto 4,9 19-nor steroides, leur procede de preparation et leur application comme medicaments
FR2586021B1 (fr) * 1985-08-09 1988-10-14 Roussel Uclaf Nouveaux produits derives de la structure 5a-oh d 9(10) 19-nor steroides
US5929262A (en) * 1995-03-30 1999-07-27 The United States Of America As Represented By The Department Of Health And Human Services Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2880233A (en) * 1956-01-05 1959-03-31 Sterling Drug Inc Compounds of the perhydrochrysene and related series and preparation thereof
US3299108A (en) * 1965-10-18 1967-01-17 Searle & Co 17alpha-alkynyl/alkenyl-13beta-alkyl-11-alkylgona-1, 3, 5 (10)-triene-3, 17beta-diols, ethers and esters thereof and intermediates thereto
US3346602A (en) * 1966-10-12 1967-10-10 Searle & Co 13beta-alkyl-11-alkylgona-1, 3, 5 (10)-trien-17-ones, ethers and esters thereof
FR2235949B1 (US07413550-20080819-C00001.png) * 1973-06-18 1978-03-17 Roussel Uclaf
FR2237906A1 (en) * 1973-06-26 1975-02-14 Roussel Uclaf 11-oxo estr-9-ene derivs. - intermediates in the synthesis of steroids

Also Published As

Publication number Publication date
IE46300B1 (en) 1983-04-20
BE862868A (fr) 1978-07-12
DK164324C (da) 1992-11-02
LU78860A1 (US07413550-20080819-C00001.png) 1978-09-18
SE440780B (sv) 1985-08-19
CA1122971A (fr) 1982-05-04
FR2377417A1 (fr) 1978-08-11
IE780077L (en) 1978-07-13
JPS5390253A (en) 1978-08-08
FR2377417B1 (US07413550-20080819-C00001.png) 1979-04-20
HU175290B (hu) 1980-06-28
GB1595131A (en) 1981-08-05
DE2801415A1 (de) 1978-07-20
JPS631320B2 (US07413550-20080819-C00001.png) 1988-01-12
DK13778A (da) 1978-07-14
US4147695A (en) 1979-04-03
SE7714612L (sv) 1978-07-14
DK164324B (da) 1992-06-09
NL7800365A (nl) 1978-07-17

Similar Documents

Publication Publication Date Title
CH633811A5 (fr) Derives steroides 4,9-dieniques 11beta-substitues, procede de preparation et compositions pharmaceutiques.
CH657368A5 (fr) Derives de 3-ceto delta-4,9 19-nor-steroides, leur preparation, les compositions les renfermant et les produits de depart pour leur preparation.
EP0280618B1 (fr) Nouveaux 19-nor stéroîdes substitués en position 7, leur préparation, leur application comme médicaments, les compositions pharmaceutiques les renfermant
CH630646A5 (fr) Derives steroides 11 beta-substitues 1,3,5(10)-trieniques, procede de preparation et compositions pharmaceutiques.
EP0558416B1 (fr) Nouveaux stéroides comportant en position 17 un radical méthylène lactone, leur procédé et des intermédiaires de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant
EP0056000B1 (fr) Dérivés 17/(alkoxycarbonyle) (formamido) méthylène/stéroides et leur préparation
EP0313960B1 (fr) Nouveaux stéroides substitués en position 10 par un radical comportant une double ou triple liaison et leur procédé de préparation
CH629823A5 (fr) Derives steroides substitues en 11beta et leur procede de preparation.
CH652726A5 (fr) Derives steroides 17-oxazolines, leur procede de preparation et leur utilisation a la preparation de corticosteroides.
CA1140110A (fr) Procede de preparation de nouveaux derives de l'androst-4-ene
EP0001029B1 (fr) Procédé de préparation d'oximes en 3 de stéroides
EP0192288B1 (fr) Nouveaux dérivés stéroides portant en 17 un radical nitrométhylène, Leur application à la préparation de produits biologiquement actifs
CH641814A5 (fr) Derives acetyleniques de l'androst-4-ene, leurs procedes de preparation et medicaments les renfermant.
CA1146531A (fr) Procede de preparation de nouveaux derives 2,2- dimethyl 19-nor steroides
EP0608178A1 (fr) Nouveau procédé de préparation de stéroides 16alpha-méthylés
CH665423A5 (fr) Steroides, leur procede de preparation, leur utilisation et intermediaires de cette utilisation.
EP0000300B1 (fr) Estra-1,3,5(10),6-tétraènes substitués, procédé de préparation et application dans la synthèse de stéroides marqués au tritium
EP0110434B1 (fr) Nouveaux produits intermédiaires stéroides substitués en 11-beta et procédé de préparation de ces produits
EP0003090B1 (fr) Nouveaux dérivés stéroides 17 alpha-aryle ou 17 alpha-hétéroaryle, leur procédé de préparation et leur application comme médicaments et les compositions pharmaceutiques les renfermant
CH627193A5 (US07413550-20080819-C00001.png)
CH633714A5 (fr) Derives 17alpha-acetyleniques de l'androst 4-ene, procede de prepararation et compositions pharmaceutiques.
CH646983A5 (fr) Derives acetyleniques chlores de l'androst-4-ene, leur preparation et medicaments les renfermant.
CA1199907A (fr) PROCEDE POUR LA PREPARATION DE DERIVES DE STEROIDES HYDROXYLES EN 5.alpha., ET LES DERIVES AINSI OBTENUS
CH633564A5 (fr) Derives du pregn 4-ene, procede de preparation et compositions pharmaceutiques.
CH629826A5 (en) Steroids, process for preparing them and their use in the synthesis of tritium-labelled steroids

Legal Events

Date Code Title Description
PL Patent ceased