CA2850763A1 - Novel quinoxaline inhibitors of pi3k - Google Patents
Novel quinoxaline inhibitors of pi3k Download PDFInfo
- Publication number
- CA2850763A1 CA2850763A1 CA2850763A CA2850763A CA2850763A1 CA 2850763 A1 CA2850763 A1 CA 2850763A1 CA 2850763 A CA2850763 A CA 2850763A CA 2850763 A CA2850763 A CA 2850763A CA 2850763 A1 CA2850763 A1 CA 2850763A1
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- CA
- Canada
- Prior art keywords
- group
- optionally substituted
- nhc
- 3alkylenen
- 4alkylenec
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Landscapes
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| JP5731978B2 (ja) * | 2008-09-26 | 2015-06-10 | インテリカイン， エルエルシー | 複素環キナーゼ阻害剤 |
| WO2011074560A1 (ja) * | 2009-12-15 | 2011-06-23 | 塩野義製薬株式会社 | 血管内皮リパーゼ阻害活性を有するオキサジアゾール誘導体 |
| CA2812089C (en) * | 2010-09-14 | 2020-02-18 | Exelixis Inc. | Inhibitors of pi3k-delta and methods of their use and manufacture |
-
2012
- 2012-10-04 AU AU2012318580A patent/AU2012318580A1/en not_active Abandoned
- 2012-10-04 JP JP2014534732A patent/JP2014528451A/ja active Pending
- 2012-10-04 CN CN201280049200.5A patent/CN104024257A/zh active Pending
- 2012-10-04 WO PCT/US2012/058800 patent/WO2013052699A2/en not_active Ceased
- 2012-10-04 EP EP12838127.4A patent/EP2763994A4/en not_active Withdrawn
- 2012-10-04 US US14/350,039 patent/US20140235643A1/en not_active Abandoned
- 2012-10-04 CA CA2850763A patent/CA2850763A1/en not_active Abandoned
- 2012-10-04 HK HK15101538.0A patent/HK1201065A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2013052699A3 (en) | 2013-06-06 |
| AU2012318580A1 (en) | 2014-05-22 |
| US20140235643A1 (en) | 2014-08-21 |
| EP2763994A2 (en) | 2014-08-13 |
| JP2014528451A (ja) | 2014-10-27 |
| CN104024257A (zh) | 2014-09-03 |
| HK1201065A1 (en) | 2015-08-21 |
| EP2763994A4 (en) | 2015-08-26 |
| WO2013052699A2 (en) | 2013-04-11 |
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