CA2701581C - Pyrimidine substituted purine derivatives - Google Patents
Pyrimidine substituted purine derivatives Download PDFInfo
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- CA2701581C CA2701581C CA2701581A CA2701581A CA2701581C CA 2701581 C CA2701581 C CA 2701581C CA 2701581 A CA2701581 A CA 2701581A CA 2701581 A CA2701581 A CA 2701581A CA 2701581 C CA2701581 C CA 2701581C
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
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| US61/075,532 | 2008-06-25 | ||
| PCT/SG2008/000379 WO2009045175A1 (en) | 2007-10-05 | 2008-10-03 | Pyrimidine substituted purine derivatives |
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| EA037871B1 (ru) * | 2016-06-16 | 2021-05-28 | Янссен Фармацевтика Нв | Производные азабензимидазола в качестве ингибиторов pi3k beta |
| CA3045596C (en) | 2016-12-02 | 2022-08-23 | Daiichi Sankyo Company, Limited | Endo-.beta.-n-acetylglucosaminidase |
| AU2018244011A1 (en) * | 2017-03-31 | 2019-11-07 | Ftg Bio Llc | Salt forms of amino pyrazine purine based selective kinase inhibitor |
| RS65386B1 (sr) | 2017-04-14 | 2024-04-30 | Biogen Ma Inc | Benzoazepinski analozi kao sredstva za inhibiciju brutonove tirozin kinaze |
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2008
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- 2008-10-03 MY MYPI20101500 patent/MY150993A/en unknown
- 2008-10-03 RU RU2010117737/04A patent/RU2518098C2/ru not_active IP Right Cessation
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- 2008-10-03 WO PCT/SG2008/000379 patent/WO2009045175A1/en not_active Ceased
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- 2008-10-03 CA CA2701581A patent/CA2701581C/en not_active Expired - Fee Related
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- 2008-10-03 KR KR1020167026687A patent/KR20160116045A/ko not_active Withdrawn
- 2008-10-03 MX MX2010003668A patent/MX2010003668A/es active IP Right Grant
- 2008-10-03 KR KR1020157013280A patent/KR101701109B1/ko not_active Expired - Fee Related
- 2008-10-03 BR BRPI0817503A patent/BRPI0817503B8/pt not_active IP Right Cessation
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2010
- 2010-03-28 IL IL204804A patent/IL204804A/en active IP Right Grant
- 2010-05-04 ZA ZA2010/03118A patent/ZA201003118B/en unknown
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2012
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2013
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- 2014-11-06 IL IL235555A patent/IL235555B/en active IP Right Grant
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|---|---|---|---|
| EEER | Examination request |
Effective date: 20130925 |
|
| MKLA | Lapsed |
Effective date: 20201005 |