CA2548172A1

CA2548172A1 - Quinoxalines useful as inhibitors of protein kinases

Quinoxalines useful as inhibitors of protein kinases Download PDF

Info

Publication number: CA2548172A1
Authority: CA; Canada
Prior art keywords: compound; phenyl; optionally substituted; nitrogen; sulfur
Prior art date: 2003-12-04
Legal status : Abandoned

Application number

CA002548172A

Other languages

English (en)

French (fr)

Inventor

Guy W. Bemis

John P. Duffy

Current Assignee

Vertex Pharmaceuticals Inc

Original Assignee

Individual

Priority date

2003-12-04

Filing date

2004-12-03

Publication date

2005-06-23

2004-12-03 Application filed by Individual filed Critical Individual

2005-06-23 Publication of CA2548172A1 publication Critical patent/CA2548172A1/en

Status Abandoned legal-status Critical Current

Links

239000003112 inhibitor Substances 0.000 title abstract description 23
102000001253 Protein Kinase Human genes 0.000 title abstract description 8
108060006633 protein kinase Proteins 0.000 title abstract description 8
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150000001875 compounds Chemical class 0.000 claims abstract description 185
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229910052760 oxygen Inorganic materials 0.000 claims description 68
229910052717 sulfur Chemical group 0.000 claims description 63
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239000011593 sulfur Chemical group 0.000 claims description 59
125000005842 heteroatom Chemical group 0.000 claims description 56
QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims description 54
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