CA1081241A - Process for the preparation of phosphonous acids - Google Patents

Process for the preparation of phosphonous acids

Info

Publication number
CA1081241A
CA1081241A CA278,750A CA278750A CA1081241A CA 1081241 A CA1081241 A CA 1081241A CA 278750 A CA278750 A CA 278750A CA 1081241 A CA1081241 A CA 1081241A
Authority
CA
Canada
Prior art keywords
acid
formula
amino
hydrogen
give
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA278,750A
Other languages
English (en)
French (fr)
Inventor
Eric K. Baylis
John G. Dingwall
Colin D. Campbell
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Application granted granted Critical
Publication of CA1081241A publication Critical patent/CA1081241A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/48—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
CA278,750A 1976-05-21 1977-05-19 Process for the preparation of phosphonous acids Expired CA1081241A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB21000/76A GB1542938A (en) 1976-05-21 1976-05-21 Aminophosphonous acids and processes for their preparation

Publications (1)

Publication Number Publication Date
CA1081241A true CA1081241A (en) 1980-07-08

Family

ID=10155485

Family Applications (1)

Application Number Title Priority Date Filing Date
CA278,750A Expired CA1081241A (en) 1976-05-21 1977-05-19 Process for the preparation of phosphonous acids

Country Status (29)

Country Link
US (1) US4147780A (en, 2012)
JP (1) JPS52151128A (en, 2012)
AR (2) AR219077A1 (en, 2012)
AT (1) AT350585B (en, 2012)
AU (1) AU516592B2 (en, 2012)
BE (1) BE854843A (en, 2012)
BG (2) BG28070A4 (en, 2012)
CA (1) CA1081241A (en, 2012)
CS (1) CS202066B2 (en, 2012)
DD (1) DD131751A5 (en, 2012)
DE (1) DE2722162A1 (en, 2012)
DK (1) DK221477A (en, 2012)
EG (1) EG12688A (en, 2012)
ES (1) ES458931A1 (en, 2012)
FI (1) FI771602A7 (en, 2012)
FR (1) FR2360601A1 (en, 2012)
GB (1) GB1542938A (en, 2012)
IE (1) IE44904B1 (en, 2012)
IL (1) IL52127A0 (en, 2012)
NL (1) NL7705602A (en, 2012)
NO (1) NO771770L (en, 2012)
NZ (1) NZ184166A (en, 2012)
OA (1) OA05666A (en, 2012)
PH (1) PH14170A (en, 2012)
PL (2) PL110527B1 (en, 2012)
PT (1) PT66581B (en, 2012)
SE (1) SE7705886L (en, 2012)
SU (2) SU805948A3 (en, 2012)
ZA (1) ZA773017B (en, 2012)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2861609D1 (en) * 1977-11-19 1982-03-11 Ciba Geigy Ag Methods of inhibiting plant and combating weeds using alpha-aminoalkanephosphonous acids
EP0002039A1 (en) * 1977-11-19 1979-05-30 Ciba-Geigy Ag Phosphonous acid derivatives, processes for their preparation and their use in combating microorganisms
IL61985A0 (en) * 1980-02-01 1981-02-27 Sparamedica Ag Phosphinic and phosphonic acid derivatives,their manufacture and pharmaceutical compositions containing them
US4473561A (en) * 1981-04-17 1984-09-25 Sumitomo Chemical Company, Limited Fungicidal composition comprising alpha-substituted ethylphosphinic acids or their salts
US4466913A (en) * 1981-06-30 1984-08-21 Maiji Seika Kaisha Ltd. Phosphorus-containing compounds and process for producing the same
US4477391A (en) * 1981-08-14 1984-10-16 Collins James F Amino acid isomers, their production and their medicinal use
SE455259B (sv) * 1984-01-30 1988-07-04 Kenogard Ab Anvendning av vissa aminoalkanfosfonsyror for bekempning av svampsjukdomar hos vexter
US5189030A (en) * 1985-06-11 1993-02-23 Ciba-Geigy Corporation 1-amino-2-phenylethanephosphonic acids as microbiocides
US5143908A (en) * 1986-11-05 1992-09-01 Merck & Co., Inc. Antibacterial agents and potentiators of carbapenem antibiotics
US5099063A (en) * 1986-11-05 1992-03-24 Merck & Co., Inc. Certain phosphinic acid derivatives having antibacterial activity
US4761405A (en) * 1987-03-04 1988-08-02 Nova Pharmaceutical Corporation Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency
JPS6413097A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Phosphonic acid derivative
US5041644A (en) * 1987-07-06 1991-08-20 Merck & Co., Inc. Peptide derivatives of β-chloro-L(Z)-dehydro-glutamic acid
US5030732A (en) * 1988-03-03 1991-07-09 Merck & Co., Inc. Aminoethylphosphinic acid derivatives
US4962097A (en) * 1988-10-28 1990-10-09 Merck & Co., Inc. Method of treating bacterial infection with phosphorus containing DHP enzyme inhibitors
US5145990A (en) * 1988-10-28 1992-09-08 Merck & Co., Inc. Phosphorous containing dhp enzyme inhibitors
US5147867A (en) * 1988-10-28 1992-09-15 Merck & Co., Inc. Phosphorus containing enzyme inhibitors
US5179173A (en) * 1991-04-10 1993-01-12 Nalco Chemical Company Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom
FI963390A7 (fi) * 1996-08-30 1998-03-01 Khomutov Radii M Kasvinsuojeluaineet
IT201600098005A1 (it) * 2016-09-29 2018-03-29 Univ Degli Studi Roma La Sapienza Analoghi e derivati di amminoacidi dicarbossilici come antibatterici

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3160632A (en) * 1961-01-30 1964-12-08 Stauffer Chemical Co Aminomethylenephosphinic acids, salts thereof, and process for their production
CH475287A (de) * 1965-10-27 1969-07-15 Monsanto Co Verfahren zur Herstellung von substituierten Aminomethylphosphinsäuren
US3424788A (en) * 1967-07-24 1969-01-28 Armour & Co Aminophosphinic acids and salts useful as bacteriostats

Also Published As

Publication number Publication date
DK221477A (da) 1977-11-22
IE44904L (en) 1977-11-21
PL106608B1 (pl) 1980-01-31
PL198267A1 (pl) 1978-03-13
AR222464A1 (es) 1981-05-29
BG27905A3 (bg) 1980-01-15
DE2722162A1 (de) 1977-12-01
BG28070A4 (bg) 1980-02-25
PL110527B1 (en) 1980-07-31
FR2360601B1 (en, 2012) 1979-09-07
AU516592B2 (en) 1981-06-11
PT66581B (en) 1978-10-20
JPS52151128A (en) 1977-12-15
EG12688A (en) 1979-06-30
CS202066B2 (en) 1980-12-31
US4147780A (en) 1979-04-03
DD131751A5 (de) 1978-07-19
GB1542938A (en) 1979-03-28
AR219077A1 (es) 1980-07-31
SU805948A3 (ru) 1981-02-15
BE854843A (fr) 1977-11-21
IL52127A0 (en) 1977-07-31
ZA773017B (en) 1978-04-26
AU2531977A (en) 1978-11-23
FI771602A7 (en, 2012) 1977-11-22
ES458931A1 (es) 1978-03-01
PT66581A (en) 1977-06-01
SU795484A3 (ru) 1981-01-07
AT350585B (de) 1979-06-11
SE7705886L (sv) 1977-11-22
PH14170A (en) 1981-03-19
OA05666A (fr) 1981-05-31
FR2360601A1 (fr) 1978-03-03
IE44904B1 (en) 1982-05-05
NO771770L (no) 1977-11-22
NZ184166A (en) 1980-03-05
NL7705602A (nl) 1977-11-23
ATA361777A (de) 1978-11-15

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