CA1066709A - Preparation of loweralkyl imidazole carboxylates - Google Patents

Preparation of loweralkyl imidazole carboxylates

Info

Publication number
CA1066709A
CA1066709A CA245,697A CA245697A CA1066709A CA 1066709 A CA1066709 A CA 1066709A CA 245697 A CA245697 A CA 245697A CA 1066709 A CA1066709 A CA 1066709A
Authority
CA
Canada
Prior art keywords
imidazole
phenylethyl
acid
carboxylate
carboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA245,697A
Other languages
English (en)
French (fr)
Inventor
Walter A.M. Helsen
Leopold Fr. C. Roevens
Jozef J.P. Heykants
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Application granted granted Critical
Publication of CA1066709A publication Critical patent/CA1066709A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA245,697A 1975-03-10 1976-02-13 Preparation of loweralkyl imidazole carboxylates Expired CA1066709A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55719475A 1975-03-10 1975-03-10

Publications (1)

Publication Number Publication Date
CA1066709A true CA1066709A (en) 1979-11-20

Family

ID=24224401

Family Applications (1)

Application Number Title Priority Date Filing Date
CA245,697A Expired CA1066709A (en) 1975-03-10 1976-02-13 Preparation of loweralkyl imidazole carboxylates

Country Status (27)

Country Link
JP (1) JPS51115473A (no)
AT (1) AT353262B (no)
AU (1) AU503733B2 (no)
BE (1) BE839120A (no)
BG (1) BG24806A3 (no)
CA (1) CA1066709A (no)
CH (1) CH629192A5 (no)
CS (1) CS203116B2 (no)
DE (1) DE2609573A1 (no)
DK (1) DK99376A (no)
ES (1) ES445450A1 (no)
FI (1) FI62292C (no)
FR (1) FR2318159A1 (no)
GB (1) GB1535566A (no)
HU (1) HU172026B (no)
IE (1) IE42652B1 (no)
IL (1) IL49190A (no)
IT (1) IT1057941B (no)
LU (1) LU74503A1 (no)
NL (1) NL7602444A (no)
NO (1) NO144884C (no)
PL (1) PL99926B1 (no)
PT (1) PT64879B (no)
SE (1) SE7601959L (no)
SU (1) SU677656A3 (no)
YU (1) YU60876A (no)
ZA (1) ZA761427B (no)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9156825B2 (en) 2012-01-13 2015-10-13 The General Hospital Corporation Anesthetic compounds and related methods of use
US9181197B2 (en) 2008-03-31 2015-11-10 The General Hospital Corporation Etomidate analogues with improved pharmacokinetic and pharmacodynamic properties

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE871675A (fr) * 1977-12-02 1979-04-30 Smithkline Corp Procede de preparation de derives de l'imidazole
JPS5671073A (en) 1979-11-12 1981-06-13 Takeda Chem Ind Ltd Imidazole derivative
JPS5671074A (en) 1979-11-12 1981-06-13 Takeda Chem Ind Ltd 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative
JPS58157768A (ja) * 1982-03-16 1983-09-19 Takeda Chem Ind Ltd 4−クロロ−2−フエニルイミダゾ−ル−5−酢酸誘導体
PL149675B1 (pl) * 1986-03-10 1990-03-31 Sposób wytwarzania nowych pochodnych kwasu 1-metyl0-1h-imidaz0l0karb0ksyl0weg0-5

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9181197B2 (en) 2008-03-31 2015-11-10 The General Hospital Corporation Etomidate analogues with improved pharmacokinetic and pharmacodynamic properties
US9156825B2 (en) 2012-01-13 2015-10-13 The General Hospital Corporation Anesthetic compounds and related methods of use
US9522136B2 (en) 2012-01-13 2016-12-20 The General Hospital Corporation Anesthetic compounds and related methods of use
US9820971B2 (en) 2012-01-13 2017-11-21 The General Hospital Corporation Anesthetic compounds and related methods of use
US10154991B2 (en) 2012-01-13 2018-12-18 Annovation Biopharma, Inc. Anesthetic compounds and related methods of use

Also Published As

Publication number Publication date
JPS51115473A (en) 1976-10-12
YU60876A (en) 1983-01-21
ZA761427B (en) 1977-10-26
ES445450A1 (es) 1977-10-16
BG24806A3 (en) 1978-05-12
DE2609573A1 (de) 1976-09-30
SU677656A3 (ru) 1979-07-30
CS203116B2 (en) 1981-02-27
PT64879A (en) 1976-04-01
NO144884C (no) 1981-12-02
AU503733B2 (en) 1979-09-20
AT353262B (de) 1979-11-12
BE839120A (nl) 1976-09-03
FR2318159A1 (fr) 1977-02-11
AU1180676A (en) 1977-09-15
NL7602444A (nl) 1976-09-14
GB1535566A (en) 1978-12-13
HU172026B (hu) 1978-05-28
SE7601959L (sv) 1976-09-13
LU74503A1 (no) 1976-09-01
DK99376A (da) 1976-09-11
CH629192A5 (en) 1982-04-15
PT64879B (en) 1978-02-06
NO760790L (no) 1976-09-13
ATA171776A (de) 1979-04-15
FI62292B (fi) 1982-08-31
IL49190A (en) 1980-07-31
FR2318159B1 (no) 1979-07-27
IE42652L (en) 1976-09-10
PL99926B1 (pl) 1978-08-31
IL49190A0 (en) 1976-05-31
FI62292C (fi) 1982-12-10
IE42652B1 (en) 1980-09-24
IT1057941B (it) 1982-03-30
NO144884B (no) 1981-08-24
FI760601A (no) 1976-09-11

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