CA1049009A - 6h-thieno (3,2-f)-s-triazolo (4,3-a)-(1,4) diazepines - Google Patents

6h-thieno (3,2-f)-s-triazolo (4,3-a)-(1,4) diazepines

Info

Publication number
CA1049009A
CA1049009A CA74191917A CA191917A CA1049009A CA 1049009 A CA1049009 A CA 1049009A CA 74191917 A CA74191917 A CA 74191917A CA 191917 A CA191917 A CA 191917A CA 1049009 A CA1049009 A CA 1049009A
Authority
CA
Canada
Prior art keywords
group
chloro
diazepine
thieno
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA74191917A
Other languages
English (en)
French (fr)
Inventor
Joseph Hellerbach
Otto Hromatka
Paul Zeller
Dieter Binder
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Application granted granted Critical
Publication of CA1049009A publication Critical patent/CA1049009A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/36—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
CA74191917A 1973-02-08 1974-02-06 6h-thieno (3,2-f)-s-triazolo (4,3-a)-(1,4) diazepines Expired CA1049009A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH179973A CH584223A5 (xx) 1973-02-08 1973-02-08

Publications (1)

Publication Number Publication Date
CA1049009A true CA1049009A (en) 1979-02-20

Family

ID=4218866

Family Applications (1)

Application Number Title Priority Date Filing Date
CA74191917A Expired CA1049009A (en) 1973-02-08 1974-02-06 6h-thieno (3,2-f)-s-triazolo (4,3-a)-(1,4) diazepines

Country Status (24)

Country Link
JP (1) JPS5833234B2 (xx)
AR (2) AR203188A1 (xx)
AT (1) AT343118B (xx)
BE (1) BE810705A (xx)
CA (1) CA1049009A (xx)
CH (1) CH584223A5 (xx)
DD (1) DD112454A5 (xx)
DE (1) DE2405682C3 (xx)
DK (1) DK137679B (xx)
FI (1) FI58129C (xx)
FR (1) FR2217007B1 (xx)
GB (2) GB1456161A (xx)
HU (2) HU173741B (xx)
IE (1) IE38883B1 (xx)
IL (1) IL44095A (xx)
LU (1) LU69338A1 (xx)
NL (1) NL174045C (xx)
NO (1) NO142260C (xx)
PH (1) PH12303A (xx)
PL (3) PL97304B1 (xx)
SE (1) SE416399B (xx)
SU (3) SU715028A3 (xx)
YU (1) YU39716B (xx)
ZA (1) ZA74472B (xx)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT338799B (de) * 1974-03-02 1977-09-12 Boehringer Sohn Ingelheim Verfahren zur herstellung neuer substituierter 6-aryl-4h-s-triazolo-(3,4c)-thieno-(2,3e)-1,4-diazepine und ihrer salze
DE2531678C3 (de) * 1975-07-16 1979-06-28 C.H. Boehringer Sohn, 6507 Ingelheim Thieno [2,3e] triazole [3,4c] 5,6-dihydro-l,4diazepine und Verfahren zu ihrer Herstellung
DE2533924C3 (de) * 1975-07-30 1979-05-03 C.H. Boehringer Sohn, 6507 Ingelheim Verfahren zur Herstellung von 6- Aryl-4H-striazolo [3,4-c] thieno [2,3-e] 1,4-diazepinen
DE2708121A1 (de) * 1977-02-25 1978-09-07 Boehringer Sohn Ingelheim Triazolo-thieno-diazepin-l-one, verfahren zu ihrer herstellung und arzneimittel
FI63033C (fi) * 1977-07-21 1983-04-11 Boehringer Sohn Ingelheim Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner
DE3502392A1 (de) * 1985-01-25 1986-07-31 Boehringer Ingelheim KG, 6507 Ingelheim Neue thieno-triazolo-1,4-diazepino-2- carbonsaeureamide, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
ES2037013T3 (es) * 1986-01-21 1993-06-16 Boehringer Ingelheim Kg Procedimiento para preparar tieno-1,4-diazepinas.
JP2582225B2 (ja) * 1994-04-15 1997-02-19 ナショナル住宅産業株式会社 建 具
WO1995032963A1 (fr) * 1994-06-01 1995-12-07 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thienylazole et compose de thienotriazolodiazepine
ATE230600T1 (de) * 1995-09-09 2003-01-15 Hoffmann La Roche Verwendung eines thienotriazoldiazepins zur erhöhung des apolopoproteins a-i niveaus

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904641A (en) * 1971-06-18 1975-09-09 Yoshitomi Pharmaceutical Triazolothienodiazepine compounds

Also Published As

Publication number Publication date
YU22874A (en) 1982-06-30
AR203188A1 (es) 1975-08-22
ATA96474A (de) 1977-09-15
IE38883B1 (en) 1978-06-21
BE810705A (fr) 1974-08-07
AU6485574A (en) 1975-07-24
DE2405682A1 (de) 1974-08-15
FR2217007B1 (xx) 1978-02-03
CH584223A5 (xx) 1977-01-31
NL7401117A (xx) 1974-08-12
GB1456161A (en) 1976-11-17
PL97275B1 (pl) 1978-02-28
NO740405L (no) 1974-08-09
SU715028A3 (ru) 1980-02-05
DE2405682C3 (de) 1981-03-12
DE2405682B2 (de) 1980-07-17
JPS5833234B2 (ja) 1983-07-18
AR217034A1 (es) 1980-02-29
PH12303A (en) 1979-01-16
HU173741B (hu) 1979-08-28
FR2217007A1 (xx) 1974-09-06
AT343118B (de) 1978-05-10
ZA74472B (en) 1974-11-27
FI58129C (fi) 1980-12-10
DK137679C (xx) 1978-09-25
IL44095A0 (en) 1974-05-16
FI58129B (fi) 1980-08-29
SU1060115A3 (ru) 1983-12-07
SE416399B (sv) 1980-12-22
JPS49102698A (xx) 1974-09-27
IL44095A (en) 1979-03-12
PL97304B1 (pl) 1978-02-28
NO142260C (no) 1980-07-23
NL174045B (nl) 1983-11-16
LU69338A1 (xx) 1975-12-09
DD112454A5 (xx) 1975-04-12
DK137679B (da) 1978-04-17
NL174045C (nl) 1984-04-16
SU747429A4 (ru) 1980-07-23
PL96107B1 (pl) 1977-12-31
GB1456162A (en) 1976-11-17
IE38883L (en) 1974-08-08
HU170423B (xx) 1977-06-28
YU39716B (en) 1985-04-30
NO142260B (no) 1980-04-14

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