BRPI1011192A2 - derivados de carboxamida e ureia aromáticas substituídas como ligantes de receptor de vaniloide, composição farmacêutica, uso e processo para preparação dos referidos derivados - Google Patents

derivados de carboxamida e ureia aromáticas substituídas como ligantes de receptor de vaniloide, composição farmacêutica, uso e processo para preparação dos referidos derivados

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Publication number
BRPI1011192A2
BRPI1011192A2 BRPI1011192A BRPI1011192A BRPI1011192A2 BR PI1011192 A2 BRPI1011192 A2 BR PI1011192A2 BR PI1011192 A BRPI1011192 A BR PI1011192A BR PI1011192 A BRPI1011192 A BR PI1011192A BR PI1011192 A2 BRPI1011192 A2 BR PI1011192A2
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BR
Brazil
Prior art keywords
derivatives
preparing
pharmaceutical composition
substituted aromatic
receptor ligands
Prior art date
Application number
BRPI1011192A
Other languages
English (en)
Inventor
Bernhard Lesch
Gregor Bahrenberg
Jean De Vry
Jeewoo Lee
Klaus Schiene
Myeong-Seop Kim
Nils Damann
Robert Frank
Sven Frormann
Thomas Christoph
Young-Soo Kim
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of BRPI1011192A2 publication Critical patent/BRPI1011192A2/pt

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    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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BRPI1011192A 2009-05-07 2010-05-06 derivados de carboxamida e ureia aromáticas substituídas como ligantes de receptor de vaniloide, composição farmacêutica, uso e processo para preparação dos referidos derivados BRPI1011192A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17627709P 2009-05-07 2009-05-07
EP09006221 2009-05-07
PCT/EP2010/002785 WO2010127855A1 (en) 2009-05-07 2010-05-06 Substituted aromatic carboxamide and urea derivatives as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
BRPI1011192A2 true BRPI1011192A2 (pt) 2016-03-15

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ID=40848721

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Application Number Title Priority Date Filing Date
BRPI1011192A BRPI1011192A2 (pt) 2009-05-07 2010-05-06 derivados de carboxamida e ureia aromáticas substituídas como ligantes de receptor de vaniloide, composição farmacêutica, uso e processo para preparação dos referidos derivados

Country Status (16)

Country Link
US (1) US8334315B2 (pt)
EP (1) EP2427436B1 (pt)
JP (1) JP5767631B2 (pt)
AR (1) AR076753A1 (pt)
AU (1) AU2010244684B2 (pt)
BR (1) BRPI1011192A2 (pt)
CA (1) CA2758289A1 (pt)
DK (1) DK2427436T3 (pt)
ES (1) ES2402805T3 (pt)
HR (1) HRP20130128T1 (pt)
MX (1) MX2011011800A (pt)
PL (1) PL2427436T3 (pt)
PT (1) PT2427436E (pt)
SI (1) SI2427436T1 (pt)
TW (1) TWI504589B (pt)
WO (1) WO2010127855A1 (pt)

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KR20140091042A (ko) 2011-11-09 2014-07-18 그뤼넨탈 게엠베하 바닐로이드 수용체 리간드로서의 co-함유 그룹으로 치환된 페닐 모이어티를 갖는 치환된 피라졸릴계 카복스아미드 및 우레아 유도체들
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BR112014010957A2 (pt) 2011-11-09 2017-06-06 Gruenenthal Gmbh derivados de ureia e carboxamida com base em pirazolila substituída transportando uma porção de fenila substituída por um grupo contendo n como ligantes de receptor de vaniloide
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