BRPI1010147A2 - processo para preparar um composto, uso de um processo e uso de um catalisador de irídio - Google Patents

processo para preparar um composto, uso de um processo e uso de um catalisador de irídio

Info

Publication number
BRPI1010147A2
BRPI1010147A2 BRPI1010147A BRPI1010147A BRPI1010147A2 BR PI1010147 A2 BRPI1010147 A2 BR PI1010147A2 BR PI1010147 A BRPI1010147 A BR PI1010147A BR PI1010147 A BRPI1010147 A BR PI1010147A BR PI1010147 A2 BRPI1010147 A2 BR PI1010147A2
Authority
BR
Brazil
Prior art keywords
preparing
compound
iridium catalyst
iridium
catalyst
Prior art date
Application number
BRPI1010147A
Other languages
English (en)
Inventor
Gazic Smilovic Ivana
Casar Zdenko
Original Assignee
Lek Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP09163227A external-priority patent/EP2270019A1/en
Priority claimed from EP09166475A external-priority patent/EP2280016A1/en
Application filed by Lek Pharmaceuticals filed Critical Lek Pharmaceuticals
Publication of BRPI1010147A2 publication Critical patent/BRPI1010147A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BRPI1010147A 2009-06-19 2010-06-18 processo para preparar um composto, uso de um processo e uso de um catalisador de irídio BRPI1010147A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP09163227A EP2270019A1 (en) 2009-06-19 2009-06-19 New synthetic route for the preparation of alpha-amino boronic esters
EP09166475A EP2280016A1 (en) 2009-07-27 2009-07-27 New synthetic route for the preparation of alpha-amino boronic esters via substituted alk-1-ynes
EP09180099 2009-12-21
PCT/EP2010/058672 WO2010146176A2 (en) 2009-06-19 2010-06-18 Process for hydrogenation of halogenoalkenes without dehalogenation

Publications (1)

Publication Number Publication Date
BRPI1010147A2 true BRPI1010147A2 (pt) 2019-09-24

Family

ID=42711772

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1010147A BRPI1010147A2 (pt) 2009-06-19 2010-06-18 processo para preparar um composto, uso de um processo e uso de um catalisador de irídio

Country Status (8)

Country Link
US (2) US8785674B2 (pt)
EP (2) EP2443129B1 (pt)
JP (2) JP2012530116A (pt)
CN (1) CN102803271B (pt)
AU (1) AU2010261710A1 (pt)
BR (1) BRPI1010147A2 (pt)
CA (1) CA2765811C (pt)
WO (2) WO2010146176A2 (pt)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ598172A (en) * 2004-03-30 2013-08-30 Millennium Pharm Inc Synthesis of boronic ester and acid compounds
CA2765811C (en) * 2009-06-19 2018-06-05 Lek Pharmaceuticals D.D. Process for hydrogenation of halogenoalkenes without dehalogenation
US9505787B2 (en) 2012-09-11 2016-11-29 Cipla Limited Process for preparing of bortezomib
EP2969202A4 (en) 2013-03-11 2016-11-30 Univ Rutgers METAL ORGANO CATALYSIS FOR ASYMMETRIC CONVERSIONS
ZA201402789B (en) 2013-04-16 2015-11-25 Cipla Ltd Process for the preparation of bortezomib mannitol ester
EP2857405A1 (en) * 2013-10-01 2015-04-08 Studiengesellschaft Kohle mbH Process for the trans-selective hydroboration of internal alkynes
CN104529881B (zh) * 2014-12-08 2017-04-12 苏州施亚生物科技有限公司 一种2‑氯‑5‑乙基吡啶的制备方法
EP3288952A4 (en) * 2015-04-30 2018-10-10 The U.S.A. As Represented By The Secretary, Department Of Health And Human Services Organotrifluoroborate mimics of amino acids and uses thereof
CN106432309B (zh) * 2015-08-12 2020-04-10 南京江原安迪科正电子研究发展有限公司 一种类α-氨基酸的三氟化硼化合物的制备方法
SI3364958T1 (sl) * 2015-10-23 2023-05-31 Navitor Pharmaceuticals, Inc. Modulatorji interakcije sestrina in gator2 ter njihova uporaba
ES3040534T3 (en) 2017-04-26 2025-11-03 Navitor Pharm Inc Modulator of sestrin-gator2 interaction for use in the treatment of treatment-resistant depression
CA3117336A1 (en) 2018-10-24 2020-04-30 Navitor Pharmaceuticals, Inc. Polymorphs of (s)-2-amino-5,5-difluoro-4,4-dimethylpentanoic acid for use in modulating mtorc1
CN111689993B (zh) * 2019-03-11 2023-04-14 凯特立斯（深圳）科技有限公司 一种新的含硼类佐米药物关键中间体手性α-氨基硼酸酯的制备方法
CN114423739B (zh) * 2019-09-25 2024-06-25 拜耳公司 在手性铱催化剂和添加剂的存在下4-取代的1,2-二氢喹啉的改进的对映选择性氢化
IL292612A (en) 2019-11-01 2022-07-01 Navitor Pharm Inc Treatment methods using mtorc1 modulator
CN110776527A (zh) * 2019-12-02 2020-02-11 山东铂源药业有限公司 一种硼替佐米中间体的制备方法
JP7758028B2 (ja) * 2021-03-05 2025-10-22 Ａｇｃ株式会社 化合物、化合物の製造方法及び表面処理剤の製造方法
CN114669333B (zh) * 2022-04-25 2023-06-23 中山大学 一种催化α-季碳醛脱羰氢化的催化剂体系和催化方法
CN117362142B (zh) * 2023-10-09 2025-12-26 奥锐特药业股份有限公司 环己烯衍生物的不对称催化氢化方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8314001D0 (en) * 1983-05-20 1983-06-29 Shell Int Research Preparation of alphahaloalkyl esters
EP0315574A3 (de) 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin-Inhibitoren
US4924026A (en) 1989-08-11 1990-05-08 International Flavors & Fragrances Inc. Triisobutylene alcohols and esters, uses thereof in perfumery and halogenated intermediates useful for preparing same
JP3407379B2 (ja) * 1993-06-10 2003-05-19 ダイキン工業株式会社 １，１，１，３，３−ペンタフルオロプロパンの製造方法
US6083903A (en) 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
US5637782A (en) * 1994-12-02 1997-06-10 Uop Process for the selective saturation of olefin-containing halogenated organic streams
US5874634A (en) * 1995-03-02 1999-02-23 Nissan Chemical Industries, Ltd. Substituted cyclopentene derivatives and method for preparing the same
JPH08259477A (ja) * 1995-03-27 1996-10-08 Daikin Ind Ltd １，１，１，３，３−ペンタフルオロプロペンの製造方法及び１，１，１，３，３−ペンタフルオロプロパンの製造方法
US7122627B2 (en) 1999-07-26 2006-10-17 Bristol-Myers Squibb Company Lactam inhibitors of Hepatitis C virus NS3 protease
WO2002045834A2 (en) * 2000-12-04 2002-06-13 University Of New Orleans Research And Technology Foundation, Inc.(A Louisiana, Us, Corporation) 'metal complexes for hydrogenation of unsaturated compounds'
NZ598172A (en) * 2004-03-30 2013-08-30 Millennium Pharm Inc Synthesis of boronic ester and acid compounds
US20070244319A1 (en) 2006-04-18 2007-10-18 Boaz Neil W Metallocenyl P-N ligands, preparation thereof, and use for asymmetric catalysis
WO2009004350A1 (en) * 2007-07-03 2009-01-08 Pliva Hrvatska D.O.O. Methods for preparing bortezomib and intermediates used in its manufacture
WO2009006473A2 (en) 2007-07-05 2009-01-08 Trustees Of Tufts College Pro-soft polypeptide proteasome inhibitors, and methods of use thereof
KR20100051828A (ko) 2007-09-12 2010-05-18 닥터 레디스 레보러터리즈 리미티드 보르테조밉 및 그의 제조방법
CA2765811C (en) * 2009-06-19 2018-06-05 Lek Pharmaceuticals D.D. Process for hydrogenation of halogenoalkenes without dehalogenation

Also Published As

Publication number Publication date
WO2010146176A3 (en) 2011-02-24
US8785674B2 (en) 2014-07-22
CA2765811C (en) 2018-06-05
JP2012530116A (ja) 2012-11-29
WO2010146172A2 (en) 2010-12-23
EP2443128A2 (en) 2012-04-25
CN102803271B (zh) 2016-03-23
JP2012530115A (ja) 2012-11-29
WO2010146172A3 (en) 2012-02-23
US9315525B2 (en) 2016-04-19
CA2765811A1 (en) 2010-12-23
WO2010146176A2 (en) 2010-12-23
EP2443129B1 (en) 2016-11-23
EP2443129A2 (en) 2012-04-25
EP2443128B1 (en) 2017-12-20
US20120220794A1 (en) 2012-08-30
CN102803271A (zh) 2012-11-28
AU2010261710A1 (en) 2012-01-19
US20120231993A1 (en) 2012-09-13

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Legal Events

Date Code Title Description
B08F Application fees: dismissal - article 86 of industrial property law
B08K Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87)

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.