BR112013010768A2 - derivados de ureia e carboxamida substituídos por heteroaromáticos como ligantes dos receptores vaniloides - Google Patents

derivados de ureia e carboxamida substituídos por heteroaromáticos como ligantes dos receptores vaniloides

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Publication number
BR112013010768A2
BR112013010768A2 BR112013010768A BR112013010768A BR112013010768A2 BR 112013010768 A2 BR112013010768 A2 BR 112013010768A2 BR 112013010768 A BR112013010768 A BR 112013010768A BR 112013010768 A BR112013010768 A BR 112013010768A BR 112013010768 A2 BR112013010768 A2 BR 112013010768A2
Authority
BR
Brazil
Prior art keywords
receptor ligands
vanilloid receptor
substituted urea
carboxamide derivatives
heteroaromatic substituted
Prior art date
Application number
BR112013010768A
Other languages
English (en)
Inventor
Bernhard Lesch
Jeewoo Lee
Robert Frank
Thomas Christoph
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of BR112013010768A2 publication Critical patent/BR112013010768A2/pt

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Child & Adolescent Psychology (AREA)
BR112013010768A 2010-11-10 2011-11-09 derivados de ureia e carboxamida substituídos por heteroaromáticos como ligantes dos receptores vaniloides BR112013010768A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP10014449 2010-11-10
PCT/EP2011/005628 WO2012062462A1 (en) 2010-11-10 2011-11-09 Substituted heteroaromatic carboxamide and urea derivatives as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
BR112013010768A2 true BR112013010768A2 (pt) 2016-07-12

Family

ID=43501425

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013010768A BR112013010768A2 (pt) 2010-11-10 2011-11-09 derivados de ureia e carboxamida substituídos por heteroaromáticos como ligantes dos receptores vaniloides

Country Status (10)

Country Link
US (1) US20120115903A1 (pt)
EP (1) EP2638034A1 (pt)
JP (1) JP2013545740A (pt)
AR (1) AR083817A1 (pt)
AU (1) AU2011328520A1 (pt)
BR (1) BR112013010768A2 (pt)
CA (1) CA2816769A1 (pt)
MX (1) MX2013005008A (pt)
TW (1) TW201305139A (pt)
WO (1) WO2012062462A1 (pt)

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US20120115903A1 (en) 2012-05-10
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