BR9900442A - Derivados de 11-acetil-12,13dioxabiciclo[8.2.1] tridecenona, processos para a sua preparação e medicamentos contendo estes compostos. - Google Patents

Derivados de 11-acetil-12,13dioxabiciclo[8.2.1] tridecenona, processos para a sua preparação e medicamentos contendo estes compostos.

Info

Publication number
BR9900442A
BR9900442A BR9900442-9A BR9900442A BR9900442A BR 9900442 A BR9900442 A BR 9900442A BR 9900442 A BR9900442 A BR 9900442A BR 9900442 A BR9900442 A BR 9900442A
Authority
BR
Brazil
Prior art keywords
derivatives
preparation
tridecenone
acetyl
compounds
Prior art date
Application number
BR9900442-9A
Other languages
English (en)
Inventor
Daniel Jasserand
Ulf Preuschoff
Christian Eeckhout
Original Assignee
Solvay Pharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Gmbh filed Critical Solvay Pharm Gmbh
Publication of BR9900442A publication Critical patent/BR9900442A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Nutrition Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

Patente de Invenção: <B>"DERIVADOS DE 11-ACETIL-12,13-DIOXABICICLO[8.2.1]TRIDECENONA, PROCESSOS PARA A SUA PREPARAçãO E MEDICAMENTOS CONTENDO ESTES COMPOSTOS"<D>. A presente invenção descreve derivados de N-desmetil-N-isopropil-eritromicina A com cadeia lateral modificada e propriedades agonísticas da motilina com ação gastrintestinal e respectiva preparação.
BR9900442-9A 1998-02-13 1999-02-10 Derivados de 11-acetil-12,13dioxabiciclo[8.2.1] tridecenona, processos para a sua preparação e medicamentos contendo estes compostos. BR9900442A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19805822A DE19805822B4 (de) 1998-02-13 1998-02-13 11-Acetyl-12,13-dioxabicyclo[8.2.1]tridecenon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
BR9900442A true BR9900442A (pt) 2000-05-02

Family

ID=7857548

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9900442-9A BR9900442A (pt) 1998-02-13 1999-02-10 Derivados de 11-acetil-12,13dioxabiciclo[8.2.1] tridecenona, processos para a sua preparação e medicamentos contendo estes compostos.

Country Status (26)

Country Link
EP (1) EP0937734B1 (pt)
JP (1) JPH11269193A (pt)
KR (1) KR100584017B1 (pt)
CN (1) CN1189473C (pt)
AR (1) AR014320A1 (pt)
AT (1) ATE486083T1 (pt)
AU (1) AU748670B2 (pt)
BR (1) BR9900442A (pt)
CA (1) CA2260315C (pt)
CZ (1) CZ294879B6 (pt)
DE (2) DE19805822B4 (pt)
DZ (1) DZ2721A1 (pt)
ES (1) ES2355187T3 (pt)
HK (1) HK1023575A1 (pt)
HU (1) HU222539B1 (pt)
ID (1) ID21968A (pt)
IL (1) IL128238A (pt)
NO (1) NO310917B1 (pt)
NZ (1) NZ334087A (pt)
PL (1) PL192281B1 (pt)
RU (1) RU2218346C2 (pt)
SK (1) SK285313B6 (pt)
TR (1) TR199900285A3 (pt)
TW (1) TW579379B (pt)
UA (1) UA57030C2 (pt)
ZA (1) ZA99678B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1489090E (pt) * 2000-08-17 2006-05-31 Kitasato Inst Novos derivados de pseudoeritromicina
GB0611907D0 (en) 2006-06-15 2006-07-26 Glaxo Group Ltd Compounds
JP2009501199A (ja) 2005-07-12 2009-01-15 グラクソ グループ リミテッド Ｇｐｒ３８アゴニストとしてのピペラジンヘテロアリール誘導体
KR101281435B1 (ko) 2005-07-26 2013-07-02 글락소 그룹 리미티드 벤질피페라진 유도체 및 그의 의학적 용도
CA2655540A1 (en) 2006-06-28 2008-01-03 Glaxo Group Limited Piperazinyl derivatives useful in the treatment of gpr38 receptor mediated diseases
MX2011008857A (es) 2009-02-27 2011-09-30 Raqualia Pharma Inc Derivados de oxiindol con actividad agonistica del receptor de motilina.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5106961A (en) * 1987-05-26 1992-04-21 Eli Lilly And Company Erythromycin ring-contracted derivatives
US4920102A (en) * 1988-04-18 1990-04-24 Eli Lilly And Company Method for treating gastrointestinal disorders
NZ232375A (en) * 1989-02-09 1992-04-28 Lilly Co Eli Insulin analogues modified at b29
DE4200145A1 (de) * 1992-01-07 1993-07-08 Kali Chemie Pharma Gmbh 7,10-epoxy-oxacyclododecan-derivate, verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US5712253A (en) * 1996-06-18 1998-01-27 Abbott Laboratories Macrocyclic 13-membered ring derivatives of erythromycins A and B

Also Published As

Publication number Publication date
ES2355187T3 (es) 2011-03-23
HUP9900263A2 (hu) 1999-09-28
KR19990072345A (ko) 1999-09-27
HU9900263D0 (en) 1999-04-28
DE19805822A1 (de) 1999-08-19
CZ294879B6 (cs) 2005-04-13
IL128238A (en) 2001-09-13
ZA99678B (en) 1999-07-28
AR014320A1 (es) 2001-02-07
AU748670B2 (en) 2002-06-06
AU1643899A (en) 1999-08-26
SK285313B6 (sk) 2006-10-05
PL331444A1 (en) 1999-08-16
CA2260315C (en) 2008-04-08
TW579379B (en) 2004-03-11
HU222539B1 (hu) 2003-08-28
NO310917B1 (no) 2001-09-17
DZ2721A1 (fr) 2003-09-01
ATE486083T1 (de) 2010-11-15
ID21968A (id) 1999-08-19
IL128238A0 (en) 1999-11-30
CZ45899A3 (cs) 1999-09-15
TR199900285A2 (xx) 1999-09-21
EP0937734A1 (de) 1999-08-25
EP0937734B1 (de) 2010-10-27
SK15099A3 (en) 2000-01-18
TR199900285A3 (tr) 1999-09-21
RU2218346C2 (ru) 2003-12-10
HUP9900263A3 (en) 2000-04-28
NZ334087A (en) 2000-07-28
PL192281B1 (pl) 2006-09-29
NO990675D0 (no) 1999-02-12
CN1189473C (zh) 2005-02-16
HK1023575A1 (en) 2000-09-15
UA57030C2 (uk) 2003-06-16
NO990675L (no) 1999-08-16
CA2260315A1 (en) 1999-08-13
CN1239718A (zh) 1999-12-29
KR100584017B1 (ko) 2006-05-30
DE59915209D1 (de) 2010-12-09
DE19805822B4 (de) 2009-02-05
JPH11269193A (ja) 1999-10-05

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO DE ACORDO COM O ART. 8O DA LPI.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.