BR9404410A - Processo para preparação de amidinas bicíclicas, amidinas bicíclicas, 3-amino-2,3,4,5,6,7,8-hexaidropirrolo(1,2-a)-pirimidina, 3-(aminometilo-2,5,6,7-tetraidro-3H-pirrolo-(1,2-a)imidazol e 3-(aminometilo)-3-metilo-2,3,4,6,7,8-hexaidropirrolo(1,2-1)pirimidina - Google Patents

Processo para preparação de amidinas bicíclicas, amidinas bicíclicas, 3-amino-2,3,4,5,6,7,8-hexaidropirrolo(1,2-a)-pirimidina, 3-(aminometilo-2,5,6,7-tetraidro-3H-pirrolo-(1,2-a)imidazol e 3-(aminometilo)-3-metilo-2,3,4,6,7,8-hexaidropirrolo(1,2-1)pirimidina

Info

Publication number
BR9404410A
BR9404410A BR9404410A BR9404410A BR9404410A BR 9404410 A BR9404410 A BR 9404410A BR 9404410 A BR9404410 A BR 9404410A BR 9404410 A BR9404410 A BR 9404410A BR 9404410 A BR9404410 A BR 9404410A
Authority
BR
Brazil
Prior art keywords
aminomethyl
pyrimidine
amino
bicyclic amidines
hexahydropyrrolo
Prior art date
Application number
BR9404410A
Other languages
English (en)
Inventor
Oleg Werbitzky
Ulrich Daum
Rachel Bregy
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4254820&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9404410(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of BR9404410A publication Critical patent/BR9404410A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polyurethanes Or Polyureas (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Adhesives Or Adhesive Processes (AREA)
BR9404410A 1993-11-11 1994-11-10 Processo para preparação de amidinas bicíclicas, amidinas bicíclicas, 3-amino-2,3,4,5,6,7,8-hexaidropirrolo(1,2-a)-pirimidina, 3-(aminometilo-2,5,6,7-tetraidro-3H-pirrolo-(1,2-a)imidazol e 3-(aminometilo)-3-metilo-2,3,4,6,7,8-hexaidropirrolo(1,2-1)pirimidina BR9404410A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH338593 1993-11-11

Publications (1)

Publication Number Publication Date
BR9404410A true BR9404410A (pt) 1995-06-20

Family

ID=4254820

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9404410A BR9404410A (pt) 1993-11-11 1994-11-10 Processo para preparação de amidinas bicíclicas, amidinas bicíclicas, 3-amino-2,3,4,5,6,7,8-hexaidropirrolo(1,2-a)-pirimidina, 3-(aminometilo-2,5,6,7-tetraidro-3H-pirrolo-(1,2-a)imidazol e 3-(aminometilo)-3-metilo-2,3,4,6,7,8-hexaidropirrolo(1,2-1)pirimidina

Country Status (15)

Country Link
US (4) US5723605A (pt)
EP (2) EP0869127B1 (pt)
JP (1) JP4348747B2 (pt)
KR (1) KR100362543B1 (pt)
CN (2) CN1042227C (pt)
AT (2) ATE175969T1 (pt)
BR (1) BR9404410A (pt)
CA (1) CA2134009C (pt)
CZ (1) CZ286335B6 (pt)
DE (2) DE59409907D1 (pt)
DK (2) DK0869127T3 (pt)
ES (2) ES2128490T5 (pt)
PT (1) PT869127E (pt)
RU (1) RU2132850C1 (pt)
SI (2) SI0662476T1 (pt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19752935A1 (de) * 1997-11-28 1999-06-02 Basf Ag Verfahren zur Herstellung von bicyclischen Amidinen, Diazacycloalkene und ein Verfahren zu deren Herstellung
WO2004032861A2 (en) * 2002-10-11 2004-04-22 Bristol-Myers Squibb Company Hexahydro-benzimidazolone compounds useful as anti-inflammatory agents
JP2008515505A (ja) 2004-10-07 2008-05-15 ノボ・ノルデイスク・エー／エス 疾病の自己管理のための方法とシステム
US8430879B2 (en) * 2007-03-22 2013-04-30 Sonoma Orthopedic Products, Inc. Segmented intramedullary structure
WO2009027248A1 (de) * 2007-08-29 2009-03-05 Basf Se Verfahren zur herstellung von aminen aus glycerin
US10383580B2 (en) 2012-12-31 2019-08-20 Abbott Diabetes Care Inc. Analysis of glucose median, variability, and hypoglycemia risk for therapy guidance
US9085712B2 (en) 2013-03-14 2015-07-21 Bayer Materialscience Llc Fast cure aspartate polysiloxane hybrid coating
EP3543270A1 (de) 2018-03-23 2019-09-25 Covestro Deutschland AG Katalysatorsystem für uretdiondispersionen
WO2019180128A1 (de) 2018-03-23 2019-09-26 Covestro Deutschland Ag Wässrige uretdiongruppenhaltige zusammensetzungen und verfahren zu deren herstellung
EP3572446A1 (de) 2018-05-24 2019-11-27 Evonik Degussa GmbH Reaktive mischung von uretdionen und katalysatoren
EP3916032A1 (de) 2020-05-29 2021-12-01 Covestro Deutschland AG Bei niedrigen temperaturen vernetzende uretdiongruppen enthaltende zusammensetzungen
IT202100005336A1 (it) 2021-03-08 2022-09-08 Versalis Spa Metodo per la preparazione di amidine.
EP4305023A1 (en) 2021-03-08 2024-01-17 Versalis S.p.A. Method for preparation of amidines
IT202200018231A1 (it) 2022-09-07 2024-03-07 Versalis Spa Metodo per la preparazione di amidine da n-(alchil lattami)

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA628948A (en) * 1961-10-10 Rohm And Haas Company Condensed heterocyclic compounds
DE730182C (de) * 1939-08-22 1943-01-07 Ig Farbenindustrie Ag Verfahren zur Herstellung von N-(Aminoalkyl)-pyrrolidonen
US2993047A (en) * 1958-03-03 1961-07-18 Rohm & Haas Condensed heterocyclic compounds
US2957885A (en) * 1958-05-14 1960-10-25 Rohm & Haas Aminosubstituted heterocyclic compounds
US2984665A (en) * 1958-05-14 1961-05-16 Rohm & Haas Condensed heterocyclic compounds
US2993049A (en) * 1958-06-18 1961-07-18 Rohm & Haas Aminomethyl-substituted condensed heterocyclic compounds
CH471804A (de) * 1965-09-09 1969-04-30 Bayer Ag Verfahren zur Herstellung von Bicyclischen Amidinen
FR1542058A (fr) * 1966-10-29 1968-10-11 San Abbott Ltd Procédé de préparation de polyuréthanes à partir d'isocyanates et de polyols à l'aide de diazabicycloalkènes comme catalyseurs
GB1182014A (en) * 1966-10-29 1970-02-25 San Abbott Ltd Urethane and Urea Catalyst
US3761436A (en) * 1969-08-19 1973-09-25 San Abbott Ltd Catalytic conversion of aminoalkyl lactams to diazabicycloalkenes
GB1327467A (en) * 1970-10-12 1973-08-22 Merck & Co Inc Pharmaceutical compositions for inhibiting indoleamine- n-methyl transferase
US3845071A (en) * 1973-03-12 1974-10-29 Richardson Merrell Inc Imidazo(1,2-a)azacycloalkanes
US4126685A (en) * 1975-01-31 1978-11-21 Imperial Chemical Industries Limited 6-Aryl-pyrrolo[1,2,9]imidazole derivatives which possess anti-hypertensive activity
US4507481A (en) * 1983-07-29 1985-03-26 Pennwalt Corporation Pyrrolo[1,2-a]imidazoles and imidazo[1,2-a]pyridines
EP0199483A1 (en) * 1985-04-09 1986-10-29 San-Apro K.K. Amidines and a method of manufacturing the same
IE60275B1 (en) * 1987-06-19 1994-06-29 Loctite Ireland Ltd Diazabicyclo and triazabicyclo primer compositions and use thereof in bonding non-polar substrates
JPH0491121A (ja) * 1990-08-07 1992-03-24 Toshiba Chem Corp 封止用樹脂組成物及び半導体封止装置
JPH0496923A (ja) * 1990-08-14 1992-03-30 Toshiba Chem Corp 封止用樹脂組成物及び半導体封止装置
JPH0496930A (ja) * 1990-08-14 1992-03-30 Toshiba Chem Corp 封止用樹脂組成物及び半導体封止装置
JPH04106120A (ja) * 1990-08-24 1992-04-08 Toshiba Chem Corp 封止用樹脂組成物及び半導体封止装置
JPH04120127A (ja) * 1990-09-11 1992-04-21 Toshiba Chem Corp 封止用樹脂組成物及び半導体封止装置

Also Published As

Publication number Publication date
CA2134009A1 (en) 1995-05-12
EP0869127B1 (de) 2001-10-10
EP0662476B2 (de) 2002-08-14
RU94040173A (ru) 1996-10-10
CN1106406A (zh) 1995-08-09
US5922869A (en) 1999-07-13
US20020028939A1 (en) 2002-03-07
CN1042227C (zh) 1999-02-24
DK0662476T3 (da) 1999-09-13
DK0662476T4 (da) 2002-10-07
DK0869127T3 (da) 2001-12-03
EP0662476B1 (de) 1999-01-20
KR950014113A (ko) 1995-06-15
ES2128490T5 (es) 2003-02-01
ES2165114T3 (es) 2002-03-01
CN1070861C (zh) 2001-09-12
CZ286335B6 (cs) 2000-03-15
CN1215727A (zh) 1999-05-05
ATE175969T1 (de) 1999-02-15
ES2128490T3 (es) 1999-05-16
US5723605A (en) 1998-03-03
SI0662476T1 (en) 1999-04-30
US6255488B1 (en) 2001-07-03
RU2132850C1 (ru) 1999-07-10
EP0662476A1 (de) 1995-07-12
DE59409907D1 (de) 2001-11-15
SI0869127T1 (pt) 2001-12-31
JP4348747B2 (ja) 2009-10-21
US6476175B2 (en) 2002-11-05
PT869127E (pt) 2002-03-28
CZ276894A3 (en) 1995-07-12
KR100362543B1 (ko) 2003-02-05
EP0869127A1 (de) 1998-10-07
DE59407697D1 (de) 1999-03-04
CA2134009C (en) 2005-03-08
JPH07188235A (ja) 1995-07-25
ATE206711T1 (de) 2001-10-15

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Legal Events

Date Code Title Description
EE Request for examination
FB36 Technical and formal requirements: requirement - article 36 of industrial property law
FF Decision: intention to grant
FG9A Patent or certificate of addition granted
B24H Lapse because of non-payment of annual fees (definitively: art 78 iv lpi)
B24F Patent annual fee: publication cancelled

Free format text: ANULADA A PUBLICACAO CODIGO 24.8 NA RPI NO 2277 DE 26/08/2014 POR TER SIDO INDEVIDA.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE AS 16A, 17A, 18A, 19A E 20A ANUIDADES.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2606 DE 15-12-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.