BR0211612A - Cristais que incluem um sal de ácido málico de n-[2-(dietilamino)etil]-5-[(5-flúor2-oxo-3h-indol-3-ilide no)metil]-2,4-dimetil-1h-pirrol-3-carboxamida, processos para a sua preparação e suas composições - Google Patents

Cristais que incluem um sal de ácido málico de n-[2-(dietilamino)etil]-5-[(5-flúor2-oxo-3h-indol-3-ilide no)metil]-2,4-dimetil-1h-pirrol-3-carboxamida, processos para a sua preparação e suas composições

Info

Publication number
BR0211612A
BR0211612A BR0211612-0A BR0211612A BR0211612A BR 0211612 A BR0211612 A BR 0211612A BR 0211612 A BR0211612 A BR 0211612A BR 0211612 A BR0211612 A BR 0211612A
Authority
BR
Brazil
Prior art keywords
indol
carboxamide
oxo
dimethyl
compositions
Prior art date
Application number
BR0211612-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Michael Hawley
Thomas J Fleck
Stephen P Prescott
Mark T Maloney
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23211067&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0211612(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BR0211612A publication Critical patent/BR0211612A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
BR0211612-0A 2001-08-15 2002-08-13 Cristais que incluem um sal de ácido málico de n-[2-(dietilamino)etil]-5-[(5-flúor2-oxo-3h-indol-3-ilide no)metil]-2,4-dimetil-1h-pirrol-3-carboxamida, processos para a sua preparação e suas composições BR0211612A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31235301P 2001-08-15 2001-08-15
PCT/US2002/025649 WO2003016305A1 (en) 2001-08-15 2002-08-13 Crystals including a malic acid salt of n-[2-(diethylamino) ethyl]-5-[(5-fluoro-2-oxo-3h-indole-3-ylidene) methyl]-2, 4-dimethyl-1h-pyrrole-3-carboxamide, processes for its preparation and compositions thereof

Publications (1)

Publication Number Publication Date
BR0211612A true BR0211612A (pt) 2004-08-24

Family

ID=23211067

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0211612-0A BR0211612A (pt) 2001-08-15 2002-08-13 Cristais que incluem um sal de ácido málico de n-[2-(dietilamino)etil]-5-[(5-flúor2-oxo-3h-indol-3-ilide no)metil]-2,4-dimetil-1h-pirrol-3-carboxamida, processos para a sua preparação e suas composições

Country Status (42)

Country Link
US (2) US20030069298A1 (cg-RX-API-DMAC7.html)
EP (3) EP1419151B1 (cg-RX-API-DMAC7.html)
JP (1) JP4159988B2 (cg-RX-API-DMAC7.html)
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CN (2) CN100439360C (cg-RX-API-DMAC7.html)
AP (1) AP1660A (cg-RX-API-DMAC7.html)
AR (1) AR036261A1 (cg-RX-API-DMAC7.html)
AU (1) AU2002324684B2 (cg-RX-API-DMAC7.html)
BG (1) BG108553A (cg-RX-API-DMAC7.html)
BR (1) BR0211612A (cg-RX-API-DMAC7.html)
CA (1) CA2455050C (cg-RX-API-DMAC7.html)
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SI (2) SI1419151T1 (cg-RX-API-DMAC7.html)
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UA (1) UA76483C2 (cg-RX-API-DMAC7.html)
WO (1) WO2003016305A1 (cg-RX-API-DMAC7.html)
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PL216524B1 (pl) 2014-04-30
HK1066542A1 (en) 2005-03-24
HRP20040112A2 (en) 2004-06-30
SI1419151T1 (sl) 2014-04-30
KR100639281B1 (ko) 2006-10-31
RS10304A (sr) 2007-02-05
BG108553A (bg) 2005-04-30
EP3168218B1 (en) 2018-11-14
EP2332934A1 (en) 2011-06-15
MA27058A1 (fr) 2004-12-20
TNSN04028A1 (fr) 2006-06-01
AU2002324684B2 (en) 2006-10-05
MY139383A (en) 2009-09-30
JP2005503386A (ja) 2005-02-03
ES2705063T3 (es) 2019-03-21
PT1419151E (pt) 2014-03-27
GEP20063777B (en) 2006-03-27
OA12650A (en) 2006-06-19
HK1088008A1 (zh) 2006-10-27
ES2623094T3 (es) 2017-07-10
SK902004A3 (sk) 2005-03-04
EA006445B1 (ru) 2005-12-29
EP2332934B1 (en) 2017-03-01
CU20040029A7 (es) 2008-03-14
CN100364991C (zh) 2008-01-30
HU229206B1 (en) 2013-09-30
CU23713B7 (es) 2011-10-05
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TR201900509T4 (tr) 2019-02-21
JP4159988B2 (ja) 2008-10-01
US20070191458A1 (en) 2007-08-16
CN100439360C (zh) 2008-12-03
WO2003016305A1 (en) 2003-02-27
CA2455050C (en) 2007-02-20
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