BR0115580A - Derivados de 3-aroilindol e a utilizaçao dos mesmos como agonistas dos receptores cb2 - Google Patents

Derivados de 3-aroilindol e a utilizaçao dos mesmos como agonistas dos receptores cb2

Info

Publication number
BR0115580A
BR0115580A BR0115580-6A BR0115580A BR0115580A BR 0115580 A BR0115580 A BR 0115580A BR 0115580 A BR0115580 A BR 0115580A BR 0115580 A BR0115580 A BR 0115580A
Authority
BR
Brazil
Prior art keywords
receptor agonists
derivatives
aroylindole
compounds
aroilindol
Prior art date
Application number
BR0115580-6A
Other languages
English (en)
Inventor
Francis Barth
Christian Congy
Carole Guillaumont
Murielle Rinaldi
Fabienne Vasse
Claude Vernhet
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of BR0115580A publication Critical patent/BR0115580A/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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Abstract

"DERIVADOS DE 3-AROILINDOL E A UTILIZAçãO DOS MESMOS COMO AGONISTAS DOS RECEPTORES CB2". Derivados de 3-aroilindol e a utilização dos mesmos como agonistas dos receptores CB~ 2~. A presente invenção refere-se aos compostos de fórmula: (I) assim como a respectiva preparação e as composições farmacêuticas que os contêm. Esses compostos são agonistas dos receptores aos canabinóides CB~ 2~.
BR0115580-6A 2000-11-22 2001-11-21 Derivados de 3-aroilindol e a utilizaçao dos mesmos como agonistas dos receptores cb2 BR0115580A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0015158A FR2816938B1 (fr) 2000-11-22 2000-11-22 Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant
PCT/FR2001/003665 WO2002042269A1 (fr) 2000-11-22 2001-11-21 Derives de 3-aroylindole et leur utilisation en tant qu'agonistes des recepteurs cb2

Publications (1)

Publication Number Publication Date
BR0115580A true BR0115580A (pt) 2003-09-09

Family

ID=8856819

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0115580-6A BR0115580A (pt) 2000-11-22 2001-11-21 Derivados de 3-aroilindol e a utilizaçao dos mesmos como agonistas dos receptores cb2

Country Status (32)

Country Link
US (1) US6995184B2 (pt)
EP (1) EP1339679B1 (pt)
JP (1) JP4264258B2 (pt)
KR (1) KR20030048161A (pt)
CN (1) CN1234688C (pt)
AR (1) AR033594A1 (pt)
AT (1) ATE301638T1 (pt)
AU (1) AU2002222001A1 (pt)
BG (1) BG107827A (pt)
BR (1) BR0115580A (pt)
CA (1) CA2427444A1 (pt)
CZ (1) CZ20031392A3 (pt)
DE (1) DE60112607T2 (pt)
DK (1) DK1339679T3 (pt)
DZ (1) DZ3443A1 (pt)
EA (1) EA005854B1 (pt)
EE (1) EE200300244A (pt)
ES (1) ES2247201T3 (pt)
FR (1) FR2816938B1 (pt)
HR (1) HRP20030417A2 (pt)
HU (1) HUP0400561A2 (pt)
IL (1) IL155634A0 (pt)
IS (1) IS6802A (pt)
MA (1) MA26959A1 (pt)
MX (1) MXPA03004549A (pt)
NO (1) NO20031952L (pt)
NZ (1) NZ525609A (pt)
PL (1) PL362276A1 (pt)
SK (1) SK6042003A3 (pt)
TW (1) TWI224592B (pt)
WO (1) WO2002042269A1 (pt)
ZA (1) ZA200303728B (pt)

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JP4667867B2 (ja) 2002-08-02 2011-04-13 メルク・シャープ・エンド・ドーム・コーポレイション 置換フロ［２，３−ｂ］ピリジン誘導体
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FR2847899B1 (fr) 2002-11-29 2006-04-28 Sanofi Synthelabo Derives d'indole-3-carboxamide, leur preparation et leur application en therapeutique
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EA011307B1 (ru) 2004-07-12 2009-02-27 Кадила Хелзкэр Лимитед Трициклические производные пиразола в качестве модуляторов каннабиноидного рецептора
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PA8854001A1 (es) 2008-12-16 2010-07-27 Abbott Lab Compuestos novedosos como ligandos de receptores de canabinoides
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FR2816938A1 (fr) 2002-05-24

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