BR0114913A - Inibidores de metaloproteinase de espiro-pirimidina-2,4,6-triona - Google Patents
Inibidores de metaloproteinase de espiro-pirimidina-2,4,6-trionaInfo
- Publication number
- BR0114913A BR0114913A BR0114913-0A BR0114913A BR0114913A BR 0114913 A BR0114913 A BR 0114913A BR 0114913 A BR0114913 A BR 0114913A BR 0114913 A BR0114913 A BR 0114913A
- Authority
- BR
- Brazil
- Prior art keywords
- spiro
- pyrimidine
- metalloproteinase inhibitors
- trione metalloproteinase
- trione
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Ophthalmology & Optometry (AREA)
- Cardiology (AREA)
- Pregnancy & Childbirth (AREA)
- Virology (AREA)
- Vascular Medicine (AREA)
- Psychology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24338900P | 2000-10-26 | 2000-10-26 | |
| PCT/IB2001/001986 WO2002034753A2 (fr) | 2000-10-26 | 2001-10-23 | Inhibiteurs de metalloproteinase spiro-pyrimidine-2,4,6-trione |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0114913A true BR0114913A (pt) | 2003-07-01 |
Family
ID=22918584
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0114913-0A BR0114913A (pt) | 2000-10-26 | 2001-10-23 | Inibidores de metaloproteinase de espiro-pirimidina-2,4,6-triona |
Country Status (32)
| Country | Link |
|---|---|
| EP (1) | EP1332146A2 (fr) |
| JP (1) | JP2004518635A (fr) |
| KR (1) | KR20040004412A (fr) |
| CN (1) | CN1501937A (fr) |
| AP (1) | AP2001002318A0 (fr) |
| AR (1) | AR035069A1 (fr) |
| AU (1) | AU2002210813A1 (fr) |
| BG (1) | BG107653A (fr) |
| BR (1) | BR0114913A (fr) |
| CA (1) | CA2425283A1 (fr) |
| CZ (1) | CZ20031083A3 (fr) |
| EA (1) | EA005762B1 (fr) |
| EC (1) | ECSP034567A (fr) |
| EE (1) | EE200300196A (fr) |
| GT (1) | GT200100213A (fr) |
| HN (1) | HN2001000244A (fr) |
| HR (1) | HRP20030332A2 (fr) |
| HU (1) | HUP0301577A3 (fr) |
| IL (1) | IL154948A0 (fr) |
| IS (1) | IS6762A (fr) |
| MA (1) | MA26957A1 (fr) |
| MX (1) | MXPA03003735A (fr) |
| NO (1) | NO20031853L (fr) |
| OA (1) | OA12529A (fr) |
| PA (1) | PA8531401A1 (fr) |
| PE (1) | PE20020589A1 (fr) |
| PL (1) | PL366201A1 (fr) |
| SK (1) | SK4972003A3 (fr) |
| SV (1) | SV2003000705A (fr) |
| TN (1) | TNSN01149A1 (fr) |
| WO (1) | WO2002034753A2 (fr) |
| ZA (1) | ZA200302190B (fr) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DOP2002000333A (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz |
| BR0207865A (pt) | 2001-02-14 | 2004-03-23 | Warner Lambert Co | Benzotiadiazinas inibidores de metaloproteinases de matriz |
| DOP2002000332A (es) | 2001-02-14 | 2002-08-30 | Warner Lambert Co | Inhibidores de piridina de metaloproteinasas de la matriz |
| PA8539501A1 (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Compuestos triazolo como inhibidores de mmp |
| DOP2002000328A (es) | 2001-02-14 | 2003-08-30 | Warner Lambert Co | Pirimidinas inhibidoras de metaloproteinasas de matriz |
| US6924276B2 (en) | 2001-09-10 | 2005-08-02 | Warner-Lambert Company | Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors |
| US6962922B2 (en) | 2001-10-12 | 2005-11-08 | Warner-Lambert Company Llc | Alkynylated quinazoline compounds |
| BR0213233A (pt) | 2001-10-12 | 2005-01-04 | Warner Lambert Co | Alcinos inibidores de metaloproteinase de matriz |
| US6894057B2 (en) | 2002-03-08 | 2005-05-17 | Warner-Lambert Company | Oxo-azabicyclic compounds |
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| US3714093A (en) * | 1970-05-19 | 1973-01-30 | American Home Prod | Spiro [heterocycloalkyl-2'(1'h)-quinazoline]-4'(3'h)-ones |
| JP2002504916A (ja) * | 1997-06-21 | 2002-02-12 | ロシュ ダイアグノスティクス ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗転移及び抗腫瘍活性を有するバルビツール酸誘導体 |
| US6265578B1 (en) * | 1999-02-12 | 2001-07-24 | Hoffmann-La Roche Inc. | Pyrimidine-2,4,6-triones |
| HN2000000137A (es) * | 1999-08-12 | 2001-02-02 | Pfizer Prod Inc | Pirimidina-2,4,6-trionas inhibidores de metaloproteinasas |
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- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/fr not_active Application Discontinuation
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