EE200300196A - Spiropürimidiin-2,4,6-trioonmetalloproteinaasi inhibiitorid - Google Patents

Spiropürimidiin-2,4,6-trioonmetalloproteinaasi inhibiitorid

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Publication number
EE200300196A
EE200300196A EEP200300196A EEP200300196A EE200300196A EE 200300196 A EE200300196 A EE 200300196A EE P200300196 A EEP200300196 A EE P200300196A EE P200300196 A EEP200300196 A EE P200300196A EE 200300196 A EE200300196 A EE 200300196A
Authority
EE
Estonia
Prior art keywords
spiropyrimidine
metalloproteinase inhibitors
trione metalloproteinase
trione
inhibitors
Prior art date
Application number
EEP200300196A
Other languages
English (en)
Inventor
Scott Bronk Brian
Carl Noe Mark
James Wythes Martin
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200300196A publication Critical patent/EE200300196A/et

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
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  • Pulmonology (AREA)
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  • Tropical Medicine & Parasitology (AREA)
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EEP200300196A 2000-10-26 2001-10-23 Spiropürimidiin-2,4,6-trioonmetalloproteinaasi inhibiitorid EE200300196A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26
PCT/IB2001/001986 WO2002034753A2 (en) 2000-10-26 2001-10-23 Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors

Publications (1)

Publication Number Publication Date
EE200300196A true EE200300196A (et) 2003-10-15

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EEP200300196A EE200300196A (et) 2000-10-26 2001-10-23 Spiropürimidiin-2,4,6-trioonmetalloproteinaasi inhibiitorid

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EP (1) EP1332146A2 (et)
JP (1) JP2004518635A (et)
KR (1) KR20040004412A (et)
CN (1) CN1501937A (et)
AP (1) AP2001002318A0 (et)
AR (1) AR035069A1 (et)
AU (1) AU2002210813A1 (et)
BG (1) BG107653A (et)
BR (1) BR0114913A (et)
CA (1) CA2425283A1 (et)
CZ (1) CZ20031083A3 (et)
EA (1) EA005762B1 (et)
EC (1) ECSP034567A (et)
EE (1) EE200300196A (et)
GT (1) GT200100213A (et)
HN (1) HN2001000244A (et)
HR (1) HRP20030332A2 (et)
HU (1) HUP0301577A3 (et)
IL (1) IL154948A0 (et)
IS (1) IS6762A (et)
MA (1) MA26957A1 (et)
MX (1) MXPA03003735A (et)
NO (1) NO20031853L (et)
OA (1) OA12529A (et)
PA (1) PA8531401A1 (et)
PE (1) PE20020589A1 (et)
PL (1) PL366201A1 (et)
SK (1) SK4972003A3 (et)
SV (1) SV2003000705A (et)
TN (1) TNSN01149A1 (et)
WO (1) WO2002034753A2 (et)
ZA (1) ZA200302190B (et)

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ES2231708T3 (es) 2001-02-14 2005-05-16 Warner-Lambert Company Llc Benzotiadicinas inhibidoras de metaloproteinasa de matriz.
DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
EP1368323B1 (en) 2001-02-14 2010-06-30 Warner-Lambert Company LLC Pyrimidine matrix metalloproteinase inhibitors
PA8539501A1 (es) 2001-02-14 2002-09-30 Warner Lambert Co Compuestos triazolo como inhibidores de mmp
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
CA2462442A1 (en) 2001-10-12 2003-04-24 Warner-Lambert Company Llc Alkyne matrix metalloproteinase inhibitors
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
US6894057B2 (en) 2002-03-08 2005-05-17 Warner-Lambert Company Oxo-azabicyclic compounds
WO2003091252A1 (en) * 2002-04-25 2003-11-06 Bristol-Myers Squibb Company Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases
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